CA2786250A1 - Thiazolo[5,4-d] pyrimidines and their use as agrochemicals - Google Patents

Thiazolo[5,4-d] pyrimidines and their use as agrochemicals Download PDF

Info

Publication number
CA2786250A1
CA2786250A1 CA2786250A CA2786250A CA2786250A1 CA 2786250 A1 CA2786250 A1 CA 2786250A1 CA 2786250 A CA2786250 A CA 2786250A CA 2786250 A CA2786250 A CA 2786250A CA 2786250 A1 CA2786250 A1 CA 2786250A1
Authority
CA
Canada
Prior art keywords
compound
lower alkyl
spp
compounds
thiazolo
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA2786250A
Other languages
English (en)
French (fr)
Inventor
William Brewster
Carla Klittich
Brent Rieder
Thomas Siddall
Chenglin Yao
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Corteva Agriscience LLC
Original Assignee
Dow AgroSciences LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dow AgroSciences LLC filed Critical Dow AgroSciences LLC
Publication of CA2786250A1 publication Critical patent/CA2786250A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/429—Thiazoles condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Dentistry (AREA)
  • Environmental Sciences (AREA)
  • Zoology (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Wood Science & Technology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pretreatment Of Seeds And Plants (AREA)
  • Plural Heterocyclic Compounds (AREA)
CA2786250A 2010-01-07 2011-01-06 Thiazolo[5,4-d] pyrimidines and their use as agrochemicals Abandoned CA2786250A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US29301410P 2010-01-07 2010-01-07
US61/293,014 2010-01-07
PCT/US2011/020351 WO2011085084A1 (en) 2010-01-07 2011-01-06 THIAZOLO[5,4-d] PYRIMIDINES AND THEIR USE AS AGROCHEMICALS

Publications (1)

Publication Number Publication Date
CA2786250A1 true CA2786250A1 (en) 2011-07-14

Family

ID=44225056

Family Applications (1)

Application Number Title Priority Date Filing Date
CA2786250A Abandoned CA2786250A1 (en) 2010-01-07 2011-01-06 Thiazolo[5,4-d] pyrimidines and their use as agrochemicals

Country Status (18)

Country Link
US (1) US8921382B2 (forum.php)
EP (1) EP2521452B1 (forum.php)
JP (1) JP5781090B2 (forum.php)
KR (1) KR101814835B1 (forum.php)
CN (1) CN102791135B (forum.php)
BR (1) BR112012016866A2 (forum.php)
CA (1) CA2786250A1 (forum.php)
CL (1) CL2012001851A1 (forum.php)
CO (1) CO6612238A2 (forum.php)
ES (1) ES2529247T3 (forum.php)
IN (1) IN2012DN06323A (forum.php)
MX (1) MX2012007954A (forum.php)
PL (1) PL2521452T3 (forum.php)
PT (1) PT2521452E (forum.php)
RU (1) RU2547721C2 (forum.php)
UA (1) UA109780C2 (forum.php)
WO (1) WO2011085084A1 (forum.php)
ZA (1) ZA201204871B (forum.php)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN104945420A (zh) 2009-06-29 2015-09-30 因塞特公司 作为pi3k抑制剂的嘧啶酮类
CA2842190A1 (en) 2011-07-19 2013-01-24 Infinity Pharmaceuticals Inc. Heterocyclic compounds and uses thereof
WO2013031694A1 (ja) * 2011-08-26 2013-03-07 富山化学工業株式会社 アミン化合物またはその塩
TWI717002B (zh) 2011-09-02 2021-01-21 美商英塞特控股公司 作為pi3k抑制劑之雜環基胺
IN2014DN07224A (forum.php) 2012-02-03 2015-04-24 Basf Se
AR089884A1 (es) 2012-02-03 2014-09-24 Basf Se Compuestos fungicidas de pirimidina
WO2013135672A1 (en) 2012-03-13 2013-09-19 Basf Se Fungicidal pyrimidine compounds
AR090548A1 (es) 2012-04-02 2014-11-19 Incyte Corp Azaheterociclobencilaminas biciclicas como inhibidores de pi3k
CN103668956B (zh) * 2012-09-21 2015-08-12 上海韬鸿化工科技有限公司 防螨虫整理剂、织物的防螨虫整理方法及防螨虫织物
EP3409115A3 (en) * 2013-03-15 2019-02-27 The Regents of The University of California Methods for identifying arthropod repellents, and compounds and compositions identified by such methods
WO2015191677A1 (en) 2014-06-11 2015-12-17 Incyte Corporation Bicyclic heteroarylaminoalkyl phenyl derivatives as pi3k inhibitors
CN105594748A (zh) * 2014-10-15 2016-05-25 浙江新安化工集团股份有限公司 一种精准定向、高效的防治鳞翅目害虫的杀虫组合物及其使用方法
CN104391070B (zh) * 2014-12-05 2016-06-08 山东省城市供排水水质监测中心 一种水中烷基汞的检测方法
HRP20210036T1 (hr) 2015-02-27 2021-03-05 Incyte Corporation Soli inhibitora pi3k i postupci za njihovo dobivanje
EP3270692A4 (en) 2015-03-18 2019-02-13 The Regents of the University of California CHEMICALS FOR PROTECTION AGAINST BRANCHES
US9988401B2 (en) 2015-05-11 2018-06-05 Incyte Corporation Crystalline forms of a PI3K inhibitor
CN105606755A (zh) * 2016-01-30 2016-05-25 郭庆龙 一种胺苯吡唑酮残留量的gc-nci-ms测定方法
WO2018139560A1 (ja) 2017-01-26 2018-08-02 三井化学アグロ株式会社 ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤
US11147272B2 (en) 2017-04-10 2021-10-19 Mitsui Chemicals Argro, Inc. Pyridone compounds and agricultural and horticultural fungicides comprising the same as active ingredients
US11000038B2 (en) 2017-04-10 2021-05-11 Mitsui Chemicals Agro, Inc. Pyridone compounds and agricultural and horticultural fungicides containing the same as active ingredients
MY190386A (en) 2017-04-11 2022-04-20 Mitsui Chemicals Agro Inc Pyridone compounds and agricultural and horticultural fungicides containing the same as active ingredients
CA3066591A1 (en) 2017-06-08 2018-12-13 Mitsui Chemicals Agro, Inc. Pyridone compounds and agricultural and horticultural fungicides containing the same as active ingredients
MA52761A (fr) 2018-06-01 2021-04-14 Incyte Corp Schéma posologique destiné au traitement de troubles liés à la pi3k
CA3104048A1 (en) 2018-07-25 2020-01-30 Mitsui Chemicals Agro, Inc. Pyridone compounds and agricultural and horticultural fungicides containing the same as active ingredients
CA3165597A1 (en) 2020-02-11 2021-08-19 Stephane BIERI Method of controlling fungi with cyclothiazomycin c
CN112010848B (zh) * 2020-09-29 2021-12-24 南通大学 含三氟甲基吡啶联芳氧基结构的1,3,4-噁二唑类化合物的制备方法和应用
CN116250525B (zh) * 2023-03-08 2024-12-24 内蒙古民族大学 一种小型哺乳类剥制标本安全防腐剂及其制备方法

Family Cites Families (29)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3309359A (en) 1965-10-22 1967-03-14 Hoffmann La Roche N-mono-acyl-5-fluorocytosine derivatives and process
US3368938A (en) 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
US3868373A (en) 1970-01-27 1975-02-25 Hoffmann La Roche 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines
CH579057A5 (forum.php) 1973-09-07 1976-08-31 Hoffmann La Roche
FR2530636A1 (fr) * 1982-07-23 1984-01-27 Rhone Poulenc Agrochimie Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides
EP0139613A1 (de) 1983-08-29 1985-05-02 Ciba-Geigy Ag N-(2-Nitrophenyl)-4-aminopyrimidin-Derivate, deren Herstellung und Verwendung
US4845081A (en) 1984-10-18 1989-07-04 University Of Florida Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes
ES2057172T3 (es) 1988-03-09 1994-10-16 Ciba Geigy Ag Agente para la proteccion de plantas contra enfermedades.
DE3821711A1 (de) * 1988-06-28 1990-02-08 Bayer Ag Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
US5034393A (en) * 1989-07-27 1991-07-23 Dowelanco Fungicidal use of pyridopyrimidine, pteridine, pyrimidopyrimidine, pyrimidopyridazine, and pyrimido-1,2,4-triazine derivatives
JP3109012B2 (ja) * 1992-06-18 2000-11-13 クミアイ化学工業株式会社 チアゾロ［５，４−ｄ］ピリミジン誘導体及び農園芸用殺菌剤
JP3217191B2 (ja) * 1992-07-16 2001-10-09 ビーエーエスエフ アクチェンゲゼルシャフト ヘテロ芳香族化合物およびこれを含有する植物保護剤
US5326766A (en) 1992-08-19 1994-07-05 Dreikorn Barry A 4-(2-(4-(2-pyridinyloxy)phenyl)ethoxy)quinazoline and analogues thereof
BR9609613A (pt) 1995-07-05 1999-05-25 Du Pont Composto composição fungicida e método de controle de doenças de plantas
KR100482919B1 (ko) 1996-03-11 2005-10-12 신젠타 파티서페이션즈 아게 살충제로서의피리미딘-4-온유도체
HRP970239B1 (en) 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
US6448262B1 (en) * 1998-11-16 2002-09-10 American Cyanamid Company Pesticidal and parasiticidal use of 2-(substituted thio) thiazolo-[4,5-b]pyridine compounds
ES2280508T3 (es) * 2001-01-31 2007-09-16 Bayer Cropscience Ag Combinacion herbicida-agente fitoprotector basada en agentes fitoprotectores de carboxilato de isoxazolina.
WO2003018051A1 (en) 2001-08-27 2003-03-06 Vic Jira Anti-fungal composition
ES2284945T3 (es) * 2001-09-10 2007-11-16 Basf Aktiengesellschaft Compuestos pesticidas y parasiticidas de alqueno di y trifluorosustituido.
US20080269238A1 (en) * 2004-04-01 2008-10-30 Takeda Pharmaceutical Company Limited Thiazolopyrimidine Derivative
EP2078721B1 (en) 2005-10-21 2014-01-22 Dow AgroSciences LLC Thieno-pyrimidine compounds having fungicidal activity
WO2008005303A2 (en) 2006-06-30 2008-01-10 Janssen Pharmaceutica N.V. Thiazolopyrimidine modulators of trpv1
EP2562161A1 (en) 2008-01-22 2013-02-27 Dow AgroSciences LLC 5-fluoro pyrimidine derivatives as fungicides
CN102215691B (zh) 2008-08-01 2015-02-04 陶氏益农公司 5-氟胞嘧啶作为杀真菌剂的用途
EP2389375B1 (en) 2009-01-23 2015-05-20 Euro-Celtique S.A. Hydroxamic acid derivatives
CN101613362B (zh) * 2009-07-31 2011-11-16 南京工业大学 3-羰基-6-乙氧甲酰基-噻唑并嘧啶类化合物及其合成方法和用途
IN2012DN00692A (forum.php) 2009-08-07 2015-06-19 Dow Agroscience Llc

Also Published As

Publication number Publication date
JP2013516476A (ja) 2013-05-13
JP5781090B2 (ja) 2015-09-16
EP2521452A1 (en) 2012-11-14
WO2011085084A1 (en) 2011-07-14
RU2547721C2 (ru) 2015-04-10
US20110166164A1 (en) 2011-07-07
KR101814835B1 (ko) 2018-01-04
RU2012133570A (ru) 2014-02-20
CL2012001851A1 (es) 2012-12-14
PL2521452T3 (pl) 2015-05-29
BR112012016866A2 (pt) 2015-09-01
ES2529247T3 (es) 2015-02-18
IN2012DN06323A (forum.php) 2015-10-02
EP2521452B1 (en) 2014-12-24
UA109780C2 (uk) 2015-10-12
US8921382B2 (en) 2014-12-30
PT2521452E (pt) 2015-02-24
CN102791135B (zh) 2015-05-20
CN102791135A (zh) 2012-11-21
CO6612238A2 (es) 2013-02-01
KR20120115538A (ko) 2012-10-18
MX2012007954A (es) 2012-08-03
EP2521452A4 (en) 2013-07-03
HK1176236A1 (en) 2013-07-26
ZA201204871B (en) 2013-09-25

Similar Documents

Publication Publication Date Title
US9000162B2 (en) 5,8-difluoro-4-(2-(4-(heteroaryloxy)-phenyl)ethylamino)quinazolines and their use as agrochemicals
EP2521452B1 (en) THIAZOLO[5,4-d]PYRIMIDINES AND THEIR USE AS AGROCHEMICALS
US8895568B2 (en) Compositions comprising substituted pteridines as agrochemicals
AU2009351623B2 (en) Pteridines and their use as agrochemicals
AU2017228717B2 (en) Pesticidal compositions and related methods
TWI495431B (zh) 殺蟲組成物
CN103188936A (zh) 杀虫组合物
US20180116224A1 (en) Pesticidal compositions and related methods
US20180125074A1 (en) Pesticidal compositions and related methods
US20180125073A1 (en) Pesticidal compositions and related methods
US20130317068A1 (en) Substituted 1,2,4-triazole compounds as a seed treatment to control pests
WO2024147134A1 (en) Agrochemical composition, methods, use, and kits
US20130317069A1 (en) 2,4-(substituted aromatic)-1,3-oxazoline compounds as a seed treatment to control pests

Legal Events

Date Code Title Description
FZDE Dead

Effective date: 20170106