CA2775925A1 - Salts, solvates and pharmaceutical compositions of macrocyclic ghrelin receptor agonists and methods of using the same - Google Patents
Salts, solvates and pharmaceutical compositions of macrocyclic ghrelin receptor agonists and methods of using the same Download PDFInfo
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- CA2775925A1 CA2775925A1 CA2775925A CA2775925A CA2775925A1 CA 2775925 A1 CA2775925 A1 CA 2775925A1 CA 2775925 A CA2775925 A CA 2775925A CA 2775925 A CA2775925 A CA 2775925A CA 2775925 A1 CA2775925 A1 CA 2775925A1
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Classifications
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- A61K31/553—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one oxygen as ring hetero atoms, e.g. loxapine, staurosporine
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D269/00—Heterocyclic compounds containing rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms according to more than one of groups C07D261/00 - C07D267/00
Landscapes
- Health & Medical Sciences (AREA)
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- Cardiology (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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- Peptides Or Proteins (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US24736209P | 2009-09-30 | 2009-09-30 | |
| US61/247,362 | 2009-09-30 | ||
| PCT/US2010/050661 WO2011041369A1 (en) | 2009-09-30 | 2010-09-29 | Salts, solvates, and pharmaceutical compositions of macrocyclic ghrelin receptor agonists and methods of using the same |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2775925A1 true CA2775925A1 (en) | 2011-04-07 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA2775925A Abandoned CA2775925A1 (en) | 2009-09-30 | 2010-09-29 | Salts, solvates and pharmaceutical compositions of macrocyclic ghrelin receptor agonists and methods of using the same |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US20110245159A1 (https=) |
| EP (1) | EP2482813A4 (https=) |
| JP (1) | JP2013506676A (https=) |
| KR (1) | KR20120081166A (https=) |
| CN (1) | CN102781441A (https=) |
| AU (1) | AU2010300689A1 (https=) |
| BR (1) | BR112012007183A2 (https=) |
| CA (1) | CA2775925A1 (https=) |
| EA (1) | EA201270497A1 (https=) |
| IL (1) | IL218938A0 (https=) |
| IN (1) | IN2012DN03297A (https=) |
| MX (1) | MX2012003912A (https=) |
| WO (1) | WO2011041369A1 (https=) |
| ZA (1) | ZA201202307B (https=) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20090198050A1 (en) * | 2003-06-18 | 2009-08-06 | Tranzyme Pharma Inc. | Macrocyclic Modulators of the Ghrelin Receptor |
| US7491695B2 (en) * | 2003-06-18 | 2009-02-17 | Tranzyme Pharma Inc. | Methods of using macrocyclic modulators of the ghrelin receptor |
| US8921521B2 (en) | 2003-06-18 | 2014-12-30 | Ocera Therapeutics, Inc. | Macrocyclic modulators of the Ghrelin receptor |
| US7476653B2 (en) * | 2003-06-18 | 2009-01-13 | Tranzyme Pharma, Inc. | Macrocyclic modulators of the ghrelin receptor |
| DK1633774T3 (da) * | 2003-06-18 | 2010-05-25 | Tranzyme Pharma Inc | Makrocykliske motilinreceptorantagonister |
| US8592377B2 (en) | 2007-03-28 | 2013-11-26 | President And Fellows Of Harvard College | Stitched polypeptides |
| ES2711526T3 (es) | 2010-08-13 | 2019-05-06 | Aileron Therapeutics Inc | Macrociclos peptidomiméticos |
| UY34094A (es) | 2011-05-27 | 2013-01-03 | Novartis Ag | Derivados de la piperidina 3-espirocíclica como agonistas de receptores de la ghrelina |
| TW201806968A (zh) | 2011-10-18 | 2018-03-01 | 艾利倫治療公司 | 擬肽巨環化合物 |
| BR112014020103A2 (pt) | 2012-02-15 | 2018-10-09 | Aileron Therapeutics, Inc. | macrociclos peptidomiméticos |
| EP2819688A4 (en) | 2012-02-15 | 2015-10-28 | Aileron Therapeutics Inc | TRIAZOL AND THIOETHER-COUPLED PEPTIDOMIMETIC MACROCYCLES |
| WO2014071241A1 (en) | 2012-11-01 | 2014-05-08 | Aileron Therapeutics, Inc. | Disubstituted amino acids and methods of preparation and use thereof |
| EP3197478A4 (en) | 2014-09-24 | 2018-05-30 | Aileron Therapeutics, Inc. | Peptidomimetic macrocycles and uses thereof |
| CN107106636A (zh) | 2014-11-12 | 2017-08-29 | 利瑞克药品有限公司 | 肠内喂养不耐受的治疗 |
| WO2016154058A1 (en) | 2015-03-20 | 2016-09-29 | Aileron Therapeutics, Inc. | Peptidomimetic macrocycles and uses thereof |
| WO2018106945A1 (en) * | 2016-12-07 | 2018-06-14 | Progenity Inc. | Gastrointestinal tract detection methods, devices and systems |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7491695B2 (en) * | 2003-06-18 | 2009-02-17 | Tranzyme Pharma Inc. | Methods of using macrocyclic modulators of the ghrelin receptor |
| US7476653B2 (en) * | 2003-06-18 | 2009-01-13 | Tranzyme Pharma, Inc. | Macrocyclic modulators of the ghrelin receptor |
| AU2005280639A1 (en) * | 2004-02-17 | 2006-03-09 | Billy T. Fowler | Methods, compositions, and apparatuses for forming macrocyclic compounds |
| EP1723159B1 (en) * | 2004-02-27 | 2019-06-12 | Melinta Therapeutics, Inc. | Macrocyclic compounds and methods of making and using the same |
| US8088733B2 (en) * | 2006-07-06 | 2012-01-03 | Tranzyme Pharma Inc. | Methods of using macrocyclic agonists of the ghrelin receptor for treatment of gastrointestinal motility disorders |
-
2010
- 2010-09-29 IN IN3297DEN2012 patent/IN2012DN03297A/en unknown
- 2010-09-29 JP JP2012532258A patent/JP2013506676A/ja not_active Withdrawn
- 2010-09-29 BR BR112012007183A patent/BR112012007183A2/pt not_active IP Right Cessation
- 2010-09-29 AU AU2010300689A patent/AU2010300689A1/en not_active Abandoned
- 2010-09-29 KR KR1020127010634A patent/KR20120081166A/ko not_active Withdrawn
- 2010-09-29 CA CA2775925A patent/CA2775925A1/en not_active Abandoned
- 2010-09-29 US US12/937,040 patent/US20110245159A1/en not_active Abandoned
- 2010-09-29 CN CN2010800547916A patent/CN102781441A/zh active Pending
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- 2010-09-29 EP EP10821147A patent/EP2482813A4/en not_active Withdrawn
- 2010-09-29 WO PCT/US2010/050661 patent/WO2011041369A1/en not_active Ceased
-
2012
- 2012-03-29 ZA ZA2012/02307A patent/ZA201202307B/en unknown
- 2012-03-29 IL IL218938A patent/IL218938A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO2011041369A1 (en) | 2011-04-07 |
| EA201270497A1 (ru) | 2012-10-30 |
| KR20120081166A (ko) | 2012-07-18 |
| EP2482813A1 (en) | 2012-08-08 |
| MX2012003912A (es) | 2012-08-17 |
| ZA201202307B (en) | 2012-12-27 |
| JP2013506676A (ja) | 2013-02-28 |
| AU2010300689A1 (en) | 2012-04-19 |
| IL218938A0 (en) | 2012-07-31 |
| US20110245159A1 (en) | 2011-10-06 |
| IN2012DN03297A (https=) | 2015-10-23 |
| CN102781441A (zh) | 2012-11-14 |
| EP2482813A4 (en) | 2013-02-27 |
| BR112012007183A2 (pt) | 2017-06-20 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FZDE | Discontinued |
Effective date: 20131001 |