CA2768356A1 - Compositions comprising a cholinesterase inhibitor for treating cognitive disorders - Google Patents
Compositions comprising a cholinesterase inhibitor for treating cognitive disorders Download PDFInfo
- Publication number
- CA2768356A1 CA2768356A1 CA2768356A CA2768356A CA2768356A1 CA 2768356 A1 CA2768356 A1 CA 2768356A1 CA 2768356 A CA2768356 A CA 2768356A CA 2768356 A CA2768356 A CA 2768356A CA 2768356 A1 CA2768356 A1 CA 2768356A1
- Authority
- CA
- Canada
- Prior art keywords
- compound
- group
- atoms
- galantamine
- cholinesterase inhibitor
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
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- 229960003980 galantamine Drugs 0.000 claims description 37
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- ADEBPBSSDYVVLD-UHFFFAOYSA-N donepezil Chemical group O=C1C=2C=C(OC)C(OC)=CC=2CC1CC(CC1)CCN1CC1=CC=CC=C1 ADEBPBSSDYVVLD-UHFFFAOYSA-N 0.000 claims description 28
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- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
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- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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Landscapes
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- Chemical Kinetics & Catalysis (AREA)
- Psychiatry (AREA)
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- Hospice & Palliative Care (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Hydrogenated Pyridines (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
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| US22642509P | 2009-07-17 | 2009-07-17 | |
| US61/226,425 | 2009-07-17 | ||
| PCT/US2010/042308 WO2011009061A1 (en) | 2009-07-17 | 2010-07-16 | Compositions comprising a cholinesterase inhibitor for treating cognitive disorders |
Publications (1)
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| CA2768356A1 true CA2768356A1 (en) | 2011-01-20 |
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| CA2768356A Abandoned CA2768356A1 (en) | 2009-07-17 | 2010-07-16 | Compositions comprising a cholinesterase inhibitor for treating cognitive disorders |
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| US4166452A (en) | 1976-05-03 | 1979-09-04 | Generales Constantine D J Jr | Apparatus for testing human responses to stimuli |
| US4256108A (en) * | 1977-04-07 | 1981-03-17 | Alza Corporation | Microporous-semipermeable laminated osmotic system |
| US4265874A (en) * | 1980-04-25 | 1981-05-05 | Alza Corporation | Method of delivering drug with aid of effervescent activity generated in environment of use |
| US5409948A (en) * | 1992-11-23 | 1995-04-25 | The United States Of America As Represented By The Secretary Of The Department Of Health And Human Services | Method for treating cognitive disorders with phenserine |
| WO2005072713A2 (en) * | 2004-01-27 | 2005-08-11 | The Feinstein Institute For Medical Research | Cholinesterase inhibitors for treating inflammation |
| US20070212253A1 (en) * | 2004-12-21 | 2007-09-13 | Elrod Scott A | Descenting systems and methods |
| MX2007008955A (es) * | 2005-01-26 | 2007-09-18 | Allergan Inc | Amidas de acido 3-aril-3-hidroxi-2-amino-propionico, amidas de acido 3-heteeroaril-3-hidroxi-2-amino-propionico y compuestos relacionados que tienen actividad analgesica y/o inmunoestimulante. |
| CA2616858A1 (en) * | 2005-07-27 | 2007-02-01 | Carlos Henrique Horta Lima | Pharmaceutical preparation containing an acetylcholinesterase ihibitor and an antidepressant with 5-ht and alpha-2-adrenoceptor blocking properties. |
| EP2275095A3 (en) * | 2005-08-26 | 2011-08-17 | Braincells, Inc. | Neurogenesis by muscarinic receptor modulation |
| US20100190792A1 (en) * | 2007-03-06 | 2010-07-29 | Allergan, Inc | Methods for treating cognitive disorders using 1-benzyl-1-hydroxy-2,3-diamino-propyl amines, 3-benzyl-3-hydroxy-2-amino-propionic acid amides and related compounds |
| US8173683B2 (en) * | 2007-03-06 | 2012-05-08 | Allergan, Inc. | Methods for treating cognitive disorders |
| WO2008109286A1 (en) * | 2007-03-06 | 2008-09-12 | Allergan, Inc. | Methods for treating cognitive disorders using 1-aryl-1-hydroxy-2,3-diamino-propyl amines, 1-heteroaryl-1-hydroxy-2,3-diamino-propyl amines and related compounds |
| DK2481407T3 (en) * | 2007-03-06 | 2019-01-07 | Allergan Inc | RELATIONSHIPS TO USE IN TREATMENT OF COGNITIVE DISORDERS |
| RU2491931C2 (ru) * | 2007-07-17 | 2013-09-10 | Аллерган, Инк. | Способы лечения тревоги |
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- 2010-07-16 DK DK10735143.9T patent/DK2453890T3/da active
- 2010-07-16 PT PT107351439T patent/PT2453890T/pt unknown
- 2010-07-16 RU RU2012103401A patent/RU2607946C2/ru not_active Application Discontinuation
- 2010-07-16 BR BR112012001047A patent/BR112012001047A2/pt not_active IP Right Cessation
- 2010-07-16 ES ES10735143T patent/ES2809298T3/es active Active
- 2010-07-16 KR KR1020127003979A patent/KR101757003B1/ko active Active
- 2010-07-16 WO PCT/US2010/042308 patent/WO2011009061A1/en active Application Filing
- 2010-07-16 JP JP2012520814A patent/JP2012533566A/ja active Pending
- 2010-07-16 EP EP10735143.9A patent/EP2453890B1/en active Active
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Also Published As
| Publication number | Publication date |
|---|---|
| US20130040938A1 (en) | 2013-02-14 |
| AU2010273977A1 (en) | 2012-02-02 |
| RU2012103401A (ru) | 2013-08-27 |
| RU2016151986A (ru) | 2018-12-19 |
| DK2453890T3 (da) | 2020-08-17 |
| KR20120090029A (ko) | 2012-08-16 |
| EP2453890A1 (en) | 2012-05-23 |
| BR112012001047A2 (pt) | 2019-09-24 |
| EP2453890B1 (en) | 2020-05-27 |
| KR101757003B1 (ko) | 2017-07-11 |
| RU2607946C2 (ru) | 2017-01-11 |
| PT2453890T (pt) | 2020-08-25 |
| WO2011009061A1 (en) | 2011-01-20 |
| CN102497861A (zh) | 2012-06-13 |
| IN2012DN01209A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 2015-04-10 |
| US20110015179A1 (en) | 2011-01-20 |
| ES2809298T3 (es) | 2021-03-03 |
| US9492543B2 (en) | 2016-11-15 |
| JP2012533566A (ja) | 2012-12-27 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FZDE | Discontinued |
Effective date: 20150716 |