CA2719115A1 - Methods, dosage forms, and kits for administering ziprasidone without food - Google Patents
Methods, dosage forms, and kits for administering ziprasidone without food Download PDFInfo
- Publication number
- CA2719115A1 CA2719115A1 CA2719115A CA2719115A CA2719115A1 CA 2719115 A1 CA2719115 A1 CA 2719115A1 CA 2719115 A CA2719115 A CA 2719115A CA 2719115 A CA2719115 A CA 2719115A CA 2719115 A1 CA2719115 A1 CA 2719115A1
- Authority
- CA
- Canada
- Prior art keywords
- ziprasidone
- dosage form
- human
- solid oral
- oral dosage
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
- MVWVFYHBGMAFLY-UHFFFAOYSA-N ziprasidone Chemical compound C1=CC=C2C(N3CCN(CC3)CCC3=CC=4CC(=O)NC=4C=C3Cl)=NSC2=C1 MVWVFYHBGMAFLY-UHFFFAOYSA-N 0.000 title claims abstract description 639
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- ZCBZSCBNOOIHFP-UHFFFAOYSA-N ziprasidone hydrochloride hydrate Chemical compound [H+].O.[Cl-].C1=CC=C2C(N3CCN(CC3)CCC3=CC=4CC(=O)NC=4C=C3Cl)=NSC2=C1 ZCBZSCBNOOIHFP-UHFFFAOYSA-N 0.000 claims description 59
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
Landscapes
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Neurology (AREA)
- General Chemical & Material Sciences (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Psychiatry (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US3494708P | 2008-03-07 | 2008-03-07 | |
| US61/034,947 | 2008-03-07 | ||
| PCT/IB2009/000442 WO2009109844A1 (en) | 2008-03-07 | 2009-03-04 | Methods, dosage forms, and kits for administering ziprasidone without food |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2719115A1 true CA2719115A1 (en) | 2009-09-11 |
Family
ID=40720011
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA2719115A Abandoned CA2719115A1 (en) | 2008-03-07 | 2009-03-04 | Methods, dosage forms, and kits for administering ziprasidone without food |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US20110002989A1 (enExample) |
| EP (1) | EP2280711A1 (enExample) |
| JP (1) | JP2009215293A (enExample) |
| KR (1) | KR20100131477A (enExample) |
| CN (1) | CN102014910A (enExample) |
| AR (1) | AR070964A1 (enExample) |
| AU (1) | AU2009220925A1 (enExample) |
| BR (1) | BRPI0909818A2 (enExample) |
| CA (1) | CA2719115A1 (enExample) |
| IL (1) | IL207792A0 (enExample) |
| MX (1) | MX2010009844A (enExample) |
| RU (1) | RU2010135831A (enExample) |
| TW (1) | TW200950783A (enExample) |
| WO (1) | WO2009109844A1 (enExample) |
| ZA (1) | ZA201005905B (enExample) |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2010082855A1 (en) * | 2009-01-15 | 2010-07-22 | Zaklady Farmaceutyczne Polpharma Sa | Pharmaceutical compositions comprising ziprasidone free base or ziprasidone hydrochloride and the method for their preparation |
| US9510148B2 (en) * | 2009-03-03 | 2016-11-29 | Mobilitie, Llc | System and method for wireless communication to permit audience participation |
| EP2991650A4 (en) * | 2013-05-03 | 2017-01-25 | Syndax Pharmaceuticals Inc. | Methods for the treatment of cancer |
| TW201602108A (zh) | 2013-07-30 | 2016-01-16 | 吉李德康乃狄克公司 | 脾酪胺酸激酶（Ｓｙｋ）抑制劑之多晶型 |
| NZ715745A (en) | 2013-07-30 | 2017-06-30 | Gilead Connecticut Inc | Formulation of syk inhibitors |
| EP3076951B1 (en) * | 2013-12-05 | 2020-09-30 | Celal Albayrak | Process for the production of drug formulations for oral administration |
| TWI662037B (zh) | 2013-12-23 | 2019-06-11 | 美商基利科學股份有限公司 | 脾酪胺酸激酶抑制劑 |
| US10474345B2 (en) * | 2014-04-04 | 2019-11-12 | Shawn SHEY | User interfaces and methods for displaying content |
| EP3193844A1 (en) * | 2014-09-19 | 2017-07-26 | The Procter and Gamble Company | Process for making a core with an active coating |
| JP6796083B2 (ja) | 2015-06-09 | 2020-12-02 | カプスゲル・ベルギウム・ナムローゼ・フェンノートシャップＣａｐｓｕｇｅｌ Ｂｅｌｇｉｕｍ ＮＶ | カプセル中の薬剤の噴霧乾燥ディスパーションからの迅速な溶解を達成するための製剤 |
| US11154510B2 (en) | 2015-06-11 | 2021-10-26 | Alrise Biosystems Gmbh | Process for the preparation of drug loaded microparticles |
| CN107714669A (zh) * | 2016-08-11 | 2018-02-23 | 广东东阳光药业有限公司 | 齐拉西酮缓释剂及其制备方法 |
| EP3672974A1 (en) | 2017-08-25 | 2020-07-01 | Gilead Sciences, Inc. | Polymorphs of syk inhibitors |
| JP2022521413A (ja) | 2019-02-22 | 2022-04-07 | クロノス バイオ インコーポレイテッド | Ｓｙｋ阻害剤としての縮合ピラジンの固体形態 |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2450748A1 (en) * | 2001-06-22 | 2003-01-03 | Pfizer Products Inc. | Pharmaceutical compositions containing polymer and drug assemblies |
| MXPA06002455A (es) * | 2003-09-02 | 2006-08-31 | Pfizer Prod Inc | Formas de dosificacion de liberacion sostenida de ziprasidona. |
| US7825106B2 (en) * | 2003-09-03 | 2010-11-02 | Agi Therapeutics Ltd. | Modified release formulations and methods of treating inflammatory bowel disease |
| EP1703898A2 (en) * | 2003-12-31 | 2006-09-27 | Alpharma, Inc. | Ziprasidone formulations |
| EP1753400A4 (en) * | 2004-06-11 | 2012-11-28 | Reddys Lab Ltd Dr | PHARMACEUTICAL FOR ZIPRASIDONE |
| SG162811A1 (en) * | 2005-06-20 | 2010-07-29 | Elan Pharma Int Ltd | Nanoparticulate and controlled release compositions comprising aryl- heterocyclic compounds |
-
2009
- 2009-03-04 WO PCT/IB2009/000442 patent/WO2009109844A1/en not_active Ceased
- 2009-03-04 CN CN2009801164839A patent/CN102014910A/zh active Pending
- 2009-03-04 RU RU2010135831/15A patent/RU2010135831A/ru not_active Application Discontinuation
- 2009-03-04 KR KR1020107022343A patent/KR20100131477A/ko not_active Ceased
- 2009-03-04 CA CA2719115A patent/CA2719115A1/en not_active Abandoned
- 2009-03-04 TW TW098106972A patent/TW200950783A/zh unknown
- 2009-03-04 EP EP09717510A patent/EP2280711A1/en not_active Withdrawn
- 2009-03-04 MX MX2010009844A patent/MX2010009844A/es not_active Application Discontinuation
- 2009-03-04 BR BRPI0909818A patent/BRPI0909818A2/pt not_active IP Right Cessation
- 2009-03-04 US US12/920,400 patent/US20110002989A1/en not_active Abandoned
- 2009-03-04 AU AU2009220925A patent/AU2009220925A1/en not_active Abandoned
- 2009-03-06 JP JP2009052853A patent/JP2009215293A/ja not_active Withdrawn
- 2009-03-06 AR ARP090100819A patent/AR070964A1/es not_active Application Discontinuation
-
2010
- 2010-08-18 ZA ZA2010/05905A patent/ZA201005905B/en unknown
- 2010-08-24 IL IL207792A patent/IL207792A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| AR070964A1 (es) | 2010-05-19 |
| AU2009220925A1 (en) | 2009-09-11 |
| JP2009215293A (ja) | 2009-09-24 |
| WO2009109844A1 (en) | 2009-09-11 |
| ZA201005905B (en) | 2011-11-30 |
| BRPI0909818A2 (pt) | 2015-10-06 |
| CN102014910A (zh) | 2011-04-13 |
| IL207792A0 (en) | 2010-12-30 |
| EP2280711A1 (en) | 2011-02-09 |
| TW200950783A (en) | 2009-12-16 |
| US20110002989A1 (en) | 2011-01-06 |
| KR20100131477A (ko) | 2010-12-15 |
| MX2010009844A (es) | 2010-09-30 |
| RU2010135831A (ru) | 2012-04-20 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| EEER | Examination request | ||
| FZDE | Discontinued |
Effective date: 20130805 |