CA2695995C - Triazole compounds that modulate hsp90 activity - Google Patents
Triazole compounds that modulate hsp90 activity Download PDFInfo
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- CA2695995C CA2695995C CA2695995A CA2695995A CA2695995C CA 2695995 C CA2695995 C CA 2695995C CA 2695995 A CA2695995 A CA 2695995A CA 2695995 A CA2695995 A CA 2695995A CA 2695995 C CA2695995 C CA 2695995C
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- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
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- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
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- C07F9/6558—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
- C07F9/65583—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system each of the hetero rings containing nitrogen as ring hetero atom
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- C07F9/65586—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system at least one of the hetero rings does not contain nitrogen as ring hetero atom
Landscapes
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US96444707P | 2007-08-13 | 2007-08-13 | |
| US60/964,447 | 2007-08-13 | ||
| PCT/US2008/009667 WO2009023211A1 (en) | 2007-08-13 | 2008-08-13 | Triazole compounds that modulate hsp90 activity |
Publications (2)
| Publication Number | Publication Date |
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| CA2695995A1 CA2695995A1 (en) | 2009-02-19 |
| CA2695995C true CA2695995C (en) | 2015-09-29 |
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| EP2035396B1 (en) | 2006-05-25 | 2014-05-14 | Synta Pharmaceuticals Corp. | Triazole compounds that modulate hsp90 activity |
| CA2677481C (en) | 2007-02-08 | 2015-07-07 | Synta Pharmaceuticals Corp. | Triazole compounds that modulate hsp90 activity |
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| US20140005145A1 (en) | 2010-12-08 | 2014-01-02 | Synta Pharmaceuticals Corp. | Combination breast cancer therapy with hsp90 inhibitory compounds |
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| CA2871540A1 (en) | 2012-05-10 | 2013-11-14 | Synta Pharmaceuticals Corp. | Treating cancer with hsp90 inhibitory compounds |
| CN103664910B (zh) * | 2012-09-14 | 2017-07-04 | 南京大学 | 含1，4‑苯并二噁烷的1，2，4‑三氮唑类衍生物及其制法与其抗菌活性 |
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| WO2017192485A1 (en) | 2016-05-03 | 2017-11-09 | Amgen Inc. | Heterocyclic triazole compounds as agonists of the apj receptor |
| EP3541792B1 (en) | 2016-11-16 | 2020-12-23 | Amgen Inc. | Triazole furan compounds as agonists of the apj receptor |
| MA46827A (fr) | 2016-11-16 | 2019-09-25 | Amgen Inc | Composés de triazole à substitution cycloalkyle en tant qu'agonistes du récepteur apj |
| WO2018097945A1 (en) | 2016-11-16 | 2018-05-31 | Amgen Inc. | Heteroaryl-substituted triazoles as apj receptor agonists |
| US10906890B2 (en) | 2016-11-16 | 2021-02-02 | Amgen Inc. | Triazole phenyl compounds as agonists of the APJ receptor |
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| US11191762B2 (en) | 2016-11-16 | 2021-12-07 | Amgen Inc. | Alkyl substituted triazole compounds as agonists of the APJ Receptor |
| US10767164B2 (en) | 2017-03-30 | 2020-09-08 | The Research Foundation For The State University Of New York | Microenvironments for self-assembly of islet organoids from stem cells differentiation |
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| CN113121505B (zh) * | 2021-03-02 | 2023-03-07 | 中国人民解放军海军军医大学 | 一种具有抗真菌与抗肿瘤双重作用的三唑酮类化合物及应用 |
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| CN101801983B (zh) | 2007-08-13 | 2014-01-29 | 辛塔制药公司 | 调控hsp90活性的三唑化合物 |
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| AU2008287367A1 (en) | 2009-02-19 |
| KR20100057030A (ko) | 2010-05-28 |
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| US9120745B2 (en) | 2015-09-01 |
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| US20110195094A1 (en) | 2011-08-11 |
| MX2010001565A (es) | 2010-04-27 |
| EP2193135A1 (en) | 2010-06-09 |
| TWI438199B (zh) | 2014-05-21 |
| IL203663A (en) | 2015-08-31 |
| CA2695995A1 (en) | 2009-02-19 |
| JP2010536753A (ja) | 2010-12-02 |
| NZ583205A (en) | 2012-03-30 |
| AU2008287367B2 (en) | 2012-02-23 |
| CN101801983B (zh) | 2014-01-29 |
| US20140296186A1 (en) | 2014-10-02 |
| CN101801983A (zh) | 2010-08-11 |
| US20150366885A1 (en) | 2015-12-24 |
| ZA201001064B (en) | 2010-10-27 |
| BRPI0815116A2 (pt) | 2015-01-27 |
| JP5596543B2 (ja) | 2014-09-24 |
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