CA2668441C - Formulations and uses of 2-hydroxy-5-phenylazobenzoic acid derivatives - Google Patents
Formulations and uses of 2-hydroxy-5-phenylazobenzoic acid derivatives Download PDFInfo
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- CA2668441C CA2668441C CA2668441A CA2668441A CA2668441C CA 2668441 C CA2668441 C CA 2668441C CA 2668441 A CA2668441 A CA 2668441A CA 2668441 A CA2668441 A CA 2668441A CA 2668441 C CA2668441 C CA 2668441C
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- balsalazide
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- A61K31/60—Salicylic acid; Derivatives thereof
- A61K31/606—Salicylic acid; Derivatives thereof having amino groups
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/63—Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide
- A61K31/635—Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide having a heterocyclic ring, e.g. sulfadiazine
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- A61K31/655—Azo (—N=N—), diazo (=N2), azoxy (>N—O—N< or N(=O)—N<), azido (—N3) or diazoamino (—N=N—N<) compounds
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- A61K31/66—Phosphorus compounds
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
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- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
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- Bioinformatics & Cheminformatics (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
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Priority Applications (1)
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| CA3004028A CA3004028C (en) | 2006-11-03 | 2007-03-23 | Formulations and uses of 2-hydroxy-5-phenylazobenzoic acid derivatives |
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| US11/592,854 | 2006-11-03 | ||
| US11/592,854 US8921344B2 (en) | 2006-11-03 | 2006-11-03 | Formulations and uses of 2-hydroxy-5-phenylazobenzoic acid derivatives |
| PCT/US2007/007438 WO2008063211A2 (en) | 2006-11-03 | 2007-03-23 | Formulations and uses of 2-hydroxy-5-phenylazobenzoic acid derivatives |
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| CA3004028A Division CA3004028C (en) | 2006-11-03 | 2007-03-23 | Formulations and uses of 2-hydroxy-5-phenylazobenzoic acid derivatives |
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| CA2668441A1 CA2668441A1 (en) | 2008-05-29 |
| CA2668441C true CA2668441C (en) | 2018-06-12 |
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| CA3004028A Active CA3004028C (en) | 2006-11-03 | 2007-03-23 | Formulations and uses of 2-hydroxy-5-phenylazobenzoic acid derivatives |
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| CA3004028A Active CA3004028C (en) | 2006-11-03 | 2007-03-23 | Formulations and uses of 2-hydroxy-5-phenylazobenzoic acid derivatives |
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| EP (1) | EP2096912B1 (enExample) |
| JP (2) | JP6067203B2 (enExample) |
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| AU (1) | AU2007322362B2 (enExample) |
| BR (1) | BRPI0717859A2 (enExample) |
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| IL (1) | IL198513B (enExample) |
| MX (1) | MX2009004826A (enExample) |
| WO (1) | WO2008063211A2 (enExample) |
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| CA2359812C (en) | 2000-11-20 | 2004-02-10 | The Procter & Gamble Company | Pharmaceutical dosage form with multiple coatings for reduced impact of coating fractures |
| EP2361620B1 (en) | 2004-02-06 | 2016-04-06 | PHARMATEL (R&D) PTY LIMITED as Trustee for the PHARMATEL (R & D) TRUST | Use of aminosalicylates in diarrhoea-predominant irritable bowel syndrome |
| US8497258B2 (en) | 2005-11-12 | 2013-07-30 | The Regents Of The University Of California | Viscous budesonide for the treatment of inflammatory diseases of the gastrointestinal tract |
| US7541384B2 (en) | 2007-06-08 | 2009-06-02 | Axcan Pharma Inc. | Mesalamine suppository |
| US8217083B2 (en) * | 2007-06-08 | 2012-07-10 | Aptalis Pharma Canada Inc. | Mesalamine suppository |
| US8436051B2 (en) * | 2007-06-08 | 2013-05-07 | Aptalis Pharma Canada Inc. | Mesalamine suppository |
| ITMI20071965A1 (it) * | 2007-10-11 | 2009-04-12 | Domenico Russo | Composizione farmaceutica comprendente sucralfato e mesalazina |
| CA2739465C (en) * | 2008-10-03 | 2017-01-31 | Dr. Falk Pharma Gmbh | Compositions and methods for the treatment of bowel diseases with granulated mesalamine |
| US20120111756A1 (en) * | 2008-12-17 | 2012-05-10 | Altheus Therapeutics, Inc. | Enema formulations |
| WO2010144865A2 (en) | 2009-06-12 | 2010-12-16 | Meritage Pharma, Inc. | Methods for treating gastrointestinal disorders |
| AU2011245455A1 (en) * | 2010-04-26 | 2012-11-15 | Salix Pharmaceuticals, Ltd. | Formulations and uses of 2-hydroxy-5-phenylazobenzoic acid derivatives for the treatment of males |
| PL3884947T3 (pl) * | 2010-12-03 | 2024-05-06 | Nalpropion Pharmaceuticals Llc | Wzrost biodostępności leku w terapii naltreksonem |
| CN103333084B (zh) * | 2013-06-09 | 2015-01-07 | 陕西新药技术开发中心 | 3,3’-偶氮双[6-(丁酰氧基)苯甲酸]及其制备方法和应用 |
| CN103483220B (zh) * | 2013-06-09 | 2015-06-17 | 陕西新药技术开发中心 | 一种化合物及其制备方法和抗溃疡性结肠炎用途 |
| CN104706582A (zh) * | 2013-12-12 | 2015-06-17 | 四川健能制药有限公司 | 含有美沙拉秦的药物组合物 |
| US10100005B1 (en) * | 2017-11-17 | 2018-10-16 | Eclipse Therapeutics, LLC | Mesalazine derivatives |
| JP2020090456A (ja) * | 2018-12-05 | 2020-06-11 | 日本化薬株式会社 | エルロチニブを有効成分とする医薬錠剤 |
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| BE791889A (fr) * | 1971-11-26 | 1973-05-24 | Pharmacia Ab | Nouveaux derives de la pyridine |
| US4298595A (en) * | 1978-12-20 | 1981-11-03 | Dynapol | Pharmaceutical preparations containing a polymeric agent for releasing 5-aminosalicylic acid or its salts into the gastrointestinal tract |
| US4960765A (en) * | 1980-03-20 | 1990-10-02 | Farmaceutisk Laboratorium Ferring A/S | Pharmaceutical composition and method for the treatment of colitis ulcerosa and Crohn's disease by oral administration |
| WO1981002671A1 (en) * | 1980-03-20 | 1981-10-01 | Ferring Farma Lab | Pharmaceutical composition and method for the treatment of colitis ulcerosa and crohn's disease by oral administration |
| EP0039306B1 (de) * | 1980-03-28 | 1984-01-11 | Ciba-Geigy Ag | Neue Azofarbstoffe, Verfahren zu deren Herstellung und deren Verwendung |
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2006
- 2006-11-03 US US11/592,854 patent/US8921344B2/en active Active
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2007
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- 2007-03-23 KR KR1020097011493A patent/KR20090118906A/ko not_active Ceased
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- 2007-03-23 DK DK07754015.1T patent/DK2096912T3/en active
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- 2007-03-23 MX MX2009004826A patent/MX2009004826A/es unknown
- 2007-03-23 CN CNA2007800491919A patent/CN101610670A/zh active Pending
- 2007-03-23 AU AU2007322362A patent/AU2007322362B2/en not_active Ceased
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Also Published As
| Publication number | Publication date |
|---|---|
| WO2008063211A3 (en) | 2008-11-20 |
| EP2096912B1 (en) | 2018-05-30 |
| CN101610670A (zh) | 2009-12-23 |
| CA3004028C (en) | 2021-07-13 |
| CA3004028A1 (en) | 2008-05-29 |
| US8921344B2 (en) | 2014-12-30 |
| JP2013032395A (ja) | 2013-02-14 |
| US20070167416A1 (en) | 2007-07-19 |
| BRPI0717859A2 (pt) | 2013-01-22 |
| WO2008063211A2 (en) | 2008-05-29 |
| IL198513B (en) | 2018-05-31 |
| IL198513A0 (en) | 2010-02-17 |
| KR20140098863A (ko) | 2014-08-08 |
| DK2096912T3 (en) | 2018-08-27 |
| KR20090118906A (ko) | 2009-11-18 |
| EP2096912A2 (en) | 2009-09-09 |
| CA2668441A1 (en) | 2008-05-29 |
| EP2096912A4 (en) | 2010-01-06 |
| JP2010509326A (ja) | 2010-03-25 |
| AU2007322362B2 (en) | 2013-06-20 |
| MX2009004826A (es) | 2009-07-17 |
| JP6067203B2 (ja) | 2017-01-25 |
| AU2007322362A1 (en) | 2008-05-29 |
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