CA2653460A1 - Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidinyl derivative and its medical use - Google Patents

Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidinyl derivative and its medical use Download PDF

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Publication number
CA2653460A1
CA2653460A1 CA002653460A CA2653460A CA2653460A1 CA 2653460 A1 CA2653460 A1 CA 2653460A1 CA 002653460 A CA002653460 A CA 002653460A CA 2653460 A CA2653460 A CA 2653460A CA 2653460 A1 CA2653460 A1 CA 2653460A1
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CA
Canada
Prior art keywords
disorders
diaza
bicyclo
pain
disease
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002653460A
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English (en)
French (fr)
Inventor
Dan Peters
Gunnar M. Olsen
Elsebet Ostergaard Nielsen
Daniel B. Timmermann
Steven Charles Loechel
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
NTG Nordic Transport Group AS
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Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of CA2653460A1 publication Critical patent/CA2653460A1/en
Abandoned legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08—Bridged systems
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Addiction (AREA)
  • Psychiatry (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Dermatology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Gynecology & Obstetrics (AREA)
  • Obesity (AREA)
  • Pregnancy & Childbirth (AREA)
  • Psychology (AREA)
  • Pulmonology (AREA)
  • Hematology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Vascular Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Rheumatology (AREA)
CA002653460A 2006-05-30 2007-05-29 Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidinyl derivative and its medical use Abandoned CA2653460A1 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US80902306P 2006-05-30 2006-05-30
DKPA200600730 2006-05-30
DKPA200600730 2006-05-30
US60/809,023 2006-05-30
PCT/EP2007/055172 WO2007138041A1 (en) 2006-05-30 2007-05-29 Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidinyl derivative and its medical use

Publications (1)

Publication Number Publication Date
CA2653460A1 true CA2653460A1 (en) 2007-12-06

Family

ID=38258823

Family Applications (3)

Application Number Title Priority Date Filing Date
CA002653460A Abandoned CA2653460A1 (en) 2006-05-30 2007-05-29 Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidinyl derivative and its medical use
CA002653681A Abandoned CA2653681A1 (en) 2006-05-30 2007-05-29 Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidinyl derivatives and their medical use
CA002653371A Abandoned CA2653371A1 (en) 2006-05-30 2007-05-29 Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidinyl derivative and its medical use

Family Applications After (2)

Application Number Title Priority Date Filing Date
CA002653681A Abandoned CA2653681A1 (en) 2006-05-30 2007-05-29 Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidinyl derivatives and their medical use
CA002653371A Abandoned CA2653371A1 (en) 2006-05-30 2007-05-29 Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidinyl derivative and its medical use

Country Status (7)

Country Link
US (3) US20090197872A1 (enExample)
EP (3) EP2029595B1 (enExample)
JP (3) JP2009538868A (enExample)
AU (3) AU2007267176A1 (enExample)
CA (3) CA2653460A1 (enExample)
MX (3) MX2008014885A (enExample)
WO (3) WO2007138041A1 (enExample)

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MX2008014885A (es) * 2006-05-30 2008-12-05 Neurosearch As Nuevos derivados de 1,4-diaza-biciclo[3.2.2]nonil pirimidinilo y su uso medico.
WO2009024517A1 (en) * 2007-08-17 2009-02-26 Neurosearch A/S Novel 1,4-diaza-bicyclo[3.2.2]nonyl heteroaryl derivatives useful as nicotinic acetylcholine receptor ligands
DE102007053771A1 (de) * 2007-11-12 2009-05-14 Merck Patent Gmbh Organische Elektrolumineszenzvorrichtungen
CA2705752A1 (en) * 2007-11-14 2009-05-22 Neurosearch A/S Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidine derivatives and their medical use
US20110046118A1 (en) * 2007-11-14 2011-02-24 Neurosearch A/S Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidine derivatives and their medical use
EP2209781A1 (en) * 2007-11-14 2010-07-28 NeuroSearch AS Novel 1,4-diaza-bicycloý3.2.2¨nonyl pyrimidine derivatives and their medical use
WO2010026176A1 (en) * 2008-09-05 2010-03-11 Neurosearch A/S 1,4 -diaza- bicyclo [3.2.2]n0nyl pyrimidine derivatives as nicotinic and monoamine receptor modulators
WO2010026177A1 (en) * 2008-09-05 2010-03-11 Neurosearch A/S 1,4-diaza-bicyclo [3.2.2] nonyl pyridine derivatives as nicotinic and monoamine receptor modulators
US20110269778A1 (en) * 2008-10-10 2011-11-03 Neurosearch A/S Novel diphenyl purine derivatives useful as modulators of nicotinic acetylcholine receptors
US20110257161A1 (en) * 2008-12-04 2011-10-20 Neurosearch A/S Novel diaza-bicyclononyl-phenyl derivatives and their medical use
WO2010084120A1 (en) * 2009-01-21 2010-07-29 Neurosearch A/S N-oxides of 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidinyl derivatives useful as nicotinic acetylcholine receptor ligands
WO2010084121A1 (en) * 2009-01-21 2010-07-29 Neurosearch A/S Novel diaza-bicyclononyl-pyrimidinyl derivatives and their medical use
TWI558398B (zh) 2009-09-22 2016-11-21 諾華公司 菸鹼乙醯膽鹼受體α７活化劑之用途

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JP2010536724A (ja) 2007-08-17 2010-12-02 ノイロサーチ アクティーゼルスカブ ニコチン性アセチルコリン受容体リガンドとして有用な１，４−ジアザ−ビシクロ（３．２．２）ノニルピリミジニル誘導体
WO2009024517A1 (en) 2007-08-17 2009-02-26 Neurosearch A/S Novel 1,4-diaza-bicyclo[3.2.2]nonyl heteroaryl derivatives useful as nicotinic acetylcholine receptor ligands
US20110046118A1 (en) * 2007-11-14 2011-02-24 Neurosearch A/S Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidine derivatives and their medical use
EP2209781A1 (en) * 2007-11-14 2010-07-28 NeuroSearch AS Novel 1,4-diaza-bicycloý3.2.2¨nonyl pyrimidine derivatives and their medical use

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