MX2008014885A - Nuevos derivados de 1,4-diaza-biciclo[3.2.2]nonil pirimidinilo y su uso medico. - Google Patents
Nuevos derivados de 1,4-diaza-biciclo[3.2.2]nonil pirimidinilo y su uso medico.Info
- Publication number
- MX2008014885A MX2008014885A MX2008014885A MX2008014885A MX2008014885A MX 2008014885 A MX2008014885 A MX 2008014885A MX 2008014885 A MX2008014885 A MX 2008014885A MX 2008014885 A MX2008014885 A MX 2008014885A MX 2008014885 A MX2008014885 A MX 2008014885A
- Authority
- MX
- Mexico
- Prior art keywords
- diaza
- bicyclo
- pyrimidin
- alkyl
- disorders
- Prior art date
Links
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Classifications
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- C07—ORGANIC CHEMISTRY
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- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/08—Bridged systems
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- A—HUMAN NECESSITIES
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- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
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- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
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- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US80902306P | 2006-05-30 | 2006-05-30 | |
| DKPA200600730 | 2006-05-30 | ||
| PCT/EP2007/055170 WO2007138039A1 (en) | 2006-05-30 | 2007-05-29 | Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidinyl derivatives and their medical use |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2008014885A true MX2008014885A (es) | 2008-12-05 |
Family
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Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2008014885A MX2008014885A (es) | 2006-05-30 | 2007-05-29 | Nuevos derivados de 1,4-diaza-biciclo[3.2.2]nonil pirimidinilo y su uso medico. |
| MX2008014889A MX2008014889A (es) | 2006-05-30 | 2007-05-29 | Nuevos derivados de 1,4-diaza-biciclo[3.2.2.]nonil pirimidinilo y su uso medico. |
| MX2008014890A MX2008014890A (es) | 2006-05-30 | 2007-05-29 | Nuevos derivados de 1,4-diaza-biciclo[3.2.2]nonil pirimidinilo y su uso medico. |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2008014889A MX2008014889A (es) | 2006-05-30 | 2007-05-29 | Nuevos derivados de 1,4-diaza-biciclo[3.2.2.]nonil pirimidinilo y su uso medico. |
| MX2008014890A MX2008014890A (es) | 2006-05-30 | 2007-05-29 | Nuevos derivados de 1,4-diaza-biciclo[3.2.2]nonil pirimidinilo y su uso medico. |
Country Status (7)
| Country | Link |
|---|---|
| US (3) | US20090197872A1 (enExample) |
| EP (3) | EP2029595B1 (enExample) |
| JP (3) | JP2009538868A (enExample) |
| AU (3) | AU2007267176A1 (enExample) |
| CA (3) | CA2653460A1 (enExample) |
| MX (3) | MX2008014885A (enExample) |
| WO (3) | WO2007138041A1 (enExample) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR20060125885A (ko) * | 2004-02-04 | 2006-12-06 | 뉴로서치 에이/에스 | 콜린 수용체 조절제로서의 디아자바이사이클릭 아릴 유도체 |
| MX2008014885A (es) * | 2006-05-30 | 2008-12-05 | Neurosearch As | Nuevos derivados de 1,4-diaza-biciclo[3.2.2]nonil pirimidinilo y su uso medico. |
| WO2009024517A1 (en) * | 2007-08-17 | 2009-02-26 | Neurosearch A/S | Novel 1,4-diaza-bicyclo[3.2.2]nonyl heteroaryl derivatives useful as nicotinic acetylcholine receptor ligands |
| DE102007053771A1 (de) * | 2007-11-12 | 2009-05-14 | Merck Patent Gmbh | Organische Elektrolumineszenzvorrichtungen |
| CA2705752A1 (en) * | 2007-11-14 | 2009-05-22 | Neurosearch A/S | Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidine derivatives and their medical use |
| US20110046118A1 (en) * | 2007-11-14 | 2011-02-24 | Neurosearch A/S | Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidine derivatives and their medical use |
| EP2209781A1 (en) * | 2007-11-14 | 2010-07-28 | NeuroSearch AS | Novel 1,4-diaza-bicycloý3.2.2¨nonyl pyrimidine derivatives and their medical use |
| WO2010026176A1 (en) * | 2008-09-05 | 2010-03-11 | Neurosearch A/S | 1,4 -diaza- bicyclo [3.2.2]n0nyl pyrimidine derivatives as nicotinic and monoamine receptor modulators |
| WO2010026177A1 (en) * | 2008-09-05 | 2010-03-11 | Neurosearch A/S | 1,4-diaza-bicyclo [3.2.2] nonyl pyridine derivatives as nicotinic and monoamine receptor modulators |
| US20110269778A1 (en) * | 2008-10-10 | 2011-11-03 | Neurosearch A/S | Novel diphenyl purine derivatives useful as modulators of nicotinic acetylcholine receptors |
| US20110257161A1 (en) * | 2008-12-04 | 2011-10-20 | Neurosearch A/S | Novel diaza-bicyclononyl-phenyl derivatives and their medical use |
| WO2010084120A1 (en) * | 2009-01-21 | 2010-07-29 | Neurosearch A/S | N-oxides of 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidinyl derivatives useful as nicotinic acetylcholine receptor ligands |
| WO2010084121A1 (en) * | 2009-01-21 | 2010-07-29 | Neurosearch A/S | Novel diaza-bicyclononyl-pyrimidinyl derivatives and their medical use |
| TWI558398B (zh) | 2009-09-22 | 2016-11-21 | 諾華公司 | 菸鹼乙醯膽鹼受體α７活化劑之用途 |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2786770B1 (fr) * | 1998-12-04 | 2001-01-19 | Synthelabo | Derives de 1,4-diazabicyclo[3.2.2.]nonane, leur preparation et leur application en therapeutique |
| JP2004518723A (ja) * | 2001-02-14 | 2004-06-24 | ワーナー−ランバート・カンパニー、リミテッド、ライアビリティ、カンパニー | ピリミジンマトリックスメタロプロテイナーゼ阻害剤 |
| EP1395257A1 (en) * | 2001-06-12 | 2004-03-10 | Elan Pharmaceuticals, Inc. | Macrocycles useful in the treatment of alzheimer's disease |
| SE0202430D0 (sv) | 2002-08-14 | 2002-08-14 | Astrazeneca Ab | New Compounds |
| CA2498291C (en) * | 2002-09-10 | 2009-04-07 | Pfizer Products Inc. | Diazabicyclic compounds useful in the treatment of cns and other disorders |
| DE60311853T2 (de) | 2002-09-30 | 2007-06-21 | Neurosearch A/S | Neue 1,4-diazabicycloalkanderivate, deren herstellung und verwendung |
| US7223753B2 (en) * | 2002-11-11 | 2007-05-29 | Neurosearch A/S | Diazabicyclic biaryl derivatives |
| EP1562945B1 (en) | 2002-11-11 | 2006-11-15 | Neurosearch A/S | 1,4-diazabicyclo(3,2,2)nonane derivatives, preparation and therapeutical use thereof |
| KR20060125885A (ko) | 2004-02-04 | 2006-12-06 | 뉴로서치 에이/에스 | 콜린 수용체 조절제로서의 디아자바이사이클릭 아릴 유도체 |
| AU2005210039B2 (en) * | 2004-02-04 | 2010-09-02 | Neurosearch A/S | Diazabicyclic aryl derivatives as nicotinic acetylcholine receptor ligands |
| JP2008530172A (ja) | 2005-02-16 | 2008-08-07 | ノイロサーチ アクティーゼルスカブ | ジアザ二環系アリール誘導体及びそれらのニコチン様アセチルコリン受容体におけるコリン作動性リガンドとしての使用 |
| MX2008014885A (es) | 2006-05-30 | 2008-12-05 | Neurosearch As | Nuevos derivados de 1,4-diaza-biciclo[3.2.2]nonil pirimidinilo y su uso medico. |
| JP2010536724A (ja) | 2007-08-17 | 2010-12-02 | ノイロサーチ アクティーゼルスカブ | ニコチン性アセチルコリン受容体リガンドとして有用な１，４−ジアザ−ビシクロ（３．２．２）ノニルピリミジニル誘導体 |
| WO2009024517A1 (en) | 2007-08-17 | 2009-02-26 | Neurosearch A/S | Novel 1,4-diaza-bicyclo[3.2.2]nonyl heteroaryl derivatives useful as nicotinic acetylcholine receptor ligands |
| US20110046118A1 (en) * | 2007-11-14 | 2011-02-24 | Neurosearch A/S | Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidine derivatives and their medical use |
| EP2209781A1 (en) * | 2007-11-14 | 2010-07-28 | NeuroSearch AS | Novel 1,4-diaza-bicycloý3.2.2¨nonyl pyrimidine derivatives and their medical use |
-
2007
- 2007-05-29 MX MX2008014885A patent/MX2008014885A/es not_active Application Discontinuation
- 2007-05-29 CA CA002653460A patent/CA2653460A1/en not_active Abandoned
- 2007-05-29 EP EP07729594A patent/EP2029595B1/en not_active Not-in-force
- 2007-05-29 EP EP07729592A patent/EP2041134A1/en not_active Withdrawn
- 2007-05-29 JP JP2009512570A patent/JP2009538868A/ja not_active Abandoned
- 2007-05-29 US US12/299,108 patent/US20090197872A1/en not_active Abandoned
- 2007-05-29 WO PCT/EP2007/055172 patent/WO2007138041A1/en not_active Ceased
- 2007-05-29 WO PCT/EP2007/055171 patent/WO2007138040A1/en not_active Ceased
- 2007-05-29 AU AU2007267176A patent/AU2007267176A1/en not_active Abandoned
- 2007-05-29 AU AU2007267177A patent/AU2007267177A1/en not_active Abandoned
- 2007-05-29 JP JP2009512571A patent/JP2009538869A/ja not_active Abandoned
- 2007-05-29 MX MX2008014889A patent/MX2008014889A/es not_active Application Discontinuation
- 2007-05-29 JP JP2009512572A patent/JP2009538870A/ja not_active Abandoned
- 2007-05-29 MX MX2008014890A patent/MX2008014890A/es not_active Application Discontinuation
- 2007-05-29 CA CA002653681A patent/CA2653681A1/en not_active Abandoned
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- 2007-05-29 AU AU2007267178A patent/AU2007267178A1/en not_active Abandoned
- 2007-05-29 WO PCT/EP2007/055170 patent/WO2007138039A1/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| US7915272B2 (en) | 2011-03-29 |
| MX2008014890A (es) | 2008-12-05 |
| MX2008014889A (es) | 2008-12-05 |
| WO2007138040A1 (en) | 2007-12-06 |
| WO2007138041A1 (en) | 2007-12-06 |
| EP2049538A1 (en) | 2009-04-22 |
| AU2007267176A1 (en) | 2007-12-06 |
| CA2653681A1 (en) | 2007-12-06 |
| WO2007138040A8 (en) | 2008-11-20 |
| WO2007138039A1 (en) | 2007-12-06 |
| JP2009538869A (ja) | 2009-11-12 |
| EP2029595B1 (en) | 2011-09-21 |
| JP2009538870A (ja) | 2009-11-12 |
| EP2041134A1 (en) | 2009-04-01 |
| US8148365B2 (en) | 2012-04-03 |
| WO2007138041A8 (en) | 2008-11-20 |
| EP2029595A1 (en) | 2009-03-04 |
| US20090197872A1 (en) | 2009-08-06 |
| AU2007267178A1 (en) | 2007-12-06 |
| AU2007267177A1 (en) | 2007-12-06 |
| US20090270403A1 (en) | 2009-10-29 |
| CA2653460A1 (en) | 2007-12-06 |
| CA2653371A1 (en) | 2007-12-06 |
| US20090181984A1 (en) | 2009-07-16 |
| JP2009538868A (ja) | 2009-11-12 |
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