MX2008014885A - Nuevos derivados de 1,4-diaza-biciclo[3.2.2]nonil pirimidinilo y su uso medico. - Google Patents
Nuevos derivados de 1,4-diaza-biciclo[3.2.2]nonil pirimidinilo y su uso medico.Info
- Publication number
- MX2008014885A MX2008014885A MX2008014885A MX2008014885A MX2008014885A MX 2008014885 A MX2008014885 A MX 2008014885A MX 2008014885 A MX2008014885 A MX 2008014885A MX 2008014885 A MX2008014885 A MX 2008014885A MX 2008014885 A MX2008014885 A MX 2008014885A
- Authority
- MX
- Mexico
- Prior art keywords
- diaza
- bicyclo
- pyrimidin
- alkyl
- disorders
- Prior art date
Links
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Classifications
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- C07—ORGANIC CHEMISTRY
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- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/08—Bridged systems
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- A—HUMAN NECESSITIES
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- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
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| US80902306P | 2006-05-30 | 2006-05-30 | |
| DKPA200600730 | 2006-05-30 | ||
| PCT/EP2007/055170 WO2007138039A1 (en) | 2006-05-30 | 2007-05-29 | Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidinyl derivatives and their medical use |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2008014885A true MX2008014885A (es) | 2008-12-05 |
Family
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Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2008014890A MX2008014890A (es) | 2006-05-30 | 2007-05-29 | Nuevos derivados de 1,4-diaza-biciclo[3.2.2]nonil pirimidinilo y su uso medico. |
| MX2008014889A MX2008014889A (es) | 2006-05-30 | 2007-05-29 | Nuevos derivados de 1,4-diaza-biciclo[3.2.2.]nonil pirimidinilo y su uso medico. |
| MX2008014885A MX2008014885A (es) | 2006-05-30 | 2007-05-29 | Nuevos derivados de 1,4-diaza-biciclo[3.2.2]nonil pirimidinilo y su uso medico. |
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| Application Number | Title | Priority Date | Filing Date |
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| MX2008014890A MX2008014890A (es) | 2006-05-30 | 2007-05-29 | Nuevos derivados de 1,4-diaza-biciclo[3.2.2]nonil pirimidinilo y su uso medico. |
| MX2008014889A MX2008014889A (es) | 2006-05-30 | 2007-05-29 | Nuevos derivados de 1,4-diaza-biciclo[3.2.2.]nonil pirimidinilo y su uso medico. |
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| EP (3) | EP2049538A1 (enExample) |
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| CA (3) | CA2653460A1 (enExample) |
| MX (3) | MX2008014890A (enExample) |
| WO (3) | WO2007138040A1 (enExample) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
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| KR20060125885A (ko) * | 2004-02-04 | 2006-12-06 | 뉴로서치 에이/에스 | 콜린 수용체 조절제로서의 디아자바이사이클릭 아릴 유도체 |
| AU2007267178A1 (en) | 2006-05-30 | 2007-12-06 | Neurosearch A/S | Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidinyl derivatives and their medical use |
| JP2010536726A (ja) | 2007-08-17 | 2010-12-02 | ノイロサーチ アクティーゼルスカブ | ニコチン性アセチルコリン受容体リガンドとして有用な新規１，４−ジアザ−ビシクロ〔３．２．２〕ノニルヘテロアリール誘導体 |
| DE102007053771A1 (de) * | 2007-11-12 | 2009-05-14 | Merck Patent Gmbh | Organische Elektrolumineszenzvorrichtungen |
| EP2209783B8 (en) * | 2007-11-14 | 2016-06-01 | Saniona A/S | Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidine derivatives and their medical use |
| JP2011503144A (ja) * | 2007-11-14 | 2011-01-27 | ノイロサーチ アクティーゼルスカブ | 新規の１，４−ジアザ−ビシクロ［３．２．２］ノニルピリミジン誘導体及びその医療への使用 |
| JP2011503146A (ja) * | 2007-11-14 | 2011-01-27 | ノイロサーチ アクティーゼルスカブ | 新規な１，４−ジアザ−ビシクロ［３．２．２］ノニルピリミジン誘導体及びこれらの医療上の使用 |
| WO2010026176A1 (en) * | 2008-09-05 | 2010-03-11 | Neurosearch A/S | 1,4 -diaza- bicyclo [3.2.2]n0nyl pyrimidine derivatives as nicotinic and monoamine receptor modulators |
| WO2010026177A1 (en) * | 2008-09-05 | 2010-03-11 | Neurosearch A/S | 1,4-diaza-bicyclo [3.2.2] nonyl pyridine derivatives as nicotinic and monoamine receptor modulators |
| WO2010040806A1 (en) * | 2008-10-10 | 2010-04-15 | Neurosearch A/S | Novel diphenyl purine derivatives useful as modulators of nicotinic acetylcholine receptors |
| US20110257161A1 (en) * | 2008-12-04 | 2011-10-20 | Neurosearch A/S | Novel diaza-bicyclononyl-phenyl derivatives and their medical use |
| WO2010084120A1 (en) * | 2009-01-21 | 2010-07-29 | Neurosearch A/S | N-oxides of 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidinyl derivatives useful as nicotinic acetylcholine receptor ligands |
| WO2010084121A1 (en) * | 2009-01-21 | 2010-07-29 | Neurosearch A/S | Novel diaza-bicyclononyl-pyrimidinyl derivatives and their medical use |
| TWI558398B (zh) | 2009-09-22 | 2016-11-21 | 諾華公司 | 菸鹼乙醯膽鹼受體α７活化劑之用途 |
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| FR2786770B1 (fr) * | 1998-12-04 | 2001-01-19 | Synthelabo | Derives de 1,4-diazabicyclo[3.2.2.]nonane, leur preparation et leur application en therapeutique |
| EP1368323B1 (en) * | 2001-02-14 | 2010-06-30 | Warner-Lambert Company LLC | Pyrimidine matrix metalloproteinase inhibitors |
| WO2002100399A1 (en) * | 2001-06-12 | 2002-12-19 | Elan Pharmaceuticals, Inc. | Macrocycles useful in the treatment of alzheimer's disease |
| SE0202430D0 (sv) | 2002-08-14 | 2002-08-14 | Astrazeneca Ab | New Compounds |
| AU2003255993A1 (en) * | 2002-09-10 | 2004-04-30 | Pfizer Products Inc. | Diazabicyclic compounds useful in the treatment of cns and other disorders |
| DE60326894D1 (de) | 2002-09-30 | 2009-05-07 | Neurosearch As | 1,4-Diazabicycloalkanderivate, deren Herstellung und Verwendung |
| ATE345342T1 (de) | 2002-11-11 | 2006-12-15 | Neurosearch As | 1,4-dizabicyclo(3,2,2)nonane derivative, verfahren zur ihre herstellung und therapeutical verwendung |
| US7223753B2 (en) * | 2002-11-11 | 2007-05-29 | Neurosearch A/S | Diazabicyclic biaryl derivatives |
| KR20060125885A (ko) * | 2004-02-04 | 2006-12-06 | 뉴로서치 에이/에스 | 콜린 수용체 조절제로서의 디아자바이사이클릭 아릴 유도체 |
| US20080227772A1 (en) * | 2004-02-04 | 2008-09-18 | Neurosearch A/S | Diazabicyclic Aryl Derivatives as Nicotinic Acetylcholine Receptor Ligands |
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| JP2010536726A (ja) | 2007-08-17 | 2010-12-02 | ノイロサーチ アクティーゼルスカブ | ニコチン性アセチルコリン受容体リガンドとして有用な新規１，４−ジアザ−ビシクロ〔３．２．２〕ノニルヘテロアリール誘導体 |
| WO2009024515A1 (en) | 2007-08-17 | 2009-02-26 | Neurosearch A/S | 1,4-diaza-bicycl0(3.2.2)n0nyl pyrimidinyl derivatives useful as nicotinic acetylcholine- receptor ligands |
| JP2011503144A (ja) * | 2007-11-14 | 2011-01-27 | ノイロサーチ アクティーゼルスカブ | 新規の１，４−ジアザ−ビシクロ［３．２．２］ノニルピリミジン誘導体及びその医療への使用 |
| JP2011503146A (ja) * | 2007-11-14 | 2011-01-27 | ノイロサーチ アクティーゼルスカブ | 新規な１，４−ジアザ−ビシクロ［３．２．２］ノニルピリミジン誘導体及びこれらの医療上の使用 |
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| WO2007138040A1 (en) | 2007-12-06 |
| US20090181984A1 (en) | 2009-07-16 |
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