CA2620491A1 - Pharmaceutical dosage forms and compositions comprising lecoztan - Google Patents
Pharmaceutical dosage forms and compositions comprising lecoztan Download PDFInfo
- Publication number
- CA2620491A1 CA2620491A1 CA002620491A CA2620491A CA2620491A1 CA 2620491 A1 CA2620491 A1 CA 2620491A1 CA 002620491 A CA002620491 A CA 002620491A CA 2620491 A CA2620491 A CA 2620491A CA 2620491 A1 CA2620491 A1 CA 2620491A1
- Authority
- CA
- Canada
- Prior art keywords
- patient
- lecozotan
- mean
- max
- dosage form
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
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Classifications
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Epidemiology (AREA)
- Addiction (AREA)
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- Pain & Pain Management (AREA)
- Reproductive Health (AREA)
- Hematology (AREA)
- Hospice & Palliative Care (AREA)
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- Child & Adolescent Psychology (AREA)
- Diabetes (AREA)
- Heart & Thoracic Surgery (AREA)
- Obesity (AREA)
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- Anesthesiology (AREA)
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- Cardiology (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US71541705P | 2005-09-09 | 2005-09-09 | |
| US60/715,417 | 2005-09-09 | ||
| PCT/US2006/034813 WO2007030589A2 (en) | 2005-09-09 | 2006-09-06 | Pharmaceutical dosage forms and compositions comprising lecoztan |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2620491A1 true CA2620491A1 (en) | 2007-03-15 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA002620491A Abandoned CA2620491A1 (en) | 2005-09-09 | 2006-09-06 | Pharmaceutical dosage forms and compositions comprising lecoztan |
Country Status (17)
| Country | Link |
|---|---|
| EP (1) | EP1928863A2 (enExample) |
| JP (1) | JP2009507850A (enExample) |
| KR (1) | KR20080043855A (enExample) |
| CN (1) | CN101258146A (enExample) |
| AR (1) | AR058033A1 (enExample) |
| AU (1) | AU2006287543A1 (enExample) |
| BR (1) | BRPI0615771A2 (enExample) |
| CA (1) | CA2620491A1 (enExample) |
| CR (1) | CR9800A (enExample) |
| EC (1) | ECSP088236A (enExample) |
| GT (1) | GT200600403A (enExample) |
| IL (1) | IL189827A0 (enExample) |
| NO (1) | NO20081100L (enExample) |
| PE (1) | PE20070334A1 (enExample) |
| RU (1) | RU2008108216A (enExample) |
| TW (1) | TW200800198A (enExample) |
| WO (1) | WO2007030589A2 (enExample) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8134029B2 (en) | 2002-09-16 | 2012-03-13 | Sunovion Pharmaceuticals Inc. | Treatment of CNS disorders with trans 4-(3,4-dichlorophenyl)-1,2,3,4-tetrahydro-1-napthalenamine |
| WO2007006003A2 (en) | 2005-07-06 | 2007-01-11 | Sepracor Inc. | Combinations of eszopiclone and trans 4-(3,4-dichlorophenyl)-1,2,3,4-tetrahydro-n-methyl-1-napthalenamine or trans 4-(3,4-dichlorophenyl)-1,2,3,4-tetrahydro-1-napthalenamine, and methods of treatment of menopause and mood, anxiety, and cognitive disorders |
| EP2429514A1 (en) * | 2009-05-13 | 2012-03-21 | Sunovion Pharmaceuticals Inc. | Compositions comprising transnorsertraline and serotonin receptor 1a agonists/ antagonists and uses thereof |
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| CA2426666A1 (en) * | 2000-09-29 | 2002-04-04 | Solvay Pharmaceuticals B.V. | Ion-strength independent sustained release pharmaceutical formulation |
| GB2407498B (en) * | 2003-10-30 | 2008-06-11 | Cipla Ltd | Oral formulations for 5-HT receptor agonists with reduced degradation of active ingredient |
| US20050215561A1 (en) * | 2004-03-19 | 2005-09-29 | Krishnendu Ghosh | Pharmaceutical dosage forms and compositions |
| KR20070112797A (ko) * | 2005-03-01 | 2007-11-27 | 와이어쓰 | 결정질 및 비결정질4-시아노-ｎ-((2ｒ)-2-[4-(2,3-디히드로-벤조[1,4]디옥신-5-일)-피페라진-1-일]-프로필)-ｎ-피리딘-2-일-벤즈아미드염산염 |
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2006
- 2006-09-06 BR BRPI0615771-8A patent/BRPI0615771A2/pt not_active Application Discontinuation
- 2006-09-06 WO PCT/US2006/034813 patent/WO2007030589A2/en not_active Ceased
- 2006-09-06 JP JP2008530186A patent/JP2009507850A/ja not_active Withdrawn
- 2006-09-06 AR ARP060103880A patent/AR058033A1/es unknown
- 2006-09-06 CA CA002620491A patent/CA2620491A1/en not_active Abandoned
- 2006-09-06 AU AU2006287543A patent/AU2006287543A1/en not_active Abandoned
- 2006-09-06 EP EP06790193A patent/EP1928863A2/en not_active Withdrawn
- 2006-09-06 TW TW095132852A patent/TW200800198A/zh unknown
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- 2006-09-06 RU RU2008108216/14A patent/RU2008108216A/ru not_active Application Discontinuation
- 2006-09-06 GT GT200600403A patent/GT200600403A/es unknown
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Also Published As
| Publication number | Publication date |
|---|---|
| WO2007030589A2 (en) | 2007-03-15 |
| PE20070334A1 (es) | 2007-05-08 |
| RU2008108216A (ru) | 2009-10-20 |
| KR20080043855A (ko) | 2008-05-19 |
| IL189827A0 (en) | 2008-11-03 |
| CR9800A (es) | 2008-04-28 |
| NO20081100L (no) | 2008-06-03 |
| JP2009507850A (ja) | 2009-02-26 |
| ECSP088236A (es) | 2008-04-28 |
| TW200800198A (en) | 2008-01-01 |
| CN101258146A (zh) | 2008-09-03 |
| BRPI0615771A2 (pt) | 2011-05-24 |
| WO2007030589A3 (en) | 2007-11-01 |
| AR058033A1 (es) | 2008-01-23 |
| EP1928863A2 (en) | 2008-06-11 |
| GT200600403A (es) | 2007-09-19 |
| AU2006287543A1 (en) | 2007-03-15 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FZDE | Discontinued |