CA2613474A1 - Compositions de nanoparticules a liberation controlee comprenant des composes d'aryle heterocyclique - Google Patents
Compositions de nanoparticules a liberation controlee comprenant des composes d'aryle heterocyclique Download PDFInfo
- Publication number
- CA2613474A1 CA2613474A1 CA002613474A CA2613474A CA2613474A1 CA 2613474 A1 CA2613474 A1 CA 2613474A1 CA 002613474 A CA002613474 A CA 002613474A CA 2613474 A CA2613474 A CA 2613474A CA 2613474 A1 CA2613474 A1 CA 2613474A1
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- Prior art keywords
- composition
- less
- ziprasidone
- release
- particles
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
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Classifications
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- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
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- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
- A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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- A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
- A61K9/145—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
- A61K9/146—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic macromolecular compounds
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4808—Preparations in capsules, e.g. of gelatin, of chocolate characterised by the form of the capsule or the structure of the filling; Capsules containing small tablets; Capsules with outer layer for immediate drug release
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- A—HUMAN NECESSITIES
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- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5084—Mixtures of one or more drugs in different galenical forms, at least one of which being granules, microcapsules or (coated) microparticles according to A61K9/16 or A61K9/50, e.g. for obtaining a specific release pattern or for combining different drugs
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
Landscapes
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
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- Veterinary Medicine (AREA)
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- Psychiatry (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US69209605P | 2005-06-20 | 2005-06-20 | |
US60/692,096 | 2005-06-20 | ||
US11/372,857 US20060240105A1 (en) | 1998-11-02 | 2006-03-10 | Multiparticulate modified release composition |
US11/372,857 | 2006-03-10 | ||
PCT/US2006/023695 WO2007027273A1 (fr) | 2005-06-20 | 2006-06-19 | Compositions de nanoparticules à libération contrôlée comprenant des composés d'aryle hétérocyclique |
Publications (1)
Publication Number | Publication Date |
---|---|
CA2613474A1 true CA2613474A1 (fr) | 2007-03-08 |
Family
ID=37809174
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CA002613474A Abandoned CA2613474A1 (fr) | 2005-06-20 | 2006-06-19 | Compositions de nanoparticules a liberation controlee comprenant des composes d'aryle heterocyclique |
Country Status (12)
Country | Link |
---|---|
EP (1) | EP1901722A4 (fr) |
KR (1) | KR20080024206A (fr) |
CN (1) | CN101879140A (fr) |
AU (1) | AU2006285349A1 (fr) |
BR (1) | BRPI0612297A2 (fr) |
CA (1) | CA2613474A1 (fr) |
EA (1) | EA200800092A1 (fr) |
HK (1) | HK1117060A1 (fr) |
IL (1) | IL188093A0 (fr) |
NO (1) | NO20076628L (fr) |
SG (1) | SG162811A1 (fr) |
WO (1) | WO2007027273A1 (fr) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BRPI0909818A2 (pt) * | 2008-03-07 | 2015-10-06 | Pfizer | métodos, formas de dosagem e conjunto para administrar ziprasidona sem alimentos |
DE102008045854A1 (de) | 2008-09-05 | 2010-03-11 | Tiefenbacher Pharmachemikalien Alfred E. Tiefenbacher Gmbh & Co. Kg | Partikel aus Ziprasidone und einem Sprengmittel enthaltende Pharmazeutische Zusammensetzung |
WO2010082855A1 (fr) * | 2009-01-15 | 2010-07-22 | Zaklady Farmaceutyczne Polpharma Sa | Compositions pharmaceutiques comprenant de la ziprasidone sous forme de base libre ou de chlorhydrate et leur méthode d'élaboration |
US20130108701A1 (en) | 2010-05-25 | 2013-05-02 | Krishna Murthy Bhavanasi | Solid Dosage Forms of Antipsychotics |
EP3082852B1 (fr) | 2013-12-16 | 2020-06-17 | Massachusetts Institute of Technology | Formulations vaccinales micromoulées ou imprimées en 3d, à libération pulsatile |
MX2016007786A (es) | 2013-12-16 | 2017-03-03 | Massachusetts Inst Technology | Formulaciones de sal de micronutrientes fortificadas. |
MA41611A (fr) * | 2015-02-23 | 2018-01-02 | Omthera Pharmaceuticals Inc | Préparations en milli-capsules comprenant des acides gras polyinsaturés libres |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5145684A (en) * | 1991-01-25 | 1992-09-08 | Sterling Drug Inc. | Surface modified drug nanoparticles |
NZ248813A (en) * | 1992-11-25 | 1995-06-27 | Eastman Kodak Co | Polymeric grinding media used in grinding pharmaceutical substances |
US6150366A (en) * | 1998-06-15 | 2000-11-21 | Pfizer Inc. | Ziprasidone formulations |
US8293277B2 (en) * | 1998-10-01 | 2012-10-23 | Alkermes Pharma Ireland Limited | Controlled-release nanoparticulate compositions |
ID29852A (id) * | 1998-11-02 | 2001-10-18 | Elan Corp Plc Cs | Komposisi pelepasan modifikasi multi partikulasi |
DE60001649T2 (de) * | 1999-05-27 | 2003-08-21 | Pfizer Prod Inc | Ziprasidonsuspension |
WO2004037289A2 (fr) * | 2002-10-25 | 2004-05-06 | Pfizer Products Inc. | Nouvelles formulations de depot injectables |
CA2537413A1 (fr) * | 2003-09-02 | 2005-03-10 | Imran Ahmed | Formes posologiques a liberation prolongee de ziprasidone |
US20080193542A1 (en) * | 2005-04-13 | 2008-08-14 | Pfizer Inc. | Injectable Deopot Formulations and Methods For Providing Sustained Release of Nanoparticle Compositions |
-
2006
- 2006-06-19 EA EA200800092A patent/EA200800092A1/ru unknown
- 2006-06-19 WO PCT/US2006/023695 patent/WO2007027273A1/fr active Application Filing
- 2006-06-19 SG SG201004372-7A patent/SG162811A1/en unknown
- 2006-06-19 AU AU2006285349A patent/AU2006285349A1/en not_active Abandoned
- 2006-06-19 KR KR1020087001338A patent/KR20080024206A/ko not_active Application Discontinuation
- 2006-06-19 BR BRPI0612297-3A patent/BRPI0612297A2/pt not_active IP Right Cessation
- 2006-06-19 CA CA002613474A patent/CA2613474A1/fr not_active Abandoned
- 2006-06-19 CN CN2010102092071A patent/CN101879140A/zh active Pending
- 2006-06-19 EP EP06773467A patent/EP1901722A4/fr not_active Withdrawn
-
2007
- 2007-12-12 IL IL188093A patent/IL188093A0/en unknown
- 2007-12-21 NO NO20076628A patent/NO20076628L/no not_active Application Discontinuation
-
2008
- 2008-09-16 HK HK08110215A patent/HK1117060A1/xx unknown
Also Published As
Publication number | Publication date |
---|---|
EP1901722A4 (fr) | 2011-06-15 |
AU2006285349A1 (en) | 2007-03-08 |
IL188093A0 (en) | 2008-03-20 |
EP1901722A1 (fr) | 2008-03-26 |
NO20076628L (no) | 2008-03-12 |
KR20080024206A (ko) | 2008-03-17 |
EA200800092A1 (ru) | 2008-06-30 |
SG162811A1 (en) | 2010-07-29 |
HK1117060A1 (en) | 2009-01-09 |
WO2007027273A1 (fr) | 2007-03-08 |
CN101879140A (zh) | 2010-11-10 |
BRPI0612297A2 (pt) | 2010-11-03 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
EEER | Examination request | ||
FZDE | Discontinued |
Effective date: 20130619 |