CA2459789A1 - Esters analogues de 3-desoxy-vitamine d3 - Google Patents
Esters analogues de 3-desoxy-vitamine d3 Download PDFInfo
- Publication number
- CA2459789A1 CA2459789A1 CA002459789A CA2459789A CA2459789A1 CA 2459789 A1 CA2459789 A1 CA 2459789A1 CA 002459789 A CA002459789 A CA 002459789A CA 2459789 A CA2459789 A CA 2459789A CA 2459789 A1 CA2459789 A1 CA 2459789A1
- Authority
- CA
- Canada
- Prior art keywords
- compound
- formula
- group
- desoxy
- alkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C401/00—Irradiation products of cholesterol or its derivatives; Vitamin D derivatives, 9,10-seco cyclopenta[a]phenanthrene or analogues obtained by chemical preparation without irradiation
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/02—Nutrients, e.g. vitamins, minerals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/12—Drugs for disorders of the metabolism for electrolyte homeostasis
- A61P3/14—Drugs for disorders of the metabolism for electrolyte homeostasis for calcium homeostasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/18—Drugs for disorders of the endocrine system of the parathyroid hormones
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Physical Education & Sports Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Rheumatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Nutrition Science (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
La présente invention concerne des composés de formule (I) ou un sel de ces composés. Dans ladite formule, la ligne en pointillés, R?1¿, R?2¿, R?3¿, R?4¿ et L portent la signification donnée dans les revendications. L'invention concerne par ailleurs l'utilisation des ces composés ou sels en tant que médicaments.
Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US32387001P | 2001-09-21 | 2001-09-21 | |
US32395701P | 2001-09-21 | 2001-09-21 | |
US60/323,957 | 2001-09-21 | ||
US60/323,870 | 2001-09-21 | ||
PCT/EP2002/010233 WO2003027065A1 (fr) | 2001-09-21 | 2002-09-12 | Esters analogues de 3-desoxy-vitamine d3 |
Publications (1)
Publication Number | Publication Date |
---|---|
CA2459789A1 true CA2459789A1 (fr) | 2003-04-03 |
Family
ID=26984180
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CA002459789A Abandoned CA2459789A1 (fr) | 2001-09-21 | 2002-09-12 | Esters analogues de 3-desoxy-vitamine d3 |
Country Status (14)
Country | Link |
---|---|
EP (1) | EP1430026A1 (fr) |
JP (1) | JP2005503434A (fr) |
KR (1) | KR100628586B1 (fr) |
CN (1) | CN1285573C (fr) |
AU (1) | AU2002338672B2 (fr) |
BR (1) | BR0212719A (fr) |
CA (1) | CA2459789A1 (fr) |
MX (1) | MXPA04002640A (fr) |
PA (1) | PA8554901A1 (fr) |
PE (1) | PE20030429A1 (fr) |
PL (1) | PL370352A1 (fr) |
RU (1) | RU2296121C2 (fr) |
UY (1) | UY27448A1 (fr) |
WO (1) | WO2003027065A1 (fr) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
PL376148A1 (en) * | 2002-10-23 | 2005-12-27 | Leo Pharma A/S | Vitamin d analogues, compositions comprising said analogues and their use |
AU2005289664A1 (en) * | 2004-09-24 | 2006-04-06 | Bioxell S.P.A. | 20-cycloalkyl,26,27-alkyl/haloalkyl vitamin D3 compounds and methods of use thereof |
WO2006051106A1 (fr) | 2004-11-12 | 2006-05-18 | Bioxell Spa | Emploi combiné de dérivés de vitamine d et d'agents antiproliférants pour le traitement de cancers de la vessie |
CN102124301B (zh) | 2008-08-22 | 2014-04-02 | Nxp股份有限公司 | 基于位置的服务 |
CN110339205B (zh) * | 2019-08-19 | 2021-08-24 | 山东德信生物科技有限公司 | 富氢水组合物在抑制六价铬诱导的df-1细胞内质网应激及自噬中的应用 |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SG70010A1 (en) * | 1996-05-23 | 2000-01-25 | Hoffmann La Roche | Fluorinated vitamin d3 analogs |
DE69814109T2 (de) * | 1997-09-08 | 2004-02-26 | F. Hoffmann-La Roche Ag | 1,3-dihydroxy-20,20-dialkyl-vitamin d3 analoga |
US6331642B1 (en) * | 1999-07-12 | 2001-12-18 | Hoffmann-La Roche Inc. | Vitamin D3 analogs |
-
2002
- 2002-09-12 WO PCT/EP2002/010233 patent/WO2003027065A1/fr not_active Application Discontinuation
- 2002-09-12 EP EP02777075A patent/EP1430026A1/fr not_active Withdrawn
- 2002-09-12 JP JP2003530656A patent/JP2005503434A/ja active Pending
- 2002-09-12 BR BR0212719-9A patent/BR0212719A/pt not_active IP Right Cessation
- 2002-09-12 CA CA002459789A patent/CA2459789A1/fr not_active Abandoned
- 2002-09-12 RU RU2004112217/04A patent/RU2296121C2/ru not_active IP Right Cessation
- 2002-09-12 MX MXPA04002640A patent/MXPA04002640A/es active IP Right Grant
- 2002-09-12 KR KR1020047004110A patent/KR100628586B1/ko not_active IP Right Cessation
- 2002-09-12 PL PL02370352A patent/PL370352A1/xx not_active Application Discontinuation
- 2002-09-12 CN CNB028185285A patent/CN1285573C/zh not_active Expired - Fee Related
- 2002-09-12 AU AU2002338672A patent/AU2002338672B2/en not_active Ceased
- 2002-09-18 PA PA20028554901A patent/PA8554901A1/es unknown
- 2002-09-19 PE PE2002000921A patent/PE20030429A1/es not_active Application Discontinuation
- 2002-09-20 UY UY27448A patent/UY27448A1/es not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
PA8554901A1 (es) | 2003-12-10 |
JP2005503434A (ja) | 2005-02-03 |
BR0212719A (pt) | 2004-08-03 |
PE20030429A1 (es) | 2003-05-15 |
RU2296121C2 (ru) | 2007-03-27 |
AU2002338672B2 (en) | 2006-03-09 |
PL370352A1 (en) | 2005-05-16 |
MXPA04002640A (es) | 2004-06-07 |
CN1556795A (zh) | 2004-12-22 |
UY27448A1 (es) | 2003-03-31 |
WO2003027065A1 (fr) | 2003-04-03 |
CN1285573C (zh) | 2006-11-22 |
RU2004112217A (ru) | 2005-07-10 |
EP1430026A1 (fr) | 2004-06-23 |
KR100628586B1 (ko) | 2006-09-26 |
KR20040035853A (ko) | 2004-04-29 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
EEER | Examination request | ||
FZDE | Discontinued |