CA2410935A1 - Novel polyamine analogues as therapeutic and diagnostic agents - Google Patents

Novel polyamine analogues as therapeutic and diagnostic agents Download PDF

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Publication number
CA2410935A1
CA2410935A1 CA002410935A CA2410935A CA2410935A1 CA 2410935 A1 CA2410935 A1 CA 2410935A1 CA 002410935 A CA002410935 A CA 002410935A CA 2410935 A CA2410935 A CA 2410935A CA 2410935 A1 CA2410935 A1 CA 2410935A1
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Prior art keywords
polyamine
analogue
derivative
derivative according
transport
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CA002410935A
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English (en)
French (fr)
Inventor
Nicolaas M. J. Vermeulin
Christine L. O'day
Heather K. Webb
Mark R. Burns
Donald E. Bergstrom
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MediQuest Therapeutics Inc
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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/81—Amides; Imides
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