CA2399509A1 - Melanin-concentrating hormone analogs - Google Patents

Melanin-concentrating hormone analogs Download PDF

Info

Publication number
CA2399509A1
CA2399509A1 CA002399509A CA2399509A CA2399509A1 CA 2399509 A1 CA2399509 A1 CA 2399509A1 CA 002399509 A CA002399509 A CA 002399509A CA 2399509 A CA2399509 A CA 2399509A CA 2399509 A1 CA2399509 A1 CA 2399509A1
Authority
CA
Canada
Prior art keywords
mch
derivative
arg
peptide
arginine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002399509A
Other languages
English (en)
French (fr)
Inventor
Maria Bednarek
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck and Co Inc
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of CA2399509A1 publication Critical patent/CA2399509A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575—Hormones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Toxicology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Nutrition Science (AREA)
  • Veterinary Medicine (AREA)
  • Endocrinology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Zoology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Investigating Or Analysing Biological Materials (AREA)
CA002399509A 2000-02-03 2001-02-01 Melanin-concentrating hormone analogs Abandoned CA2399509A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US17996700P 2000-02-03 2000-02-03
US60/179,967 2000-02-03
PCT/US2001/003293 WO2001057070A1 (en) 2000-02-03 2001-02-01 Melanin-concentrating hormone analogs

Publications (1)

Publication Number Publication Date
CA2399509A1 true CA2399509A1 (en) 2001-08-09

Family

ID=22658736

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002399509A Abandoned CA2399509A1 (en) 2000-02-03 2001-02-01 Melanin-concentrating hormone analogs

Country Status (4)

Country Link
EP (1) EP1255770A4 (enExample)
JP (1) JP2003522184A (enExample)
CA (1) CA2399509A1 (enExample)
WO (1) WO2001057070A1 (enExample)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6221613B1 (en) 1998-12-31 2001-04-24 Synaptic Pharmaceutical Corporation DNA encoding a human melanin concentrating hormone receptor (MCH1) and uses thereof
JP4780365B2 (ja) * 2000-07-05 2011-09-28 武田薬品工業株式会社 Ｍｃｈ受容体アンタゴニスト・アゴニストのスクリーニング方法
DE60143525D1 (de) 2000-07-05 2011-01-05 Takeda Pharmaceutical Verfahren zum screenen von mhc-rezeptorantagonisten oder -agonisten
WO2002097037A2 (en) * 2001-05-31 2002-12-05 Merck & Co., Inc. Melanin-concentrating hormone analogs
JP2004537581A (ja) 2001-08-08 2004-12-16 メルク　エンド　カムパニー　インコーポレーテッド メラニン濃縮ホルモン拮抗物質
US7273846B2 (en) 2002-01-09 2007-09-25 Merck & Co., Inc. Selective melanin-concentrating hormone type-1 receptor agonists
JP2014527801A (ja) * 2011-09-01 2014-10-23 ユニバーシティ オブ サザン カリフォルニア ハイスループットペプチドミメティックを調製するための方法、経口バイオアベイラブルな薬物およびそれを含有する組成物

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5049655A (en) * 1989-03-22 1991-09-17 The Salk Institute For Biological Studies Melanin-concentrating hormones
US5849708A (en) * 1995-06-06 1998-12-15 Joslin Diabetes Center, Inc. Promotion of eating behavior

Also Published As

Publication number Publication date
WO2001057070A1 (en) 2001-08-09
EP1255770A4 (en) 2004-12-08
EP1255770A1 (en) 2002-11-13
JP2003522184A (ja) 2003-07-22

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Legal Events

Date Code Title Description
EEER Examination request
FZDE Dead