CA2242097A1 - Imidazotriazolopyrimidines, procedes pour les preparer, et leur utilisation en tant que compositions pharmaceutiques - Google Patents

Imidazotriazolopyrimidines, procedes pour les preparer, et leur utilisation en tant que compositions pharmaceutiques Download PDF

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Publication number
CA2242097A1
CA2242097A1 CA002242097A CA2242097A CA2242097A1 CA 2242097 A1 CA2242097 A1 CA 2242097A1 CA 002242097 A CA002242097 A CA 002242097A CA 2242097 A CA2242097 A CA 2242097A CA 2242097 A1 CA2242097 A1 CA 2242097A1
Authority
CA
Canada
Prior art keywords
preparing
pharmaceutical compositions
imidazotriazolopyrimidines
imidazotriazolopyrimidinone
fundamental
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
CA002242097A
Other languages
English (en)
Other versions
CA2242097C (fr
Inventor
Ulrike Kuefner-Muehl
Werner Kummer
Gerald Pohl
Wolfram Gaida
Erich Lehr
Joachim Mierau
Thomas Weiser
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Boehringer Ingelheim International GmbH
Original Assignee
Boehringer Ingelheim International GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to DE19629378A priority Critical patent/DE19629378A1/de
Priority claimed from DE19629378A external-priority patent/DE19629378A1/de
Priority to PT97933683T priority patent/PT880524E/pt
Priority to IL12645397A priority patent/IL126453A0/xx
Priority to DE59701467T priority patent/DE59701467D1/de
Priority to BR9710747A priority patent/BR9710747A/pt
Priority to AT97933683T priority patent/ATE191913T1/de
Priority to CZ982654A priority patent/CZ265498A3/cs
Priority to JP10505626A priority patent/JP3020281B2/ja
Priority to EP99119410A priority patent/EP0978517A3/fr
Priority to PCT/EP1997/003841 priority patent/WO1998003511A1/fr
Priority to ES97933683T priority patent/ES2147453T3/es
Priority to CA002256736A priority patent/CA2256736A1/fr
Priority to AU36955/97A priority patent/AU3695597A/en
Priority to EP97933683A priority patent/EP0880524B1/fr
Priority to CN97194506A priority patent/CN1219936A/zh
Priority to HU9902311A priority patent/HUP9902311A3/hu
Priority to PL97328824A priority patent/PL328824A1/xx
Priority to TR1998/01659T priority patent/TR199801659T2/xx
Priority to ZA976331A priority patent/ZA976331B/xx
Priority to SK1144-98A priority patent/SK114498A3/sk
Priority to EE9800451A priority patent/EE9800451A/xx
Priority to DK97933683T priority patent/DK0880524T3/da
Priority to HR19629378.2A priority patent/HRP970395A2/hr
Priority to IDP972495A priority patent/ID19106A/id
Application filed by Boehringer Ingelheim International GmbH filed Critical Boehringer Ingelheim International GmbH
Priority to CA002242097A priority patent/CA2242097C/fr
Priority to BG102707A priority patent/BG102707A/xx
Priority to NO983860A priority patent/NO983860L/no
Priority to ZA9808189A priority patent/ZA988189B/xx
Priority to PL98329578A priority patent/PL329578A1/xx
Priority to BR9900187-0A priority patent/BR9900187A/pt
Priority to AU17418/99A priority patent/AU1741899A/en
Priority to IDP990618D priority patent/ID23607A/id
Publication of CA2242097A1 publication Critical patent/CA2242097A1/fr
Priority to US09/559,806 priority patent/US6492377B1/en
Priority to GR20000401543T priority patent/GR3033842T3/el
Publication of CA2242097C publication Critical patent/CA2242097C/fr
Application granted granted Critical
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/14—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CA002242097A 1996-07-20 1998-06-26 Imidazotriazolopyrimidines, procedes pour les preparer, et leur utilisation en tant que compositions pharmaceutiques Expired - Fee Related CA2242097C (fr)

Priority Applications (34)

Application Number Priority Date Filing Date Title
DE19629378A DE19629378A1 (de) 1996-07-20 1996-07-20 Neue Triazolopurine, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
CN97194506A CN1219936A (zh) 1996-07-20 1997-07-17 新的三唑并嘌呤、其制备方法及其作为药品的用途
DE59701467T DE59701467D1 (de) 1996-07-20 1997-07-17 Adenosin-antagonisten, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel
BR9710747A BR9710747A (pt) 1996-07-20 1997-07-17 Novas triazolopurinas processos para a sua prepara-Æo e seu emprego como medicamento
AT97933683T ATE191913T1 (de) 1996-07-20 1997-07-17 Adenosin-antagonisten, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel
CZ982654A CZ265498A3 (cs) 1996-07-20 1997-07-17 Triazolové deriváty, způsob jejich výroby a farmaceutický prostředek s jejich obsahem
JP10505626A JP3020281B2 (ja) 1996-07-20 1997-07-17 新規なトリアゾロプリン類、その調製方法及び医薬組成物としての使用
EP99119410A EP0978517A3 (fr) 1996-07-20 1997-07-17 Triszolopurines, procédé pour leur préparation et leur application comme médicaments
PCT/EP1997/003841 WO1998003511A1 (fr) 1996-07-20 1997-07-17 Nouvelles triazolopurines, procede pour les preparer et leur utilisation comme medicaments
ES97933683T ES2147453T3 (es) 1996-07-20 1997-07-17 Antagonistas de adenosina, procedimiento para su preparacion y su uso como medicamentos.
CA002256736A CA2256736A1 (fr) 1996-07-20 1997-07-17 Nouvelles triazolopurines, procede pour les preparer et leur utilisation comme medicaments
AU36955/97A AU3695597A (en) 1996-07-20 1997-07-17 New triazolopurines, method of preparing them and their use as drugs
EP97933683A EP0880524B1 (fr) 1996-07-20 1997-07-17 Antagonistes d'adenosine, procede pour les preparer et leur utilisation comme medicaments
DK97933683T DK0880524T3 (da) 1996-07-20 1997-07-17 Adenosinantagonister, fremgangsmåde til fremstilling deraf og deres anvendelse som medikamenter
HU9902311A HUP9902311A3 (en) 1996-07-20 1997-07-17 New triazolopurines, method of preparing them and their use as drugs
PL97328824A PL328824A1 (en) 1996-07-20 1997-07-17 Novel triazolopurines, method of obtaining them and their application as drugs
TR1998/01659T TR199801659T2 (xx) 1996-07-20 1997-07-17 Yeni triazolopurinler, haz�rlama y�ntemi, ila� olarak kullan�m�.
ZA976331A ZA976331B (en) 1996-07-20 1997-07-17 New imidazotriazolopyrimidines processes for their preparation and their use as pharmaceutical compositions
PT97933683T PT880524E (pt) 1996-07-20 1997-07-17 Antagonistas de adenosina processo para a sua preparacao e sua utilizacao como medicamentos
EE9800451A EE9800451A (et) 1996-07-20 1997-07-17 Uued imidasotriasolopürimidiinid, nende valmistamismeetod ja kasutamine ravimainetena
IL12645397A IL126453A0 (en) 1996-07-20 1997-07-17 New triazolopurines method of preparing them and their use as drugs
SK1144-98A SK114498A3 (en) 1996-07-20 1997-07-17 Imidazo triazolo pyrimidinone derivatives, method of preparing them and their use
HR19629378.2A HRP970395A2 (en) 1996-07-20 1997-07-18 New triazolopurines, method for preparing them and their use as drugs
IDP972495A ID19106A (id) 1996-07-20 1997-07-18 Senyawa-senyawa triazolopurina baru dan proses-proses pembuatannya serta penggunaannya sebagai komposisi farmasi
CA002242097A CA2242097C (fr) 1996-07-20 1998-06-26 Imidazotriazolopyrimidines, procedes pour les preparer, et leur utilisation en tant que compositions pharmaceutiques
BG102707A BG102707A (en) 1996-07-20 1998-08-20 New triazolopurinpurines, method for their preparation and appplication as medicamentous forms
NO983860A NO983860L (no) 1996-07-20 1998-08-21 Nye triazolopuriner, fremgangsmÕte for deres fremstilling og deres anvendelse som legemidler
ZA9808189A ZA988189B (en) 1998-06-25 1998-09-08 New imidazotriazolopyrimidines, processes for preparing them and their use as pharmaceutical compositions.
PL98329578A PL329578A1 (en) 1998-06-25 1998-11-06 Derivatives of imidazotriazolepyrimidine, method of obtaining them and their application as drugs
BR9900187-0A BR9900187A (pt) 1998-06-25 1999-01-27 Novas imidazotriazolpirimidinonas, processo para a sua preparação e seu emprego como medicamento
AU17418/99A AU1741899A (en) 1996-07-20 1999-02-19 New imidazotriazolopyrimidinones, processes for preparing them and their use as pharmaceutical compositions
IDP990618D ID23607A (id) 1998-06-25 1999-06-25 Imidazotriazolopirimidinon, proses pembuatannya dan penggunaannya sebagai komposisi sediaan farmasi
US09/559,806 US6492377B1 (en) 1998-06-25 2000-04-26 Imidazotriazolopyrimidines with adenosine-antagonistic activity
GR20000401543T GR3033842T3 (en) 1996-07-20 2000-06-30 New triazolopurines, method of preparing them and their use as drugs

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
DE19629378A DE19629378A1 (de) 1996-07-20 1996-07-20 Neue Triazolopurine, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
AU36955/97A AU3695597A (en) 1996-07-20 1997-07-17 New triazolopurines, method of preparing them and their use as drugs
US9058798P 1998-06-25 1998-06-25
CA002242097A CA2242097C (fr) 1996-07-20 1998-06-26 Imidazotriazolopyrimidines, procedes pour les preparer, et leur utilisation en tant que compositions pharmaceutiques

Publications (2)

Publication Number Publication Date
CA2242097A1 true CA2242097A1 (fr) 1999-12-26
CA2242097C CA2242097C (fr) 2003-05-13

Family

ID=32966498

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002242097A Expired - Fee Related CA2242097C (fr) 1996-07-20 1998-06-26 Imidazotriazolopyrimidines, procedes pour les preparer, et leur utilisation en tant que compositions pharmaceutiques

Country Status (1)

Country Link
CA (1) CA2242097C (fr)

Also Published As

Publication number Publication date
CA2242097C (fr) 2003-05-13

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