CA2056009A1 - Heterocyclically substituted piperazinoalkylbenzoxazine and piperazinolkylbenzothiazine compounds, processes for preparing them, and medicaments containing them - Google Patents

Heterocyclically substituted piperazinoalkylbenzoxazine and piperazinolkylbenzothiazine compounds, processes for preparing them, and medicaments containing them

Info

Publication number
CA2056009A1
CA2056009A1 CA002056009A CA2056009A CA2056009A1 CA 2056009 A1 CA2056009 A1 CA 2056009A1 CA 002056009 A CA002056009 A CA 002056009A CA 2056009 A CA2056009 A CA 2056009A CA 2056009 A1 CA2056009 A1 CA 2056009A1
Authority
CA
Canada
Prior art keywords
denotes
formula
lower alkyl
compound
group
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002056009A
Other languages
English (en)
French (fr)
Inventor
Daniel Jasserand
Francois Floc'h
Richard White
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Abbott Products GmbH
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of CA2056009A1 publication Critical patent/CA2056009A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/10—1,4-Thiazines; Hydrogenated 1,4-thiazines
    • C07D279/14—1,4-Thiazines; Hydrogenated 1,4-thiazines condensed with carbocyclic rings or ring systems
    • C07D279/16—1,4-Thiazines; Hydrogenated 1,4-thiazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/34—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings
    • C07D265/36—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings condensed with one six-membered ring

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Immunology (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Plural Heterocyclic Compounds (AREA)
CA002056009A 1990-11-24 1991-11-22 Heterocyclically substituted piperazinoalkylbenzoxazine and piperazinolkylbenzothiazine compounds, processes for preparing them, and medicaments containing them Abandoned CA2056009A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DEP4037427.0 1990-11-24
DE4037427A DE4037427A1 (de) 1990-11-24 1990-11-24 Heterocyclisch substituierte piperazinoalkylbenzoxazin und -thiazin-verbindungen sowie verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel

Publications (1)

Publication Number Publication Date
CA2056009A1 true CA2056009A1 (en) 1992-05-25

Family

ID=6418854

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002056009A Abandoned CA2056009A1 (en) 1990-11-24 1991-11-22 Heterocyclically substituted piperazinoalkylbenzoxazine and piperazinolkylbenzothiazine compounds, processes for preparing them, and medicaments containing them

Country Status (16)

Country Link
EP (1) EP0488008A1 (show.php)
JP (1) JPH05140156A (show.php)
KR (1) KR920009826A (show.php)
CN (1) CN1062140A (show.php)
AU (1) AU644496B2 (show.php)
CA (1) CA2056009A1 (show.php)
DE (1) DE4037427A1 (show.php)
FI (1) FI915518A7 (show.php)
HU (1) HUT62004A (show.php)
IE (1) IE914074A1 (show.php)
IL (1) IL99949A0 (show.php)
MX (1) MX9102192A (show.php)
NO (1) NO914577L (show.php)
PT (1) PT99570A (show.php)
TW (1) TW218876B (show.php)
ZA (1) ZA918341B (show.php)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2667068B1 (fr) * 1990-09-26 1994-09-09 Adir Nouvelles amines alkyl heterocycliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.
AU638154B2 (en) * 1990-10-04 1993-06-17 Suntory Limited Benzoxazine derivative and herbicide containing same as an active ingredient
WO1994018195A1 (fr) * 1993-02-05 1994-08-18 Yamanouchi Pharmaceutical Co., Ltd. Nouveau derive de benzoxazine, medicament le contenant, et son intermediaire
FR2702477B1 (fr) * 1993-03-08 1995-04-28 Synthelabo Dérivés de benzoxazine, leur préparation et leur application en thérapeutique.
FR2755690B1 (fr) * 1996-11-08 1998-12-18 Adir Nouveaux derives aminomethyl heterocycliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1244481A (en) * 1967-11-08 1971-09-02 Wyeth John & Brother Ltd Benzothiazine derivatives and the preparation thereof
EP0186310A1 (en) * 1984-11-28 1986-07-02 Takeda Chemical Industries, Ltd. 1,4-Benzothiazine Derivatives, their production and use
EP0233728A1 (en) * 1986-02-11 1987-08-26 Takeda Chemical Industries, Ltd. 1,4-Benzoxazine derivatives their production and use
FR2667068B1 (fr) * 1990-09-26 1994-09-09 Adir Nouvelles amines alkyl heterocycliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.

Also Published As

Publication number Publication date
IE914074A1 (en) 1992-06-03
HUT62004A (en) 1993-03-29
CN1062140A (zh) 1992-06-24
NO914577L (no) 1992-05-25
HU913482D0 (en) 1992-01-28
TW218876B (show.php) 1994-01-11
JPH05140156A (ja) 1993-06-08
ZA918341B (en) 1992-07-29
AU8809191A (en) 1992-05-28
FI915518A0 (fi) 1991-11-22
MX9102192A (es) 1994-08-31
KR920009826A (ko) 1992-06-25
PT99570A (pt) 1992-10-30
DE4037427A1 (de) 1992-05-27
FI915518L (fi) 1992-05-25
FI915518A7 (fi) 1992-05-25
EP0488008A1 (de) 1992-06-03
NO914577D0 (no) 1991-11-22
AU644496B2 (en) 1993-12-09
IL99949A0 (en) 1992-08-18

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Legal Events

Date Code Title Description
FZDE Discontinued