CA1339897C - Inhibiteurs a base d'acide boronique peptidique pour proteases de type trypsine - Google Patents

Inhibiteurs a base d'acide boronique peptidique pour proteases de type trypsine

Info

Publication number
CA1339897C
CA1339897C CA000616135A CA616135A CA1339897C CA 1339897 C CA1339897 C CA 1339897C CA 000616135 A CA000616135 A CA 000616135A CA 616135 A CA616135 A CA 616135A CA 1339897 C CA1339897 C CA 1339897C
Authority
CA
Canada
Prior art keywords
phe
boroarg
boc
compound
pro
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
CA000616135A
Other languages
English (en)
Inventor
Ashokkumar Bhikkappa Shenvi
Charles Adrian Kettner
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bristol Myers Squibb Pharma Co
Original Assignee
DuPont Merck Pharmaceutical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US07/178,368 external-priority patent/US5187157A/en
Application filed by DuPont Merck Pharmaceutical Co filed Critical DuPont Merck Pharmaceutical Co
Priority to CA000616135A priority Critical patent/CA1339897C/fr
Application granted granted Critical
Publication of CA1339897C publication Critical patent/CA1339897C/fr
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
CA000616135A 1987-06-05 1991-08-16 Inhibiteurs a base d'acide boronique peptidique pour proteases de type trypsine Expired - Fee Related CA1339897C (fr)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CA000616135A CA1339897C (fr) 1987-06-05 1991-08-16 Inhibiteurs a base d'acide boronique peptidique pour proteases de type trypsine

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US5967087A 1987-06-05 1987-06-05
US07/059,670 1987-06-05
US07/178,368 US5187157A (en) 1987-06-05 1988-04-06 Peptide boronic acid inhibitors of trypsin-like proteases
US07/178,368 1988-04-06
CA000568224A CA1328332C (fr) 1987-06-05 1988-05-31 Inhibiteurs de type derives acide boronique de peptides pour des proteases semblables a la trypsine
CA000616135A CA1339897C (fr) 1987-06-05 1991-08-16 Inhibiteurs a base d'acide boronique peptidique pour proteases de type trypsine

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
CA000568224A Division CA1328332C (fr) 1987-06-05 1988-05-31 Inhibiteurs de type derives acide boronique de peptides pour des proteases semblables a la trypsine

Publications (1)

Publication Number Publication Date
CA1339897C true CA1339897C (fr) 1998-06-02

Family

ID=27167960

Family Applications (2)

Application Number Title Priority Date Filing Date
CA000616134A Expired - Fee Related CA1333208C (fr) 1987-06-05 1991-08-16 Peptides contenant de l'acide boronique inhibant les proteases apparentees a la trypsine
CA000616135A Expired - Fee Related CA1339897C (fr) 1987-06-05 1991-08-16 Inhibiteurs a base d'acide boronique peptidique pour proteases de type trypsine

Family Applications Before (1)

Application Number Title Priority Date Filing Date
CA000616134A Expired - Fee Related CA1333208C (fr) 1987-06-05 1991-08-16 Peptides contenant de l'acide boronique inhibant les proteases apparentees a la trypsine

Country Status (1)

Country Link
CA (2) CA1333208C (fr)

Also Published As

Publication number Publication date
CA1333208C (fr) 1994-11-22

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