CA1215981A - Piperidine derivatives, the preparation and use thereof - Google Patents
Piperidine derivatives, the preparation and use thereofInfo
- Publication number
- CA1215981A CA1215981A CA000437468A CA437468A CA1215981A CA 1215981 A CA1215981 A CA 1215981A CA 000437468 A CA000437468 A CA 000437468A CA 437468 A CA437468 A CA 437468A CA 1215981 A CA1215981 A CA 1215981A
- Authority
- CA
- Canada
- Prior art keywords
- formula
- hereinbefore defined
- alkyl
- compound
- represent
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/04—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19823235565 DE3235565A1 (de) | 1982-09-25 | 1982-09-25 | Piperidinderivate, ihre herstellung und verwendung |
DEP3235565.3 | 1982-09-25 |
Publications (1)
Publication Number | Publication Date |
---|---|
CA1215981A true CA1215981A (en) | 1986-12-30 |
Family
ID=6174159
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CA000437468A Expired CA1215981A (en) | 1982-09-25 | 1983-09-23 | Piperidine derivatives, the preparation and use thereof |
Country Status (23)
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4601897A (en) * | 1985-11-06 | 1986-07-22 | Pfizer Inc. | Prazosin-pirbuterol combination for bronchodilation |
JPS62212385A (ja) * | 1986-03-13 | 1987-09-18 | Kotobuki Seiyaku Kk | キナゾリン誘導体並びに血圧降下剤及びその製法 |
EP1317258B1 (en) * | 2000-06-28 | 2009-02-11 | Merck & Co., Inc. | Use of allopurinol for the treatment of hypertension |
AU2003251732B2 (en) | 2002-07-01 | 2008-09-18 | Tibotec Pharmaceuticals Ltd. | New mutational profiles in HIV-1 reverse transcriptase correlated with phenotypic drug resistance |
FR2854633B1 (fr) * | 2003-05-07 | 2005-06-24 | Sanofi Synthelabo | Derives de piperidinyl-et piperazinyl-alkylcarbamates, leur preparation et leur application en therapeutique |
FR2866885B1 (fr) * | 2004-02-26 | 2007-08-31 | Sanofi Synthelabo | Derives de piperidinylalkylcarbamates, leur prepation et leur application en therapeutique |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4309541A (en) * | 1978-09-20 | 1982-01-05 | Ciba-Geigy Corporation | Piperidinyl-lactams |
EP0009465A1 (de) * | 1978-09-20 | 1980-04-02 | Ciba-Geigy Ag | N-(1-(4-Amino-2-chinazolinyl)-3- oder -4-piperidyl-lactame, Verfahren zu ihrer Herstellung, sowie pharmazeutische Präparate enthaltend diese Verbindungen |
FR2483920A1 (fr) * | 1980-06-09 | 1981-12-11 | Synthelabo | Nouveaux derives de quinazoline, leur procede de preparation et leur application en therapeutique |
-
1982
- 1982-09-25 DE DE19823235565 patent/DE3235565A1/de not_active Withdrawn
-
1983
- 1983-08-25 EP EP83108375A patent/EP0104445A3/de not_active Withdrawn
- 1983-09-13 SU SU833641410A patent/SU1187720A3/ru active
- 1983-09-14 US US06/531,842 patent/US4539323A/en not_active Expired - Fee Related
- 1983-09-15 FI FI833292A patent/FI833292A7/fi not_active Application Discontinuation
- 1983-09-20 PH PH29564A patent/PH20015A/en unknown
- 1983-09-20 JP JP58174020A patent/JPS5978187A/ja active Pending
- 1983-09-21 IL IL69777A patent/IL69777A/xx unknown
- 1983-09-22 CS CS836919A patent/CS235342B2/cs unknown
- 1983-09-22 GR GR72505A patent/GR78973B/el unknown
- 1983-09-23 CA CA000437468A patent/CA1215981A/en not_active Expired
- 1983-09-23 NO NO833423A patent/NO833423L/no unknown
- 1983-09-23 ES ES525876A patent/ES8501762A1/es not_active Expired
- 1983-09-23 YU YU01921/83A patent/YU192183A/xx unknown
- 1983-09-23 DD DD83255091A patent/DD212517A5/de unknown
- 1983-09-23 PL PL1983243878A patent/PL139590B1/pl unknown
- 1983-09-23 AU AU19396/83A patent/AU561118B2/en not_active Withdrawn - After Issue
- 1983-09-23 PT PT77380A patent/PT77380B/pt unknown
- 1983-09-23 NZ NZ205716A patent/NZ205716A/xx unknown
- 1983-09-23 HU HU833307A patent/HU191637B/hu unknown
- 1983-09-23 ZA ZA837081A patent/ZA837081B/xx unknown
- 1983-09-23 DK DK436583A patent/DK436583A/da not_active Application Discontinuation
- 1983-09-24 KR KR1019830004475A patent/KR840006222A/ko not_active Withdrawn
-
1984
- 1984-07-16 ES ES534351A patent/ES8504182A1/es not_active Expired
- 1984-07-16 ES ES534350A patent/ES534350A0/es active Granted
- 1984-07-16 ES ES534349A patent/ES8504180A1/es not_active Expired
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MKEX | Expiry |