CA1197504A - Process and intermediates for 6'-amino penicillanoyloxymethyl penicillanate 1,1 dioxide - Google Patents

Process and intermediates for 6'-amino penicillanoyloxymethyl penicillanate 1,1 dioxide

Info

Publication number
CA1197504A
CA1197504A CA000430615A CA430615A CA1197504A CA 1197504 A CA1197504 A CA 1197504A CA 000430615 A CA000430615 A CA 000430615A CA 430615 A CA430615 A CA 430615A CA 1197504 A CA1197504 A CA 1197504A
Authority
CA
Canada
Prior art keywords
compound
dioxide
formula
acid
penicillanate
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA000430615A
Other languages
English (en)
French (fr)
Inventor
David L. Hageman
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Ltd Great Britain
Original Assignee
Pfizer Ltd Great Britain
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Ltd Great Britain filed Critical Pfizer Ltd Great Britain
Application granted granted Critical
Publication of CA1197504A publication Critical patent/CA1197504A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
CA000430615A 1982-06-21 1983-06-17 Process and intermediates for 6'-amino penicillanoyloxymethyl penicillanate 1,1 dioxide Expired CA1197504A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US390,465 1982-06-21
US06/390,465 US4375434A (en) 1982-06-21 1982-06-21 Process for 6'-amino-penicillanoyloxymethyl penicillanate 1,1-dioxide

Publications (1)

Publication Number Publication Date
CA1197504A true CA1197504A (en) 1985-12-03

Family

ID=23542564

Family Applications (1)

Application Number Title Priority Date Filing Date
CA000430615A Expired CA1197504A (en) 1982-06-21 1983-06-17 Process and intermediates for 6'-amino penicillanoyloxymethyl penicillanate 1,1 dioxide

Country Status (7)

Country Link
US (1) US4375434A (https=)
EP (1) EP0097489A1 (https=)
JP (2) JPS597194A (https=)
CA (1) CA1197504A (https=)
DK (1) DK283383A (https=)
ES (1) ES8501406A1 (https=)
GR (1) GR77548B (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4478748A (en) * 1981-02-20 1984-10-23 Pfizer Inc. Bis-esters of alkanediols
US4375434A (en) * 1982-06-21 1983-03-01 Pfizer Inc. Process for 6'-amino-penicillanoyloxymethyl penicillanate 1,1-dioxide
US4530792A (en) * 1982-11-01 1985-07-23 Pfizer Inc. Process and intermediates for preparation of 1,1-dioxopenicillanoyloxymethyl 6-beta-aminopenicillanate

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2613172A1 (de) * 1976-03-27 1977-10-06 Bayer Ag Verfahren zur herstellung von penicillinen und cephalosporinen
IE49881B1 (en) 1979-02-13 1986-01-08 Leo Pharm Prod Ltd B-lactam intermediates
DE3064734D1 (en) * 1979-05-02 1983-10-13 Ici Plc Acetals and their preparation
US4244951A (en) * 1979-05-16 1981-01-13 Pfizer Inc. Bis-esters of methanediol with penicillins and penicillanic acid 1,1-dioxide
GB2086880A (en) * 1980-11-12 1982-05-19 Pfizer Ltd Process for Preparing beta -Lactam Antibiotics and Intermediates Therefor
US4375434A (en) * 1982-06-21 1983-03-01 Pfizer Inc. Process for 6'-amino-penicillanoyloxymethyl penicillanate 1,1-dioxide

Also Published As

Publication number Publication date
JPH01117889A (ja) 1989-05-10
DK283383D0 (da) 1983-06-20
JPS597194A (ja) 1984-01-14
DK283383A (da) 1983-12-22
JPH0445514B2 (https=) 1992-07-27
US4375434A (en) 1983-03-01
GR77548B (https=) 1984-09-24
EP0097489A1 (en) 1984-01-04
ES523438A0 (es) 1984-11-16
ES8501406A1 (es) 1984-11-16

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Legal Events

Date Code Title Description
MKEC Expiry (correction)
MKEX Expiry