CA1104131A - 4-desoxy-thiazolo-¬5,4-c|rifamycin derivatives, a process for preparing them and their use as antimicrobial agents - Google Patents

4-desoxy-thiazolo-¬5,4-c|rifamycin derivatives, a process for preparing them and their use as antimicrobial agents

Info

Publication number
CA1104131A
CA1104131A CA326,394A CA326394A CA1104131A CA 1104131 A CA1104131 A CA 1104131A CA 326394 A CA326394 A CA 326394A CA 1104131 A CA1104131 A CA 1104131A
Authority
CA
Canada
Prior art keywords
rifamycin
thiazolo
methyl
deoxy
alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA326,394A
Other languages
English (en)
French (fr)
Inventor
Renato Cricchio
Marisa Berti
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Gruppo Lepetit SpA
Original Assignee
Gruppo Lepetit SpA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gruppo Lepetit SpA filed Critical Gruppo Lepetit SpA
Application granted granted Critical
Publication of CA1104131A publication Critical patent/CA1104131A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains three hetero rings
    • C07D513/18—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CA326,394A 1978-04-27 1979-04-26 4-desoxy-thiazolo-¬5,4-c|rifamycin derivatives, a process for preparing them and their use as antimicrobial agents Expired CA1104131A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT27738A/78 1978-04-27
IT22738/78A IT1111173B (it) 1978-04-27 1978-04-27 Derivati rifamicinici

Publications (1)

Publication Number Publication Date
CA1104131A true CA1104131A (en) 1981-06-30

Family

ID=11199867

Family Applications (1)

Application Number Title Priority Date Filing Date
CA326,394A Expired CA1104131A (en) 1978-04-27 1979-04-26 4-desoxy-thiazolo-¬5,4-c|rifamycin derivatives, a process for preparing them and their use as antimicrobial agents

Country Status (10)

Country Link
US (2) US4212873A (enExample)
EP (1) EP0005140B1 (enExample)
JP (1) JPS54144366A (enExample)
AU (1) AU529476B2 (enExample)
CA (1) CA1104131A (enExample)
DE (2) DE2963915D1 (enExample)
DK (1) DK149860C (enExample)
IE (1) IE47875B1 (enExample)
IT (1) IT1111173B (enExample)
NZ (1) NZ190292A (enExample)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8531887D0 (en) * 1985-12-30 1986-02-05 Lepetit Spa Rifamycin sv derivatives

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1470426A (en) * 1974-08-30 1977-04-14 Lepetit Spa Rifamycins
GB1523198A (en) * 1976-05-28 1978-08-31 Lepetit Spa Thiazolo-rifamycin derivatives
GB1523199A (en) * 1976-05-28 1978-08-31 Lepetit Spa Rifamycin sv derivatives
US4042633A (en) * 1976-06-07 1977-08-16 Gulf Oil Canada Limited Process for preparing diisopropyl ether
CH629212A5 (it) * 1976-10-18 1982-04-15 Erba Farmitalia Procedimento per la preparazione di composti di rifamicina.

Also Published As

Publication number Publication date
AU4545079A (en) 1979-11-01
NZ190292A (en) 1982-03-23
DE2906931A1 (de) 1979-10-31
IT1111173B (it) 1986-01-13
JPS54144366A (en) 1979-11-10
DK172579A (da) 1979-10-28
IE47875B1 (en) 1984-07-11
AU529476B2 (en) 1983-06-09
EP0005140A3 (en) 1979-11-28
IT7822738A0 (it) 1978-04-27
DK149860B (da) 1986-10-13
EP0005140B1 (en) 1982-10-27
DE2963915D1 (en) 1982-12-02
IE790853L (en) 1979-10-27
US4212873A (en) 1980-07-15
DK149860C (da) 1987-12-14
US4234485A (en) 1980-11-18
JPS6318594B2 (enExample) 1988-04-19
EP0005140A2 (en) 1979-11-14

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Legal Events

Date Code Title Description
MKEX Expiry