BRPI0812161A2 - Processo para a preparação do derivado de dibenzo[b,d]azepin-6-ona - Google Patents

Processo para a preparação do derivado de dibenzo[b,d]azepin-6-ona

Info

Publication number
BRPI0812161A2
BRPI0812161A2 BRPI0812161-3A2A BRPI0812161A BRPI0812161A2 BR PI0812161 A2 BRPI0812161 A2 BR PI0812161A2 BR PI0812161 A BRPI0812161 A BR PI0812161A BR PI0812161 A2 BRPI0812161 A2 BR PI0812161A2
Authority
BR
Brazil
Prior art keywords
azepin
ona
dibenzo
derivative
preparing
Prior art date
Application number
BRPI0812161-3A2A
Other languages
English (en)
Inventor
Fabienne Hoffmann-Emery
Roland Jakob-Roetne
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of BRPI0812161A2 publication Critical patent/BRPI0812161A2/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D223/00Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
    • C07D223/14Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D223/18Dibenzazepines; Hydrogenated dibenzazepines
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D225/00Heterocyclic compounds containing rings of more than seven members having one nitrogen atom as the only ring hetero atom
    • C07D225/04Heterocyclic compounds containing rings of more than seven members having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D225/08Heterocyclic compounds containing rings of more than seven members having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems condensed with two six-membered rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
BRPI0812161-3A2A 2007-05-25 2008-05-15 Processo para a preparação do derivado de dibenzo[b,d]azepin-6-ona BRPI0812161A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP07108904 2007-05-25
PCT/EP2008/055937 WO2008145525A2 (en) 2007-05-25 2008-05-15 Process for the preparation of dibenzo [b,d]azepin-6-one derivative

Publications (1)

Publication Number Publication Date
BRPI0812161A2 true BRPI0812161A2 (pt) 2014-12-16

Family

ID=39776364

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0812161-3A2A BRPI0812161A2 (pt) 2007-05-25 2008-05-15 Processo para a preparação do derivado de dibenzo[b,d]azepin-6-ona

Country Status (12)

Country Link
US (1) US7579464B2 (pt)
EP (1) EP2164830B1 (pt)
JP (2) JP5745841B2 (pt)
KR (1) KR101494918B1 (pt)
CN (1) CN101679278B (pt)
AU (1) AU2008257734B2 (pt)
BR (1) BRPI0812161A2 (pt)
CA (1) CA2686645C (pt)
ES (1) ES2422602T3 (pt)
IL (1) IL202016A (pt)
MX (1) MX2009012277A (pt)
WO (1) WO2008145525A2 (pt)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7579464B2 (en) * 2007-05-25 2009-08-25 Hoffmann-La Roche Inc. Process for preparation of enantiomerically pure compounds
US9133126B2 (en) 2012-09-21 2015-09-15 Bristol-Myers Squibb Company Fluoroalkyl dibenzoazepinone compounds
ES2751082T3 (es) * 2015-10-30 2020-03-30 Pipeline Therapeutics Inc Compuestos de dibenzo azepina y su uso en el tratamiento de enfermedades y trastornos óticos

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP3008227B2 (ja) * 1991-12-18 2000-02-14 第一製薬株式会社 メンチル n−(2−フルオロシクロプロピル)カルバメート誘導体及びその製法
US6528505B1 (en) * 1998-06-22 2003-03-04 Elan Pharmaceuticals, Inc. Cyclic amino acid compounds pharmaceutical compositions comprising same and methods for inhibiting β-amyloid peptide release and/or its synthesis by use of such compounds
US7074742B2 (en) * 2000-09-18 2006-07-11 E. I. Du Pont De Nemours And Company Pyridinyl amides and imides for use as fungicides
CA2514267C (en) * 2003-02-04 2011-05-17 F. Hoffmann-La Roche Ag Malonamide derivatives as gamma-secretase inhibitors
SI1711470T1 (sl) * 2003-09-09 2009-08-31 Hoffmann La Roche Derivati malonamida, ki blokirajo aktivnost gama-sekretaze
DE10341699A1 (de) 2003-09-10 2005-04-28 Symrise Gmbh & Co Kg Verfahren zur Herstellung unsymmetrischer Kohlensäureester
CN1894217B (zh) * 2003-10-06 2011-09-21 弗·哈夫曼-拉罗切有限公司 用作γ-分泌酶抑制剂的取代的二苯并氮杂*和苯并二氮杂*
JP2008528514A (ja) * 2005-01-25 2008-07-31 セルジーン・コーポレーション 4−アミノ−2−(3−メチル−2,6−ジオキソピペリジン−3−イル)−イソインドール−1,3−ジオンを使用する方法及び組成物
US7579464B2 (en) * 2007-05-25 2009-08-25 Hoffmann-La Roche Inc. Process for preparation of enantiomerically pure compounds

Also Published As

Publication number Publication date
WO2008145525A3 (en) 2009-08-13
EP2164830A2 (en) 2010-03-24
JP2014037431A (ja) 2014-02-27
US7579464B2 (en) 2009-08-25
CN101679278A (zh) 2010-03-24
MX2009012277A (es) 2009-11-25
IL202016A0 (en) 2010-06-16
CA2686645A1 (en) 2008-12-04
IL202016A (en) 2014-11-30
JP5745841B2 (ja) 2015-07-08
AU2008257734A1 (en) 2008-12-04
KR101494918B1 (ko) 2015-02-23
US20080293933A1 (en) 2008-11-27
CA2686645C (en) 2015-05-05
CN101679278B (zh) 2013-08-14
JP2010527955A (ja) 2010-08-19
AU2008257734B2 (en) 2012-12-06
WO2008145525A2 (en) 2008-12-04
ES2422602T3 (es) 2013-09-12
KR20100016476A (ko) 2010-02-12
EP2164830B1 (en) 2013-05-29

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Legal Events

Date Code Title Description
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 11A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2514 DE 12-03-2019 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.