BRPI0810408A2 - Polimorfos de ibandronaro de sódio - Google Patents
Polimorfos de ibandronaro de sódioInfo
- Publication number
- BRPI0810408A2 BRPI0810408A2 BRPI0810408-5A2A BRPI0810408A BRPI0810408A2 BR PI0810408 A2 BRPI0810408 A2 BR PI0810408A2 BR PI0810408 A BRPI0810408 A BR PI0810408A BR PI0810408 A2 BRPI0810408 A2 BR PI0810408A2
- Authority
- BR
- Brazil
- Prior art keywords
- ibandronaro
- sodium polymorphs
- polymorphs
- sodium
- ibandronaro sodium
- Prior art date
Links
- DGAQECJNVWCQMB-PUAWFVPOSA-M Ilexoside XXIX Chemical compound C[C@@H]1CC[C@@]2(CC[C@@]3(C(=CC[C@H]4[C@]3(CC[C@@H]5[C@@]4(CC[C@@H](C5(C)C)OS(=O)(=O)[O-])C)C)[C@@H]2[C@]1(C)O)C)C(=O)O[C@H]6[C@@H]([C@H]([C@@H]([C@H](O6)CO)O)O)O.[Na+] DGAQECJNVWCQMB-PUAWFVPOSA-M 0.000 title 1
- 229910052708 sodium Inorganic materials 0.000 title 1
- 239000011734 sodium Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
- C07F9/3804—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)] not used, see subgroups
- C07F9/3839—Polyphosphonic acids
- C07F9/3873—Polyphosphonic acids containing nitrogen substituent, e.g. N.....H or N-hydrocarbon group which can be substituted by halogen or nitro(so), N.....O, N.....S, N.....C(=X)- (X =O, S), N.....N, N...C(=X)...N (X =O, S)
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/66—Phosphorus compounds
- A61K31/662—Phosphorus acids or esters thereof having P—C bonds, e.g. foscarnet, trichlorfon
- A61K31/663—Compounds having two or more phosphorus acid groups or esters thereof, e.g. clodronic acid, pamidronic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/12—Drugs for disorders of the metabolism for electrolyte homeostasis
- A61P3/14—Drugs for disorders of the metabolism for electrolyte homeostasis for calcium homeostasis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Physical Education & Sports Medicine (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Molecular Biology (AREA)
- General Chemical & Material Sciences (AREA)
- Biochemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Rheumatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Hematology (AREA)
- Endocrinology (AREA)
- Diabetes (AREA)
- Obesity (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Analysing Materials By The Use Of Radiation (AREA)
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN849CH2007 | 2007-04-19 | ||
IN400CH2008 | 2008-02-15 | ||
US3148808P | 2008-02-26 | 2008-02-26 | |
PCT/US2008/060727 WO2008131160A1 (en) | 2007-04-19 | 2008-04-18 | Ibandronate sodium polymorphs |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0810408A2 true BRPI0810408A2 (pt) | 2014-11-04 |
Family
ID=39577238
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0810408-5A2A BRPI0810408A2 (pt) | 2007-04-19 | 2008-04-18 | Polimorfos de ibandronaro de sódio |
Country Status (8)
Country | Link |
---|---|
US (1) | US20100125149A1 (pt) |
EP (3) | EP2316840A1 (pt) |
JP (1) | JP2010524967A (pt) |
KR (1) | KR20100014728A (pt) |
AU (1) | AU2008242788A1 (pt) |
BR (1) | BRPI0810408A2 (pt) |
NZ (1) | NZ580042A (pt) |
WO (1) | WO2008131160A1 (pt) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP2128166A1 (en) * | 2008-05-20 | 2009-12-02 | Chemo Ibérica, S.A. | Polymorphic forms of Ibandronate sodium and processes for preparation thereof |
TR201110526A2 (tr) * | 2011-01-06 | 2012-07-23 | Bi̇lgi̇ç Mahmut | Kemik hastalıklarının tedavisinde kullanılmak üzere suda çözünebilir farmasötik formülasyonlar. |
TR201110524A2 (tr) * | 2011-01-06 | 2012-07-23 | Bi̇lgi̇ç Mahmut | Kemik hastalıklarının tedavisinde kullanılmak üzere suda çözünebilir yeni formülasyonlar. |
WO2013179305A1 (en) * | 2012-06-01 | 2013-12-05 | Hetero Research Foundation | Ibandronate sodium solid dispersion |
Family Cites Families (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3623397A1 (de) * | 1986-07-11 | 1988-01-14 | Boehringer Mannheim Gmbh | Neue diphosphonsaeurederivate, verfahren zu deren herstellung und diese verbindungen enthaltende arzneimittel |
MX2007000087A (es) * | 2004-06-23 | 2007-11-06 | Teva Pharma | Acido ibandronico solido y cristalino. |
DE602005025977D1 (de) * | 2004-08-23 | 2011-03-03 | Teva Pharma | Kristalline form des ibandronat-natriums und herstellungsverfahren dafür |
US7214818B2 (en) * | 2004-10-29 | 2007-05-08 | Hoffmann-La Roche Inc. | Method for synthesizing bisphosphonate |
HUE042316T2 (hu) | 2005-02-01 | 2019-06-28 | Atnahs Pharma Uk Ltd | Az Ibandronát A polimorf orvosi alkalmazása |
EP2363401A1 (en) | 2005-02-01 | 2011-09-07 | F. Hoffmann-La Roche AG | Ibandronate polymorph B |
WO2007013097A1 (en) * | 2005-07-25 | 2007-02-01 | Natco Pharma Limited | Improved process for the preparation of ibandronate sodium |
WO2007074475A2 (en) | 2005-12-27 | 2007-07-05 | Natco Pharma Limited | Novel polymorphic forms of ibandronate |
EP2046342A4 (en) * | 2006-07-28 | 2011-05-04 | Reddys Lab Ltd Dr | CRYSTALLINE FORM WITH IBANDRONIC ACID AND PROCESS FOR PREPARING THE SAME |
US20090012047A1 (en) * | 2006-11-16 | 2009-01-08 | Eran Turgeman | Crystalline forms of ibandronate sodium |
EP1923394A1 (en) * | 2006-11-16 | 2008-05-21 | Sandoz A/S | Reagent and use thereof for the production of bisphosphonates |
EP2144919B1 (en) * | 2007-04-11 | 2015-12-02 | F. Hoffmann-La Roche AG | Multi step synthesis of ibandronate |
-
2008
- 2008-04-18 EP EP11152244A patent/EP2316840A1/en not_active Withdrawn
- 2008-04-18 BR BRPI0810408-5A2A patent/BRPI0810408A2/pt not_active IP Right Cessation
- 2008-04-18 NZ NZ580042A patent/NZ580042A/en not_active IP Right Cessation
- 2008-04-18 WO PCT/US2008/060727 patent/WO2008131160A1/en active Application Filing
- 2008-04-18 KR KR1020097020552A patent/KR20100014728A/ko not_active Application Discontinuation
- 2008-04-18 EP EP11152192A patent/EP2316841A1/en not_active Withdrawn
- 2008-04-18 JP JP2010504261A patent/JP2010524967A/ja active Pending
- 2008-04-18 EP EP08746196A patent/EP2134731A1/en not_active Withdrawn
- 2008-04-18 US US12/596,518 patent/US20100125149A1/en not_active Abandoned
- 2008-04-18 AU AU2008242788A patent/AU2008242788A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
KR20100014728A (ko) | 2010-02-10 |
EP2316841A1 (en) | 2011-05-04 |
EP2316840A1 (en) | 2011-05-04 |
NZ580042A (en) | 2011-12-22 |
US20100125149A1 (en) | 2010-05-20 |
JP2010524967A (ja) | 2010-07-22 |
WO2008131160A1 (en) | 2008-10-30 |
AU2008242788A1 (en) | 2008-10-30 |
EP2134731A1 (en) | 2009-12-23 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE AS 5A, 6A E 7A ANUIDADES. |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2329 DE 25-08-2015 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013. |
|
B350 | Update of information on the portal [chapter 15.35 patent gazette] |