BRPI0807125A2 - Processo para a preparação de compostos de uréia substituídos por piperidinil - Google Patents
Processo para a preparação de compostos de uréia substituídos por piperidinilInfo
- Publication number
- BRPI0807125A2 BRPI0807125A2 BRPI0807125-0A2A BRPI0807125A BRPI0807125A2 BR PI0807125 A2 BRPI0807125 A2 BR PI0807125A2 BR PI0807125 A BRPI0807125 A BR PI0807125A BR PI0807125 A2 BRPI0807125 A2 BR PI0807125A2
- Authority
- BR
- Brazil
- Prior art keywords
- piperidinil
- preparation
- urea compounds
- compounds replaced
- replaced
- Prior art date
Links
- XSQUKJJJFZCRTK-UHFFFAOYSA-N Urea Chemical class NC(N)=O XSQUKJJJFZCRTK-UHFFFAOYSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/56—Nitrogen atoms
- C07D211/58—Nitrogen atoms attached in position 4
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/92—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with a hetero atom directly attached to the ring nitrogen atom
- C07D211/96—Sulfur atom
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Heart & Thoracic Surgery (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Cardiology (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US88711407P | 2007-01-29 | 2007-01-29 | |
US97217707P | 2007-09-13 | 2007-09-13 | |
PCT/US2008/052196 WO2008094862A1 (en) | 2007-01-29 | 2008-01-28 | Processes for the preparation of piperidinyl-substituted urea compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0807125A2 true BRPI0807125A2 (pt) | 2014-04-08 |
Family
ID=39493517
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0807125-0A2A BRPI0807125A2 (pt) | 2007-01-29 | 2008-01-28 | Processo para a preparação de compostos de uréia substituídos por piperidinil |
Country Status (15)
Country | Link |
---|---|
US (1) | US20080207908A1 (pt) |
EP (1) | EP2125729A1 (pt) |
JP (1) | JP2010516785A (pt) |
KR (1) | KR20090107045A (pt) |
CN (1) | CN101663273A (pt) |
AR (1) | AR065079A1 (pt) |
AU (1) | AU2008210723A1 (pt) |
BR (1) | BRPI0807125A2 (pt) |
CA (1) | CA2675448A1 (pt) |
EA (1) | EA200901063A1 (pt) |
EC (1) | ECSP099599A (pt) |
IL (1) | IL199654A0 (pt) |
MX (1) | MX2009008093A (pt) |
TW (1) | TW200838851A (pt) |
WO (1) | WO2008094862A1 (pt) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20090197916A1 (en) * | 2007-01-29 | 2009-08-06 | Arete Therapeutics, Inc | Soluble epoxide hydrolase inhibitors for treatment of metabolic syndrome and related disorders |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB9216298D0 (en) * | 1991-08-15 | 1992-09-16 | Ici Plc | Piperidine derivatives |
US7081454B2 (en) * | 2001-03-28 | 2006-07-25 | Bristol-Myers Squibb Co. | Tyrosine kinase inhibitors |
JP4648317B2 (ja) * | 2003-08-01 | 2011-03-09 | 中外製薬株式会社 | マロニル−CoAデカルボキシラーゼ阻害剤として有用なピペリジン化合物 |
TW200808723A (en) * | 2006-03-13 | 2008-02-16 | Univ California | Conformationally restricted urea inhibitors of soluble epoxide hydrolase |
-
2008
- 2008-01-28 CN CN200880003369A patent/CN101663273A/zh active Pending
- 2008-01-28 KR KR1020097015884A patent/KR20090107045A/ko not_active Application Discontinuation
- 2008-01-28 MX MX2009008093A patent/MX2009008093A/es not_active Application Discontinuation
- 2008-01-28 AU AU2008210723A patent/AU2008210723A1/en not_active Abandoned
- 2008-01-28 WO PCT/US2008/052196 patent/WO2008094862A1/en active Application Filing
- 2008-01-28 EP EP08728391A patent/EP2125729A1/en not_active Withdrawn
- 2008-01-28 JP JP2009547453A patent/JP2010516785A/ja not_active Withdrawn
- 2008-01-28 CA CA002675448A patent/CA2675448A1/en not_active Abandoned
- 2008-01-28 BR BRPI0807125-0A2A patent/BRPI0807125A2/pt not_active IP Right Cessation
- 2008-01-28 US US12/021,090 patent/US20080207908A1/en not_active Abandoned
- 2008-01-28 EA EA200901063A patent/EA200901063A1/ru unknown
- 2008-01-28 TW TW097103103A patent/TW200838851A/zh unknown
- 2008-01-29 AR ARP080100360A patent/AR065079A1/es unknown
-
2009
- 2009-07-02 IL IL199654A patent/IL199654A0/en unknown
- 2009-08-27 EC EC2009009599A patent/ECSP099599A/es unknown
Also Published As
Publication number | Publication date |
---|---|
AU2008210723A1 (en) | 2008-08-07 |
CA2675448A1 (en) | 2008-08-07 |
TW200838851A (en) | 2008-10-01 |
AR065079A1 (es) | 2009-05-13 |
JP2010516785A (ja) | 2010-05-20 |
CN101663273A (zh) | 2010-03-03 |
KR20090107045A (ko) | 2009-10-12 |
EA200901063A1 (ru) | 2009-12-30 |
EP2125729A1 (en) | 2009-12-02 |
IL199654A0 (en) | 2010-04-15 |
US20080207908A1 (en) | 2008-08-28 |
WO2008094862A1 (en) | 2008-08-07 |
ECSP099599A (es) | 2009-09-29 |
MX2009008093A (es) | 2009-08-12 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08L | Patent application lapsed because of non payment of annual fee [chapter 8.12 patent gazette] |
Free format text: REFERENTE AO NAO RECOLHIMENTO DAS 3A, 4A, 5A E 6A ANUIDADES. |
|
B08I | Publication cancelled [chapter 8.9 patent gazette] |
Free format text: ANULADA A PUBLICACAO CODIGO 8.12 NA RPI NO 2277 DE 26/08/2014 POR TER SIDO INDEVIDA. |
|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE AS 3A, 4A, 5A, 6A, 7A, 8A, 9A, 10A, 11A E 12A ANUIDADES. |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2602 DE 17-11-2020 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013. |