BRPI0821386A2 - Processo para a preparação de r-lansoprazol amorfo estável - Google Patents
Processo para a preparação de r-lansoprazol amorfo estávelInfo
- Publication number
- BRPI0821386A2 BRPI0821386A2 BRPI0821386-0A BRPI0821386A BRPI0821386A2 BR PI0821386 A2 BRPI0821386 A2 BR PI0821386A2 BR PI0821386 A BRPI0821386 A BR PI0821386A BR PI0821386 A2 BRPI0821386 A2 BR PI0821386A2
- Authority
- BR
- Brazil
- Prior art keywords
- lansoprazole
- preparation
- stable amorphous
- amorphous
- stable
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN2489MU2007 | 2007-12-18 | ||
PCT/IN2008/000842 WO2009087672A1 (en) | 2007-12-18 | 2008-12-18 | A process for preparation of stable amorphous r-lansoprazole |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0821386A2 true BRPI0821386A2 (pt) | 2015-06-16 |
Family
ID=40651360
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0821386-0A BRPI0821386A2 (pt) | 2007-12-18 | 2008-12-18 | Processo para a preparação de r-lansoprazol amorfo estável |
Country Status (6)
Country | Link |
---|---|
US (1) | US20100280077A1 (pt) |
EP (1) | EP2222663A1 (pt) |
AU (1) | AU2008346115A1 (pt) |
BR (1) | BRPI0821386A2 (pt) |
NZ (2) | NZ593629A (pt) |
WO (1) | WO2009087672A1 (pt) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TWI289557B (en) * | 1999-06-17 | 2007-11-11 | Takeda Chemical Industries Ltd | A crystal of a hydrate of (R)-2-[[[3-methyl-4-(2,2,2-trifluoroethoxy)-2-pyridyl]methyl]sulfinyl]-1H-benzimidazole |
CA2717578A1 (en) * | 2008-03-18 | 2009-09-24 | Dr. Reddy's Laboratories Ltd. | Dexlansoprazole process and polymorphs |
NZ589150A (en) | 2008-05-14 | 2012-03-30 | Watson Pharma Private Ltd | Stable r (+) -lansoprazole amine salt and a process for preparing the same |
IT1391758B1 (it) * | 2008-11-11 | 2012-01-27 | Dipharma Francis Srl | Procedimento per la preparazione di dexlansoprazolo amorfo |
WO2011004387A2 (en) | 2009-06-18 | 2011-01-13 | Matrix Laboratories Ltd | Process for the preparation of dexlansoprazole polymorphic forms |
EP2663306A4 (en) * | 2011-01-12 | 2014-01-01 | Hetero Research Foundation | POLYMORPHS OF DEXLANSOPRAZOLE SALTS |
WO2013140120A1 (en) | 2012-03-22 | 2013-09-26 | Cipla Limited | Glycerol solvate forms of (r) - 2 - [ [ [3 -methyl -4 (2,2, 2 - trifluoroethoxy) pyridin- 2 - yl] methyl] sulphinyl] - 1h - ben zimidazole |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS6150978A (ja) * | 1984-08-16 | 1986-03-13 | Takeda Chem Ind Ltd | ピリジン誘導体およびその製造法 |
TWI289557B (en) * | 1999-06-17 | 2007-11-11 | Takeda Chemical Industries Ltd | A crystal of a hydrate of (R)-2-[[[3-methyl-4-(2,2,2-trifluoroethoxy)-2-pyridyl]methyl]sulfinyl]-1H-benzimidazole |
CN1117747C (zh) * | 2000-06-19 | 2003-08-13 | 中国科学院成都有机化学研究所 | 光学纯兰索拉唑的制备方法 |
CA2417311C (en) * | 2000-08-04 | 2012-07-10 | Takeda Chemical Industries, Ltd. | Crystalline alkali metal salts of lansoprazole and their production and use |
KR20100002278A (ko) * | 2000-12-01 | 2010-01-06 | 다케다 야쿠힌 고교 가부시키가이샤 | (r)- 또는 (s)-란소프라졸의 결정 |
DE60314105T2 (de) * | 2002-03-05 | 2008-01-24 | Astrazeneca Ab | Alkylammoniumsalze von omeprazol und esomeprazol |
CA2771725C (en) * | 2002-10-16 | 2015-08-18 | Takeda Pharmaceutical Company Limited | Solid preparation comprising a non-toxic base and a proton pump inhibitor |
ES2259269B1 (es) * | 2005-03-03 | 2007-11-01 | Esteve Quimica, S.A. | Procedimiento para la preparacion de derivados de 2-(2-piridilmetilsulfinil)-bencimidazol opticamente activos. |
NZ589150A (en) * | 2008-05-14 | 2012-03-30 | Watson Pharma Private Ltd | Stable r (+) -lansoprazole amine salt and a process for preparing the same |
-
2008
- 2008-12-18 NZ NZ593629A patent/NZ593629A/xx not_active IP Right Cessation
- 2008-12-18 AU AU2008346115A patent/AU2008346115A1/en not_active Abandoned
- 2008-12-18 NZ NZ585944A patent/NZ585944A/en not_active IP Right Cessation
- 2008-12-18 WO PCT/IN2008/000842 patent/WO2009087672A1/en active Application Filing
- 2008-12-18 BR BRPI0821386-0A patent/BRPI0821386A2/pt not_active IP Right Cessation
- 2008-12-18 EP EP08870010A patent/EP2222663A1/en not_active Withdrawn
- 2008-12-18 US US12/808,351 patent/US20100280077A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
AU2008346115A1 (en) | 2009-07-16 |
NZ593629A (en) | 2012-11-30 |
WO2009087672A1 (en) | 2009-07-16 |
NZ585944A (en) | 2011-11-25 |
US20100280077A1 (en) | 2010-11-04 |
EP2222663A1 (en) | 2010-09-01 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
BRPI0911254A2 (pt) | processo para a preparação de um composto | |
BRPI0916609A2 (pt) | Processo para a preparação de um macrociclo | |
BRPI0820733A2 (pt) | Processo para a preparação de macrociclo | |
BRPI0816258A2 (pt) | processo para a preparação de compostos úteis como inibidores de sglt | |
BRPI0810842A2 (pt) | Processo para a carbonilação de dimetil éter | |
BRPI0910916A2 (pt) | Processo para a produção de um dianidroaçúcar | |
BRPI0915572A2 (pt) | processo para a fabricação de epicloroidrina | |
BRPI1015061A2 (pt) | "processo para a preparação contínua de isocianatos" | |
BR112012014490A2 (pt) | processo para a preparação substituída de 1-o-acil-2-desóxi-2-fluoro-4-tio-beta-d-arabinofuranoses | |
BRPI0810067A2 (pt) | Processo para a preparação de capecitabina | |
BRPI0810817A2 (pt) | Processo para a carbonilação de dimetil éter | |
BRPI1013561A8 (pt) | processo para a preparação de alogliptina | |
BRPI0815784A2 (pt) | Processo para a preparação de 1,2-propanodiol | |
BRPI1006679A2 (pt) | "processo para a preparação de um composto de estireno halogenado" | |
BRPI0810850A2 (pt) | Processo para carbonilação de dimetil éter | |
BRPI0812422A2 (pt) | Processo de preparação de um aldeído hidroxiaromático | |
BRPI0816911A2 (pt) | Processo para preparação de 4-aminobut-2-enolidas | |
BRPI0810846A2 (pt) | Processo para carbonilção de dimetil éter | |
BRPI1010128A2 (pt) | "processo para a fabricação do 2,3,3,3 - tetrafluropropeno" | |
BRPI0817747A2 (pt) | Processo para a preparação de derivados de ácido 2-di-halogenoacil-3-amino-acrílico | |
BRPI0811644A2 (pt) | Processo para a produção de pirazóis | |
BRPI0809652A2 (pt) | Processo melhorado para a síntese de solifenacina | |
BRPI0915365A2 (pt) | Processo para a preparação de 2-triflúor-metil-5-alquil-piridinas substituídas na posição 1 | |
BRPI0813960A2 (pt) | Processo para produção de biarilas | |
BRPI1013830A2 (pt) | Processo para a iodação de compostos aromáticos |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application fees: application dismissed [chapter 8.6 patent gazette] |
Free format text: REFERENTE AS 5A, 6A E 7A ANUIDADES. |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2343 DE 01-12-2015 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013. |