BRPI0608185A2 - processo para redução do tamanho de partìcula de aripiprazol - Google Patents
processo para redução do tamanho de partìcula de aripiprazolInfo
- Publication number
- BRPI0608185A2 BRPI0608185A2 BRPI0608185-1A BRPI0608185A BRPI0608185A2 BR PI0608185 A2 BRPI0608185 A2 BR PI0608185A2 BR PI0608185 A BRPI0608185 A BR PI0608185A BR PI0608185 A2 BRPI0608185 A2 BR PI0608185A2
- Authority
- BR
- Brazil
- Prior art keywords
- particle size
- reducing
- aripiprazole
- aripiprazole particle
- micronized
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Medical Preparation Storing Or Oral Administration Devices (AREA)
- Quinoline Compounds (AREA)
Abstract
PROCESSOS PARA REDUçãO DO TAMANHO DE PARTìCULA DE ARIPIPRAZOL. Forma II de aripiprazol micronizado que tem um formato de partícula e é caracterizada por 90% ou mais das partículas terem um tamanho de partícula de aproximadamente 30 pim, e a Forma II de aripiprazol micronizado não ter mais de 10% por peso de aripiprazol do Tipo C, conforme determinado pela difração de raios X e processos para sua obtenção.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US75346605P | 2005-12-22 | 2005-12-22 | |
PCT/US2006/048761 WO2007075871A2 (en) | 2005-12-22 | 2006-12-22 | Processes for reducing particle size of aripiprazole |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0608185A2 true BRPI0608185A2 (pt) | 2009-11-17 |
Family
ID=38218601
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0608185-1A BRPI0608185A2 (pt) | 2005-12-22 | 2006-12-22 | processo para redução do tamanho de partìcula de aripiprazol |
Country Status (7)
Country | Link |
---|---|
US (1) | US20070272777A1 (pt) |
EP (1) | EP1919453A2 (pt) |
JP (1) | JP2008537540A (pt) |
BR (1) | BRPI0608185A2 (pt) |
IL (1) | IL191286A0 (pt) |
TW (1) | TW200800202A (pt) |
WO (1) | WO2007075871A2 (pt) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2550726A1 (en) * | 2003-12-16 | 2005-06-30 | Teva Pharmaceutical Industries Ltd. | Methods of preparing aripiprazole crystalline forms |
US7714129B2 (en) | 2003-12-16 | 2010-05-11 | Teva Pharmaceutical Industries Ltd. | Methods of preparing anhydrous aripiprazole form II |
ATE429906T1 (de) * | 2006-01-05 | 2009-05-15 | Teva Pharma | Trockene aripiprazolformulierungen |
ES2318693T5 (es) * | 2006-01-05 | 2018-10-04 | Teva Pharmaceutical Industries Ltd | Procedimiento de granulación en húmedo para la preparación de composiciones farmacéuticas de aripiprazol |
KR101408370B1 (ko) * | 2012-06-26 | 2014-06-18 | 주식회사지씨비 | 아리피프라졸-유기산 공결정을 함유하는 제제 및 이의 제조 방법 |
AR096131A1 (es) | 2013-04-30 | 2015-12-09 | Otsuka Pharma Co Ltd | Preparado oral sólido que comprende aripiprazol y un método para producir un preparado oral sólido que comprende aripiprazol |
EP2838513B1 (en) * | 2013-04-30 | 2017-04-05 | Otsuka Pharmaceutical Co., Ltd. | Oral solid preparation comprising aripiprazole and method for producing oral solid preparation comprising aripiprazole |
CN105924393A (zh) * | 2016-07-05 | 2016-09-07 | 陕西省食品药品检验所 | 一种阿立哌唑新晶型及其制备方法 |
Family Cites Families (19)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS54130587A (en) * | 1978-03-30 | 1979-10-09 | Otsuka Pharmaceut Co Ltd | Carbostyryl derivative |
US5006528A (en) * | 1988-10-31 | 1991-04-09 | Otsuka Pharmaceutical Co., Ltd. | Carbostyril derivatives |
DE69112917T2 (de) * | 1990-06-15 | 1996-05-15 | Merck & Co Inc | Kristallisationsverfahren zur Verbesserung der Kristallstruktur und -grösse. |
US6221153B1 (en) * | 1998-06-09 | 2001-04-24 | Trevor Percival Castor | Method for producing large crystals of complex molecules |
WO2001070697A1 (en) * | 2000-03-20 | 2001-09-27 | Teva Pharmaceutical Industries Ltd. | Processes for preparing 6-hydroxy-3,4-dihydroquinolinone, cilostazol and n-(4-methoxyphenyl)-3-chloropropionamide |
AR033485A1 (es) * | 2001-09-25 | 2003-12-26 | Otsuka Pharma Co Ltd | Sustancia medicinal de aripiprazol de baja higroscopicidad y proceso para la preparacion de la misma |
DE60302139T3 (de) * | 2003-01-09 | 2011-02-24 | Otsuka Pharmaceutical Co., Ltd. | Verfahren zur herstellung von aripiprazole |
AU2003230192A1 (en) * | 2003-03-21 | 2004-10-11 | Hetero Drugs Limited | Novel crystalline forms of aripiprazole |
WO2004106322A2 (en) * | 2003-04-25 | 2004-12-09 | Cadila Healthcare Limited | Polymorphs of aripiprazole |
US7456181B2 (en) * | 2003-07-25 | 2008-11-25 | Hetero Drugs Limited | Aripiprazole crystalline forms |
US7166418B2 (en) * | 2003-09-03 | 2007-01-23 | Matsushita Electric Industrial Co., Ltd. | Sulfonamide compound, polymer compound, resist material and pattern formation method |
TWI371274B (en) * | 2003-10-23 | 2012-09-01 | Bristol Myers Squibb Co | Process for making sterile aripiprazole of desired mean particle size |
CA2550726A1 (en) * | 2003-12-16 | 2005-06-30 | Teva Pharmaceutical Industries Ltd. | Methods of preparing aripiprazole crystalline forms |
EP1765782A1 (en) * | 2004-02-05 | 2007-03-28 | Teva Pharmaceutical Industries Ltd | Method of making 7-(4-bromobutoxy)-3,4-dihydrocarbostyril |
US20050277650A1 (en) * | 2004-04-20 | 2005-12-15 | Sundaram Venkataraman | Process for preparing aripirazole hydrate |
DE102005048695A1 (de) * | 2004-10-12 | 2006-05-18 | Chemagis Ltd. | Verfahren zur Herstellung und Reinigung von Carbostyrilverbindungen wie beispielsweise Aripiprazol und 7-(4-Halobutoxy)-3,4-dihydro-2(1H)-quinolinonen |
US20060079690A1 (en) * | 2004-10-12 | 2006-04-13 | Vladimir Naddaka | Processes for preparing 7-hydroxy-3,4-dihydro-2(1H)-quinolinone and the use in aripiprazole preparation thereof |
ES2526415T3 (es) * | 2005-03-17 | 2015-01-12 | Synthon B.V. | Comprimidos farmacéuticos de aripiprazol cristalino de tipo II |
WO2006097343A1 (en) * | 2005-03-17 | 2006-09-21 | Synthon B.V. | Process of making crystalline type ii aripiprazole |
-
2006
- 2006-12-22 US US11/644,567 patent/US20070272777A1/en not_active Abandoned
- 2006-12-22 JP JP2007556441A patent/JP2008537540A/ja active Pending
- 2006-12-22 EP EP06845942A patent/EP1919453A2/en not_active Withdrawn
- 2006-12-22 BR BRPI0608185-1A patent/BRPI0608185A2/pt not_active IP Right Cessation
- 2006-12-22 WO PCT/US2006/048761 patent/WO2007075871A2/en active Application Filing
- 2006-12-22 TW TW095148588A patent/TW200800202A/zh unknown
-
2008
- 2008-05-06 IL IL191286A patent/IL191286A0/en unknown
Also Published As
Publication number | Publication date |
---|---|
JP2008537540A (ja) | 2008-09-18 |
WO2007075871A9 (en) | 2007-08-16 |
WO2007075871A2 (en) | 2007-07-05 |
WO2007075871A3 (en) | 2008-04-03 |
TW200800202A (en) | 2008-01-01 |
IL191286A0 (en) | 2009-08-03 |
US20070272777A1 (en) | 2007-11-29 |
EP1919453A2 (en) | 2008-05-14 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 5A E 6A ANUIDADES. |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2211 DE 21/05/2013. |