BRPI0607461A2 - dispositivo para liberação de agonistas de trpv1 - Google Patents

dispositivo para liberação de agonistas de trpv1

Info

Publication number
BRPI0607461A2
BRPI0607461A2 BRPI0607461-8A BRPI0607461A BRPI0607461A2 BR PI0607461 A2 BRPI0607461 A2 BR PI0607461A2 BR PI0607461 A BRPI0607461 A BR PI0607461A BR PI0607461 A2 BRPI0607461 A2 BR PI0607461A2
Authority
BR
Brazil
Prior art keywords
trpv1 agonist
release device
agonist release
delivery devices
drug delivery
Prior art date
Application number
BRPI0607461-8A
Other languages
English (en)
Inventor
Naweed Muhammad
Gene Curtis Jamieson
Keith R Bley
Original Assignee
Neurogesx Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Neurogesx Inc filed Critical Neurogesx Inc
Publication of BRPI0607461A2 publication Critical patent/BRPI0607461A2/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K36/00—Medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicines
    • A61K36/18—Magnoliophyta (angiosperms)
    • A61K36/185—Magnoliopsida (dicotyledons)
    • A61K36/81—Solanaceae (Potato family), e.g. tobacco, nightshade, tomato, belladonna, capsicum or jimsonweed
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
    • A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
    • A61K9/7084—Transdermal patches having a drug layer or reservoir, and one or more separate drug-free skin-adhesive layers, e.g. between drug reservoir and skin, or surrounding the drug reservoir; Liquid-filled reservoir patches
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Natural Medicines & Medicinal Plants (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dermatology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Microbiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Mycology (AREA)
  • Organic Chemistry (AREA)
  • Alternative & Traditional Medicine (AREA)
  • Biotechnology (AREA)
  • Botany (AREA)
  • Medical Informatics (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Materials For Medical Uses (AREA)

Abstract

DISPOSITIVO PARA LIBERAçãO DE AGONISTAS DE TRPV1. São descritas aqui dispositivos de distribuição de fármaco incluindo uma camada de revestimento oclusivo e um depósito de fármaco contendo um agonista de TRPV1 e um solvente não-hidrofílico. O depósito de fármaco pode tomar várias formas, tal como uma matriz polimérica adesiva, reservatório de líquido ou gotículas de micro-reservatório. Métodos de fabricação e uso dos dispositivos de distribuição de fármaco também são descritos.
BRPI0607461-8A 2005-02-14 2006-02-14 dispositivo para liberação de agonistas de trpv1 BRPI0607461A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US65292305P 2005-02-14 2005-02-14
PCT/US2006/005453 WO2006089012A2 (en) 2005-02-14 2006-02-14 Device for delivery of trpv1 agonists

Publications (1)

Publication Number Publication Date
BRPI0607461A2 true BRPI0607461A2 (pt) 2009-09-08

Family

ID=36917039

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0607461-8A BRPI0607461A2 (pt) 2005-02-14 2006-02-14 dispositivo para liberação de agonistas de trpv1

Country Status (11)

Country Link
US (1) US20060204561A1 (pt)
EP (1) EP1858495A2 (pt)
JP (1) JP2008530139A (pt)
KR (1) KR20070121666A (pt)
CN (1) CN101189000A (pt)
AU (1) AU2006214289A1 (pt)
BR (1) BRPI0607461A2 (pt)
CA (1) CA2597651A1 (pt)
NO (1) NO20074680L (pt)
WO (1) WO2006089012A2 (pt)
ZA (1) ZA200707492B (pt)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2004091521A2 (en) 2003-04-10 2004-10-28 Neurogesx, Inc. Methods and compositions for administration of trpv1 agonists
US20060222690A1 (en) * 2005-03-30 2006-10-05 Bley Keith R Low-concentration capsaicin patch and methods for treating neuropathic pain
US7943666B2 (en) * 2006-07-24 2011-05-17 Trinity Laboratories, Inc. Esters of capsaicin for treating pain
BRPI0814697B8 (pt) 2007-07-10 2021-05-25 Agile Therapeutics Inc dispositivo de liberação de fármacos
US20100292660A1 (en) * 2007-07-10 2010-11-18 Agis Kydonieus Dermal delivery device with ultrasonic weld
WO2009142993A1 (en) * 2008-05-21 2009-11-26 The Regents Of The University Of California Topical application of analgesic for pain relief
US9211274B2 (en) 2012-02-01 2015-12-15 Warsaw Orthopedic, Inc. TRPV1 compounds in a biodegradable polymer carrier
EP3086863B2 (en) * 2013-12-24 2023-01-11 The Procter & Gamble Company Cosmetic compositions and methods providing enhanced penetration of skin care actives
US11607026B2 (en) 2014-05-30 2023-03-21 Johnson & Johnson Consumer Inc. Device for delivery of skin care composition
JP2018501194A (ja) * 2014-10-31 2018-01-18 アヴェント インコーポレイテッド 膀胱収縮の抑制に関連する用途のための方法および装置
US10549129B2 (en) 2016-06-24 2020-02-04 The Procter & Gamble Company Cosmetic compositions and methods providing enhanced penetration of skin care actives
JP6635881B2 (ja) * 2016-06-27 2020-01-29 ユニ・チャーム株式会社 温感シート
CN115006374A (zh) * 2022-07-13 2022-09-06 广州文翰生物科技有限公司 香兰基丁醚在制备治疗头屑和体癣产品中的应用

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US4544668A (en) * 1983-07-14 1985-10-01 The Procter & Gamble Company Compounds and compositions useful for producing analgesia
US4564633A (en) * 1983-07-14 1986-01-14 The Procter & Gamble Company Compositions and methods useful for producing analgesia
US4493848A (en) * 1983-07-14 1985-01-15 The Procter & Gamble Company Compositions and methods useful for producing analgesia
US4544669A (en) * 1983-07-14 1985-10-01 The Procter & Gamble Company Compounds and compositions useful for producing analgesia
US4532139A (en) * 1983-07-14 1985-07-30 The Procter & Gamble Company Compounds and compositions useful for producing analgesia
US4599342A (en) * 1984-01-16 1986-07-08 The Procter & Gamble Company Pharmaceutical products providing enhanced analgesia
US4927687A (en) * 1984-10-01 1990-05-22 Biotek, Inc. Sustained release transdermal drug delivery composition
IE58110B1 (en) * 1984-10-30 1993-07-14 Elan Corp Plc Controlled release powder and process for its preparation
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USRE37934E1 (en) * 1986-08-28 2002-12-10 Lts Lohmann Therapie-Systeme Ag Transdermal therapeutic system
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DE69130924T2 (de) * 1990-08-29 1999-08-05 Us Health Capsaicin oder seine derivate oder analoge enthaltendes vogelfutter
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Also Published As

Publication number Publication date
CN101189000A (zh) 2008-05-28
WO2006089012A3 (en) 2007-05-18
EP1858495A2 (en) 2007-11-28
NO20074680L (no) 2007-11-13
JP2008530139A (ja) 2008-08-07
US20060204561A1 (en) 2006-09-14
KR20070121666A (ko) 2007-12-27
ZA200707492B (en) 2009-02-25
CA2597651A1 (en) 2006-08-24
WO2006089012A2 (en) 2006-08-24
AU2006214289A1 (en) 2006-08-24

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Legal Events

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B08L Patent application lapsed because of non payment of annual fee [chapter 8.12 patent gazette]

Free format text: REFERENTE AO NAO RECOLHIMENTO DAS 5A E 8A ANUIDADES.

B08H Application fees: decision cancelled [chapter 8.8 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.12 NA RPI 2260 DE 29/04/2014

B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

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B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2268 DE 24/06/2014.