BRPI0516942A - método e composição para reduzir o peso corporal em um mamìfero - Google Patents
método e composição para reduzir o peso corporal em um mamìferoInfo
- Publication number
- BRPI0516942A BRPI0516942A BRPI0516942-9A BRPI0516942A BRPI0516942A BR PI0516942 A BRPI0516942 A BR PI0516942A BR PI0516942 A BRPI0516942 A BR PI0516942A BR PI0516942 A BRPI0516942 A BR PI0516942A
- Authority
- BR
- Brazil
- Prior art keywords
- body weight
- mammal
- fatty acid
- composition
- estrogen
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/045—Hydroxy compounds, e.g. alcohols; Salts thereof, e.g. alcoholates
- A61K31/05—Phenols
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/20—Carboxylic acids, e.g. valproic acid having a carboxyl group bound to a chain of seven or more carbon atoms, e.g. stearic, palmitic, arachidic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/20—Carboxylic acids, e.g. valproic acid having a carboxyl group bound to a chain of seven or more carbon atoms, e.g. stearic, palmitic, arachidic acids
- A61K31/201—Carboxylic acids, e.g. valproic acid having a carboxyl group bound to a chain of seven or more carbon atoms, e.g. stearic, palmitic, arachidic acids having one or two double bonds, e.g. oleic, linoleic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/20—Carboxylic acids, e.g. valproic acid having a carboxyl group bound to a chain of seven or more carbon atoms, e.g. stearic, palmitic, arachidic acids
- A61K31/202—Carboxylic acids, e.g. valproic acid having a carboxyl group bound to a chain of seven or more carbon atoms, e.g. stearic, palmitic, arachidic acids having three or more double bonds, e.g. linolenic
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/357—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having two or more oxygen atoms in the same ring, e.g. crown ethers, guanadrel
- A61K31/36—Compounds containing methylenedioxyphenyl groups, e.g. sesamin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A61K31/566—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol having an oxo group in position 17, e.g. estrone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Hematology (AREA)
- Diabetes (AREA)
- Obesity (AREA)
- Child & Adolescent Psychology (AREA)
- Nutrition Science (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
Abstract
MéTODO E COMPOSIçãO PARA REDUZIR O PESO CORPORAL EM UM MAMìFERO. A invenção refere-se a composições e métodos para reduzir o peso corporal de um mamífero. A presente invenção é voltada para métodos para reduzir o peso corporal em um mamífero que compreende a administração de quantidades terapeuticamente eficazes de um éster de ácido graxo de um estrogênio ou de um derivado de estrogênio e um ácido graxo, e um composto termogênico. Além disso, a presente invenção é voltada para composições que compreendem um éster de ácido graxo de um estrogênio ou de um derivado de estrogênio e um ácido graxo, e um composto termogênico.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US10/969,249 US20060084637A1 (en) | 2004-10-18 | 2004-10-18 | Methods of using fatty-acid esters of estrogens and thermogenic compounds for reducing the body weight of a mammal and compositions containing the same |
PCT/EP2005/011155 WO2006042733A2 (en) | 2004-10-18 | 2005-10-17 | Methods of using fatty-acid esters of estrogens and thermogenic compounds for reducing the body weight of a mammal and compositions containing the same |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0516942A true BRPI0516942A (pt) | 2008-09-23 |
Family
ID=36087651
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0516942-9A BRPI0516942A (pt) | 2004-10-18 | 2005-10-17 | método e composição para reduzir o peso corporal em um mamìfero |
Country Status (9)
Country | Link |
---|---|
US (2) | US20060084637A1 (pt) |
EP (1) | EP1812111A2 (pt) |
JP (1) | JP2008516920A (pt) |
KR (1) | KR20070084319A (pt) |
CN (1) | CN101080250A (pt) |
BR (1) | BRPI0516942A (pt) |
CA (1) | CA2584385A1 (pt) |
MX (1) | MX2007004574A (pt) |
WO (1) | WO2006042733A2 (pt) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2008147373A2 (en) * | 2006-06-26 | 2008-12-04 | Manhattan Pharmaceuticals, Inc. | Methods and compositions for reducing body weight using an estrogen fatty ester in an oil |
ES2302449B1 (es) * | 2006-10-30 | 2009-06-12 | Oleoyl-Estrone Developments, S.L. | Monoesteres de estrogenos con acido linoleico conjugado y usos de los mismos. |
US20110098358A1 (en) * | 2008-06-11 | 2011-04-28 | Ricom Corporation | Human beta3 adrenergic receptor ligand, and food or pharmaceutical product containing the same |
US8476227B2 (en) | 2010-01-22 | 2013-07-02 | Ethicon Endo-Surgery, Inc. | Methods of activating a melanocortin-4 receptor pathway in obese subjects |
US9044606B2 (en) | 2010-01-22 | 2015-06-02 | Ethicon Endo-Surgery, Inc. | Methods and devices for activating brown adipose tissue using electrical energy |
JP6479818B2 (ja) * | 2013-05-10 | 2019-03-06 | シーエヌアイシー ファンデーション セントロ ナショナル デ インベスティゲイショネス カーディオバスキュレアス カルロス ザ サード | 骨髄増殖性新生物の治療に適した化合物 |
US10080884B2 (en) | 2014-12-29 | 2018-09-25 | Ethicon Llc | Methods and devices for activating brown adipose tissue using electrical energy |
US10092738B2 (en) | 2014-12-29 | 2018-10-09 | Ethicon Llc | Methods and devices for inhibiting nerves when activating brown adipose tissue |
CN107029237B (zh) * | 2016-02-04 | 2021-06-25 | 康建胜 | 产热增强化合物增强去甲肾上腺素类化合物诱导褐色脂肪细胞产热的应用 |
CA3203170A1 (en) * | 2020-12-24 | 2022-06-30 | Kuen Yong Lee | Fatty acid- modified polymer nanoparticles, and use thereof |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4442113A (en) * | 1981-05-07 | 1984-04-10 | A/S Ferrosan | Long-term weight reduction of obese patients using femoxetine |
ES2094687B1 (es) * | 1994-08-02 | 1997-12-16 | S A L V A T Lab Sa | Combinacion farmaceutica contra la obesidad o el sobrepeso. |
PT771817E (pt) * | 1995-10-30 | 2003-06-30 | Oleoyl Estrone Developments S | Mono-esteres de oleato de estrogenos para o tratamento da obesidade e/ou excesso de peso |
US20030095925A1 (en) * | 1997-10-01 | 2003-05-22 | Dugger Harry A. | Buccal, polar and non-polar spray or capsule containing drugs for treating metabolic disorders |
BR0114836A (pt) * | 2000-10-20 | 2003-07-01 | Pfizer Prod Inc | Agonistas de receptores beta-3 adrenérgicos e suas aplicações |
JP2003013329A (ja) * | 2001-06-26 | 2003-01-15 | Sanai Fujita | 動物骨製繊維及びその製造方法 |
US6821961B2 (en) * | 2001-08-24 | 2004-11-23 | Michael P. Girouard | Monounsaturated fatty acids of at least 20 carbon atoms and perhydrocyclopentanophenanthrene nucleus combination molecules and their use as weight-loss agents |
EP1545484A4 (en) * | 2002-10-05 | 2010-01-13 | Hanmi Pharm Ind Co Ltd | PHARMACEUTICAL COMPOSITION COMPRISING CRYSTALLINE SIBUTRAMINE METHANESULFONATE HEMIHYDRATE |
US20040122033A1 (en) * | 2002-12-10 | 2004-06-24 | Nargund Ravi P. | Combination therapy for the treatment of obesity |
EP1579872B8 (en) * | 2002-12-27 | 2012-11-07 | Takeda Pharmaceutical Company Limited | Body weight gain inhibitor |
-
2004
- 2004-10-18 US US10/969,249 patent/US20060084637A1/en not_active Abandoned
-
2005
- 2005-10-17 CA CA002584385A patent/CA2584385A1/en not_active Abandoned
- 2005-10-17 JP JP2007536116A patent/JP2008516920A/ja active Pending
- 2005-10-17 WO PCT/EP2005/011155 patent/WO2006042733A2/en not_active Application Discontinuation
- 2005-10-17 EP EP05800631A patent/EP1812111A2/en not_active Withdrawn
- 2005-10-17 CN CNA2005800435318A patent/CN101080250A/zh active Pending
- 2005-10-17 KR KR1020077011227A patent/KR20070084319A/ko not_active Application Discontinuation
- 2005-10-17 MX MX2007004574A patent/MX2007004574A/es not_active Application Discontinuation
- 2005-10-17 BR BRPI0516942-9A patent/BRPI0516942A/pt not_active Application Discontinuation
-
2006
- 2006-06-21 US US11/472,694 patent/US20070049569A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
US20060084637A1 (en) | 2006-04-20 |
KR20070084319A (ko) | 2007-08-24 |
WO2006042733A2 (en) | 2006-04-27 |
EP1812111A2 (en) | 2007-08-01 |
JP2008516920A (ja) | 2008-05-22 |
CN101080250A (zh) | 2007-11-28 |
CA2584385A1 (en) | 2006-04-27 |
MX2007004574A (es) | 2007-08-14 |
US20070049569A1 (en) | 2007-03-01 |
WO2006042733A3 (en) | 2006-12-28 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B11A | Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing | ||
B11Y | Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette] | ||
B15K | Others concerning applications: alteration of classification |
Ipc: A61K 31/05 (2006.01), A61P 1/14 (2006.01), A61K 31 |