BRPI0507664A - compostos com atividade antitumor - Google Patents
compostos com atividade antitumorInfo
- Publication number
- BRPI0507664A BRPI0507664A BRPI0507664-1A BRPI0507664A BRPI0507664A BR PI0507664 A BRPI0507664 A BR PI0507664A BR PI0507664 A BRPI0507664 A BR PI0507664A BR PI0507664 A BRPI0507664 A BR PI0507664A
- Authority
- BR
- Brazil
- Prior art keywords
- compounds
- antitumor activity
- antitumor
- optionally
- formula
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7028—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages
- A61K31/7034—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin
- A61K31/704—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin attached to a condensed carbocyclic ring system, e.g. sennosides, thiocolchicosides, escin, daunorubicin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Abstract
COMPOSTOS COM ATIVIDADE ANTITUMOR. A presente invenção refere-se ao uso de compostos de fórmula (I), onde X, Y e Z são definidos como na descrição da invenção, para a preparação de um medicamento antitumor, opcionalmente em combinação com diferentes substâncias biologicamente ativas.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT000230A ITMI20040230A1 (it) | 2004-02-12 | 2004-02-12 | Composti ad attivita' antitumorale |
PCT/EP2005/001257 WO2005077354A1 (en) | 2004-02-12 | 2005-02-08 | Compounds having antitumor activity |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0507664A true BRPI0507664A (pt) | 2007-07-17 |
Family
ID=34856910
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0507664-1A BRPI0507664A (pt) | 2004-02-12 | 2005-02-08 | compostos com atividade antitumor |
Country Status (20)
Country | Link |
---|---|
US (1) | US7652066B2 (pt) |
EP (1) | EP1713461B1 (pt) |
JP (1) | JP2007522165A (pt) |
KR (1) | KR101220331B1 (pt) |
CN (1) | CN1917867B (pt) |
AR (1) | AR047742A1 (pt) |
AT (1) | ATE476973T1 (pt) |
AU (1) | AU2005211906B2 (pt) |
BR (1) | BRPI0507664A (pt) |
CA (1) | CA2556069C (pt) |
CY (1) | CY1111048T1 (pt) |
DE (1) | DE602005022828D1 (pt) |
DK (1) | DK1713461T3 (pt) |
ES (1) | ES2350695T3 (pt) |
HK (1) | HK1099687A1 (pt) |
IT (1) | ITMI20040230A1 (pt) |
PL (1) | PL1713461T3 (pt) |
SI (1) | SI1713461T1 (pt) |
TW (1) | TWI361802B (pt) |
WO (1) | WO2005077354A1 (pt) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US8314144B2 (en) * | 2004-02-12 | 2012-11-20 | Defiante Farmaceutica, S.A. | Compounds having antitumor activity |
WO2008109991A1 (en) | 2007-03-09 | 2008-09-18 | University Health Network | Inhibitors of carnitine palmitoyltransferase and treating cancer |
US8680282B2 (en) | 2007-08-01 | 2014-03-25 | University Health Network | Cyclic inhibitors of carnitine palmitoyltransferase and treating cancer |
JP5474047B2 (ja) * | 2008-04-29 | 2014-04-16 | エフ.ホフマン−ラ ロシュ アーゲー | 4−ジメチルアミノ酪酸誘導体 |
JP2011525530A (ja) * | 2008-06-24 | 2011-09-22 | ダラ・バイオサイエンシズ,インコーポレイテッド | 酵素阻害剤およびその使用 |
JP5746988B2 (ja) * | 2012-02-15 | 2015-07-08 | ライオン株式会社 | カプセル皮膜及びカプセル |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IT1299266B1 (it) * | 1998-05-15 | 2000-02-29 | Sigma Tau Ind Farmaceuti | Inibitori reversibili della carnitina palmitoil trasferasi |
CA2391277A1 (en) * | 1999-11-12 | 2001-05-17 | The Johns Hopkins University School Of Medicine | Treating cancer by increasing intracellular malonyl coa levels |
-
2004
- 2004-02-12 IT IT000230A patent/ITMI20040230A1/it unknown
-
2005
- 2005-02-05 TW TW094103976A patent/TWI361802B/zh not_active IP Right Cessation
- 2005-02-08 KR KR1020067015984A patent/KR101220331B1/ko not_active IP Right Cessation
- 2005-02-08 DK DK05707260.5T patent/DK1713461T3/da active
- 2005-02-08 JP JP2006552526A patent/JP2007522165A/ja not_active Ceased
- 2005-02-08 DE DE602005022828T patent/DE602005022828D1/de active Active
- 2005-02-08 CA CA2556069A patent/CA2556069C/en not_active Expired - Fee Related
- 2005-02-08 WO PCT/EP2005/001257 patent/WO2005077354A1/en not_active Application Discontinuation
- 2005-02-08 US US10/585,972 patent/US7652066B2/en not_active Expired - Fee Related
- 2005-02-08 PL PL05707260T patent/PL1713461T3/pl unknown
- 2005-02-08 BR BRPI0507664-1A patent/BRPI0507664A/pt not_active IP Right Cessation
- 2005-02-08 EP EP05707260A patent/EP1713461B1/en active Active
- 2005-02-08 ES ES05707260T patent/ES2350695T3/es active Active
- 2005-02-08 CN CN2005800046288A patent/CN1917867B/zh not_active Expired - Fee Related
- 2005-02-08 AT AT05707260T patent/ATE476973T1/de active
- 2005-02-08 SI SI200531145T patent/SI1713461T1/sl unknown
- 2005-02-08 AU AU2005211906A patent/AU2005211906B2/en not_active Ceased
- 2005-02-11 AR ARP050100510A patent/AR047742A1/es not_active Application Discontinuation
-
2007
- 2007-05-29 HK HK07105653.0A patent/HK1099687A1/xx not_active IP Right Cessation
-
2010
- 2010-11-03 CY CY20101100990T patent/CY1111048T1/el unknown
Also Published As
Publication number | Publication date |
---|---|
WO2005077354A1 (en) | 2005-08-25 |
CN1917867B (zh) | 2011-03-16 |
CA2556069C (en) | 2013-04-23 |
ITMI20040230A1 (it) | 2004-05-12 |
CA2556069A1 (en) | 2005-08-25 |
CY1111048T1 (el) | 2015-06-11 |
DK1713461T3 (da) | 2010-11-22 |
EP1713461A1 (en) | 2006-10-25 |
TWI361802B (en) | 2012-04-11 |
DE602005022828D1 (de) | 2010-09-23 |
KR20060134059A (ko) | 2006-12-27 |
KR101220331B1 (ko) | 2013-01-09 |
US20080227683A1 (en) | 2008-09-18 |
US7652066B2 (en) | 2010-01-26 |
AR047742A1 (es) | 2006-02-15 |
TW200530154A (en) | 2005-09-16 |
HK1099687A1 (en) | 2007-08-24 |
ATE476973T1 (de) | 2010-08-15 |
AU2005211906B2 (en) | 2009-07-30 |
PL1713461T3 (pl) | 2011-01-31 |
AU2005211906A1 (en) | 2005-08-25 |
EP1713461B1 (en) | 2010-08-11 |
CN1917867A (zh) | 2007-02-21 |
ES2350695T3 (es) | 2011-01-26 |
JP2007522165A (ja) | 2007-08-09 |
SI1713461T1 (sl) | 2010-12-31 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B25D | Requested change of name of applicant approved |
Owner name: DEFIANTE FARMACEUTICA, S.A. (PT) Free format text: ALTERADO DE: DEFIANTE FARMACEUTICA LDA |
|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 10A ANUIDADE. |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2308 DE 31/03/2015. |