BR9914399A - Composto de piridopirazina, processo para sua produção e seu uso - Google Patents
Composto de piridopirazina, processo para sua produção e seu usoInfo
- Publication number
- BR9914399A BR9914399A BR9914399-2A BR9914399A BR9914399A BR 9914399 A BR9914399 A BR 9914399A BR 9914399 A BR9914399 A BR 9914399A BR 9914399 A BR9914399 A BR 9914399A
- Authority
- BR
- Brazil
- Prior art keywords
- production
- compound
- pyridopyrazine
- pyridopyrazine compound
- solvate
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/14—Decongestants or antiallergics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Abstract
"COMPOSTO DE PIRIDOPIRAZINA, PROCESSO PARA SUA PRODUçãO E SEU USO". A invenção provê sal composto de piridopirazina novo da fórmula seguinte e seu cristal, que apresentam solubilidade e estabilidade muito satisfatórias. Mais particularmente, são providos o composto da fórmula acima, seu solvato e seus cristais.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP27444098 | 1998-09-29 | ||
PCT/JP1999/005182 WO2000018768A1 (fr) | 1998-09-29 | 1999-09-22 | Nouveaux sels d'un compose de pyridopyrazine et cristaux desdits sels |
Publications (1)
Publication Number | Publication Date |
---|---|
BR9914399A true BR9914399A (pt) | 2002-01-22 |
Family
ID=17541719
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR9914399-2A BR9914399A (pt) | 1998-09-29 | 1999-09-22 | Composto de piridopirazina, processo para sua produção e seu uso |
Country Status (13)
Country | Link |
---|---|
EP (1) | EP1118615A4 (pt) |
KR (1) | KR20010075287A (pt) |
CN (1) | CN1328555A (pt) |
AU (1) | AU5758199A (pt) |
BR (1) | BR9914399A (pt) |
CA (1) | CA2345362A1 (pt) |
CZ (1) | CZ20011164A3 (pt) |
HK (1) | HK1042896A1 (pt) |
HU (1) | HUP0103947A3 (pt) |
IL (1) | IL142147A0 (pt) |
TR (2) | TR200200971T2 (pt) |
WO (1) | WO2000018768A1 (pt) |
ZA (1) | ZA200102566B (pt) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
MY140561A (en) | 2002-02-20 | 2009-12-31 | Nycomed Gmbh | Dosage form containing pde 4 inhibitor as active ingredient |
EP1511516B1 (en) * | 2002-05-28 | 2008-12-17 | Nycomed GmbH | Topically applicable pharmaceutical preparation |
JP2006501269A (ja) * | 2002-09-16 | 2006-01-12 | アルコン マニュファクチャリング,リミティド | 血管新生を処置するためのpdeivインヒビターの使用 |
EA009985B1 (ru) | 2003-03-10 | 2008-04-28 | Никомед Гмбх | Новый способ получения рофлумиласта |
CA2601250C (en) | 2005-03-16 | 2014-10-28 | Nycomed Gmbh | Taste masked dosage form containing roflumilast |
KR20120073300A (ko) * | 2009-09-30 | 2012-07-04 | 뗑따마르 에스아에스 | 휴대 가방 또는 조끼 |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0008864A1 (en) * | 1978-08-15 | 1980-03-19 | FISONS plc | Pyridopyrazine and quinoxaline derivatives, processes for their preparation, and pharmaceutical compositions containing them |
AU594512B2 (en) * | 1986-09-16 | 1990-03-08 | Merck Patent Gesellschaft Mit Beschrankter Haftung | Hydroxy indole derivatives |
GB9413975D0 (en) * | 1994-07-11 | 1994-08-31 | Fujisawa Pharmaceutical Co | New heterobicyclic derivatives |
-
1999
- 1999-09-22 TR TR2002/00971T patent/TR200200971T2/xx unknown
- 1999-09-22 WO PCT/JP1999/005182 patent/WO2000018768A1/ja not_active Application Discontinuation
- 1999-09-22 AU AU57581/99A patent/AU5758199A/en not_active Abandoned
- 1999-09-22 BR BR9914399-2A patent/BR9914399A/pt not_active IP Right Cessation
- 1999-09-22 KR KR1020017003667A patent/KR20010075287A/ko not_active Application Discontinuation
- 1999-09-22 CA CA002345362A patent/CA2345362A1/en not_active Abandoned
- 1999-09-22 IL IL14214799A patent/IL142147A0/xx unknown
- 1999-09-22 EP EP99944776A patent/EP1118615A4/en not_active Withdrawn
- 1999-09-22 CN CN99813617A patent/CN1328555A/zh active Pending
- 1999-09-22 HU HU0103947A patent/HUP0103947A3/hu unknown
- 1999-09-22 TR TR2001/00893T patent/TR200100893T2/xx unknown
- 1999-09-22 CZ CZ20011164A patent/CZ20011164A3/cs unknown
-
2001
- 2001-03-28 ZA ZA200102566A patent/ZA200102566B/en unknown
-
2002
- 2002-06-11 HK HK02104375.5A patent/HK1042896A1/zh unknown
Also Published As
Publication number | Publication date |
---|---|
CN1328555A (zh) | 2001-12-26 |
WO2000018768A1 (fr) | 2000-04-06 |
EP1118615A4 (en) | 2002-02-27 |
ZA200102566B (en) | 2002-07-18 |
CA2345362A1 (en) | 2000-04-06 |
HUP0103947A3 (en) | 2002-06-28 |
KR20010075287A (ko) | 2001-08-09 |
HUP0103947A2 (hu) | 2002-04-29 |
IL142147A0 (en) | 2002-03-10 |
EP1118615A1 (en) | 2001-07-25 |
HK1042896A1 (zh) | 2002-08-30 |
AU5758199A (en) | 2000-04-17 |
TR200100893T2 (tr) | 2001-11-21 |
CZ20011164A3 (cs) | 2001-12-12 |
TR200200971T2 (tr) | 2002-06-21 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
NL1002835A1 (nl) | Synergistisch stabilisatormengsel. | |
DK0562956T3 (da) | Hidtil ukendte naphthylalkylaminer, fremgangsmåde til fremstilling heraf og farmaceutiske midler, som indeholder dem | |
NO930517L (no) | Benzimidazolylderivater, legemidler inneholdende disse, og fremgangsmaate for deres fremstilling | |
MX9304756A (es) | 9-[(glicilo substituido)amido]-6-desmetil-6-desoxitetraciclinas, metodo para su produccion y composiciones farmaceuticas que las contienen. | |
DK0606046T3 (da) | Arylsulfonamido-substituerede hydroxamsyrederivater | |
MX9302214A (es) | Derivados de taxol y proceso para su preparacion | |
NO963370D0 (no) | Nye mercaptoacetylamido-1,3,4,5-tetrahydro-benzo[cÅazepin-3-on-disulfidderivater som er anvendbare som inhibitorer av enkefalinase og ACE | |
EA200200510A1 (ru) | 4-карбоксиамино-2-этил-1,2,3,4-тетрагидрохинолин в кристаллической форме как ингибитор сетр | |
NO991494D0 (no) | <beta>-sulfonylhydroksaminsyrer som matriksmetalloproteinaseinhibitorer | |
DK0700380T3 (da) | N-Alkylthiopolyaminderivater som radioprotektive midler | |
FI934298A (fi) | Kristallin tiagabine-hydrokloridmonohydrat, dess framstaellning och dess anvaendning | |
BR9503536A (pt) | Composto processo para sua preparação seu uso e composição farmacêutica | |
NO922380L (no) | Substituerte 4-fenyl-4-piperidinkarboksamider med baade lokal anestetisk og analgetisk effekt samt fremgangsmaater for deres fremstilling | |
BR9914399A (pt) | Composto de piridopirazina, processo para sua produção e seu uso | |
NO954609D0 (no) | Niopecotiske syrederivater som antitrombiske forbindelser | |
BR0011339A (pt) | Composto, uso, e processo para preparar o mesmo, composição farmacêutica, e, método para tratar uma condição de doença mediada por metaloproteinase | |
MX9400165A (es) | Derivados de ter-butilergolina, proceso para su produccion y composiciones farmaceuticas que los contienen. | |
DK0861250T3 (da) | Amindin- og isothiourinstofderivater som inhibitorer for nitrogenmonoxidsyntase | |
ATE214051T1 (de) | Substituierte tetrahydropyridinderivate, verfahren zu ihrer herstellung und diese enthaltende arzneimittel | |
DK0745081T3 (da) | Indan-2-mercaptoacetylamiddisulfidderivater, der er anvendelige som enkephalinase-inhibitorer | |
DK0736009T3 (da) | N-oxider af 4-arylpiperaziner og 4-arylpiperidiner som antipsykotiske medikamenter | |
UA26459C2 (uk) | Іhгібітор впливу амілоїдhих білків | |
DK486589D0 (da) | Stabile oxapenem-3-carboxylsyrer og deres anvendelse som beta-lactamase-inhibitorer | |
ES2125474T3 (es) | Derivados de piridazinona o sus sales, procedimentos para su produccion y agentes anti-shock que los contienen. | |
BR9815448A (pt) | Derivados de imino-aza-antraciclinona para o tratamento de amiloidose |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 5A, 6A, 7A E 8A ANUIDADES. |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 1913 DE 04/09/2007. |