BR9912126A - Benximidazóis substituìdos, sua preparação e seu emprego como agente contra protozoários parasitários - Google Patents
Benximidazóis substituìdos, sua preparação e seu emprego como agente contra protozoários parasitáriosInfo
- Publication number
- BR9912126A BR9912126A BR9912126-3A BR9912126A BR9912126A BR 9912126 A BR9912126 A BR 9912126A BR 9912126 A BR9912126 A BR 9912126A BR 9912126 A BR9912126 A BR 9912126A
- Authority
- BR
- Brazil
- Prior art keywords
- preparation
- substituted
- agent against
- benximidazoles
- parasitic protozoa
- Prior art date
Links
- 230000003071 parasitic effect Effects 0.000 title abstract 2
- 125000000217 alkyl group Chemical group 0.000 abstract 2
- 150000001556 benzimidazoles Chemical class 0.000 abstract 2
- 239000003795 chemical substances by application Substances 0.000 abstract 2
- WKBOTKDWSSQWDR-UHFFFAOYSA-N Bromine atom Chemical group [Br] WKBOTKDWSSQWDR-UHFFFAOYSA-N 0.000 abstract 1
- 239000013543 active substance Substances 0.000 abstract 1
- GDTBXPJZTBHREO-UHFFFAOYSA-N bromine Chemical group BrBr GDTBXPJZTBHREO-UHFFFAOYSA-N 0.000 abstract 1
- 229910052794 bromium Chemical group 0.000 abstract 1
- 229910052801 chlorine Inorganic materials 0.000 abstract 1
- 239000000460 chlorine Substances 0.000 abstract 1
- 125000001309 chloro group Chemical group Cl* 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Tropical Medicine & Parasitology (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
Patente de Invenção: <B>"BENZIMIDAZóIS SUBSTITUìDOS, SUA PREPARAçãO E SEU EMPREGO COMO AGENTE CONTRA PROTOZOáRIOS PARASITáRIOS"<D>. A presente invenção refere-se a novos benzimidazóis substituídos, sua preparação e seu emprego como agentes contra protozoários parasitários. As substâncias ativas são caracterizadas pela fórmula (I), na qual X¹ representa cloro ou bromo, R¹ representa hidrogênio ou C~ 1-4~-alquila, R³ representa fluoralquila, R² representa o radical (a), R^ 4^ representa alquila ou fenila substituída, R^ 5^ representa alquila.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19831985A DE19831985A1 (de) | 1998-07-16 | 1998-07-16 | Substituierte Benzimidazole, ihre Herstellung und ihre Verwendung als Mittel gegen parasitäre Protozoen |
PCT/EP1999/004650 WO2000004022A1 (de) | 1998-07-16 | 1999-07-05 | Substituierte benzimidazole, ihre herstellung und ihre verwendung als mittel gegen parasitäre protozoen |
Publications (1)
Publication Number | Publication Date |
---|---|
BR9912126A true BR9912126A (pt) | 2001-04-10 |
Family
ID=7874277
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR9912126-3A BR9912126A (pt) | 1998-07-16 | 1999-07-05 | Benximidazóis substituìdos, sua preparação e seu emprego como agente contra protozoários parasitários |
Country Status (18)
Country | Link |
---|---|
US (3) | US6620833B1 (pt) |
EP (1) | EP1097154B1 (pt) |
JP (1) | JP2002520414A (pt) |
KR (1) | KR100596667B1 (pt) |
CN (1) | CN1117753C (pt) |
AT (1) | ATE251164T1 (pt) |
AU (1) | AU4906799A (pt) |
BR (1) | BR9912126A (pt) |
CA (1) | CA2337351A1 (pt) |
DE (2) | DE19831985A1 (pt) |
DK (1) | DK1097154T3 (pt) |
ES (1) | ES2211119T3 (pt) |
HK (1) | HK1040710B (pt) |
HU (1) | HUP0104820A3 (pt) |
ID (1) | ID26837A (pt) |
NZ (1) | NZ509352A (pt) |
TW (1) | TW584634B (pt) |
WO (1) | WO2000004022A1 (pt) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE10049468A1 (de) * | 2000-10-06 | 2002-04-11 | Bayer Ag | N-Alkoxyalkyl-substituierte Benzimidazole, ihre Herstellung und ihre Verwendung als Mittel gegen parasitäre Protozoen |
DE102004042958A1 (de) * | 2004-09-02 | 2006-03-09 | Bayer Healthcare Ag | Neue antiparasitäre Kombination von Wirkstoffen |
DE102005000746A1 (de) * | 2005-01-05 | 2006-07-13 | Bayer Healthcare Ag | Bekämpfung der Histomoniasis |
DE102009038950A1 (de) | 2009-08-26 | 2011-03-03 | Bayer Animal Health Gmbh | Neue antiparasitäre Kombination von Wirkstoffen |
KR20210056356A (ko) * | 2018-09-06 | 2021-05-18 | 닛폰 스이산 가부시키가이샤 | 연어목 어류의 근육의 융해를 방지하는 방법 |
Family Cites Families (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3271249A (en) * | 1963-06-24 | 1966-09-06 | S B Penick & Co Inc | Dihalobenzimidazoles for poultry disease treatment |
GB1122988A (en) | 1964-10-22 | 1968-08-07 | Fisons Pest Control Ltd | Benzimidazole derivatives |
GB1163711A (en) | 1966-01-13 | 1969-09-10 | Fisons Pest Control Ltd | Substituted Benzimidazoles and Biocidally-Active Compositions |
AU413408B2 (en) | 1966-09-19 | 1971-05-19 | 2-cyanobenzimidazoles | |
DE2040175A1 (de) | 1970-08-13 | 1972-02-17 | Wolfgang Dr Ritter | Verfahren zur Herstellung von N-substituierten N-Chlormethylcarbamidsaeureestern |
DE2119518A1 (de) | 1971-04-22 | 1972-10-26 | Farbenfabriken Bayer Ag, 5090 Leverkusen | Verfahren zur Herstellung von N-substituiertenN-Chlormethylcarbamidsäureestern und -thiolestern |
US3738994A (en) | 1971-08-13 | 1973-06-12 | Merck & Co Inc | 2-cyano-polyhalobenzimidazoles |
FR2521141A1 (fr) | 1982-02-09 | 1983-08-12 | Rhone Poulenc Agrochimie | Nouveaux derives du cyano-2 benzimidazole, leur preparation et leur utilisation comme fongicides |
FR2559150B1 (fr) | 1984-02-06 | 1986-06-27 | Rhone Poulenc Agrochimie | Nouveaux derives du cyano-2 benzimidazole, leur preparation et leur utilisation comme fongicides |
FR2594437A1 (fr) | 1986-02-19 | 1987-08-21 | Rhone Poulenc Agrochimie | Nouveaux derives du cyano-2 benzimidazole, leur preparation, les compositions les contenant et leur utilisation comme fongicide |
NZ221729A (en) | 1986-09-15 | 1989-07-27 | Janssen Pharmaceutica Nv | Imidazolyl methyl-substituted benzimidazole derivatives and pharmaceutical compositions |
DE4237617A1 (de) | 1992-11-06 | 1994-05-11 | Bayer Ag | Verwendung von substituierten Benzimidazolen |
US5331003A (en) | 1993-03-26 | 1994-07-19 | Eli Lilly And Company | Anticoccidial methods |
DE19519821A1 (de) * | 1995-05-31 | 1996-12-05 | Bayer Ag | Mittel gegen parasitäre Protozoen |
IT1282789B1 (it) | 1996-06-07 | 1998-03-31 | Electronic Systems Spa | Dispositivo di misurazione senza contatto di spessore per materiali non metallici in film,fogli,nastri o simili |
-
1998
- 1998-07-16 DE DE19831985A patent/DE19831985A1/de not_active Withdrawn
-
1999
- 1999-07-05 NZ NZ509352A patent/NZ509352A/en unknown
- 1999-07-05 US US09/743,440 patent/US6620833B1/en not_active Expired - Fee Related
- 1999-07-05 AT AT99932812T patent/ATE251164T1/de not_active IP Right Cessation
- 1999-07-05 CN CN99810383A patent/CN1117753C/zh not_active Expired - Fee Related
- 1999-07-05 AU AU49067/99A patent/AU4906799A/en not_active Abandoned
- 1999-07-05 CA CA002337351A patent/CA2337351A1/en not_active Abandoned
- 1999-07-05 JP JP2000560128A patent/JP2002520414A/ja not_active Withdrawn
- 1999-07-05 DK DK99932812T patent/DK1097154T3/da active
- 1999-07-05 BR BR9912126-3A patent/BR9912126A/pt not_active Application Discontinuation
- 1999-07-05 ES ES99932812T patent/ES2211119T3/es not_active Expired - Lifetime
- 1999-07-05 DE DE59907215T patent/DE59907215D1/de not_active Expired - Fee Related
- 1999-07-05 KR KR1020007014939A patent/KR100596667B1/ko not_active IP Right Cessation
- 1999-07-05 WO PCT/EP1999/004650 patent/WO2000004022A1/de active IP Right Grant
- 1999-07-05 EP EP99932812A patent/EP1097154B1/de not_active Expired - Lifetime
- 1999-07-05 HU HU0104820A patent/HUP0104820A3/hu unknown
- 1999-07-05 ID IDW20010111A patent/ID26837A/id unknown
- 1999-07-06 TW TW088111400A patent/TW584634B/zh not_active IP Right Cessation
-
2002
- 2002-03-27 HK HK02102363.3A patent/HK1040710B/zh not_active IP Right Cessation
-
2003
- 2003-07-03 US US10/613,818 patent/US20040010025A1/en not_active Abandoned
-
2006
- 2006-11-17 US US11/601,036 patent/US20070066671A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
CN1315954A (zh) | 2001-10-03 |
WO2000004022A1 (de) | 2000-01-27 |
EP1097154A1 (de) | 2001-05-09 |
KR20010078750A (ko) | 2001-08-21 |
HK1040710A1 (en) | 2002-06-21 |
US20070066671A1 (en) | 2007-03-22 |
NZ509352A (en) | 2003-05-30 |
HK1040710B (zh) | 2004-05-07 |
US6620833B1 (en) | 2003-09-16 |
EP1097154B1 (de) | 2003-10-01 |
DE59907215D1 (de) | 2003-11-06 |
US20040010025A1 (en) | 2004-01-15 |
KR100596667B1 (ko) | 2006-07-06 |
HUP0104820A3 (en) | 2003-12-29 |
ES2211119T3 (es) | 2004-07-01 |
JP2002520414A (ja) | 2002-07-09 |
HUP0104820A2 (hu) | 2002-04-29 |
DE19831985A1 (de) | 2000-01-20 |
ID26837A (id) | 2001-02-15 |
DK1097154T3 (da) | 2003-12-29 |
CA2337351A1 (en) | 2000-01-27 |
CN1117753C (zh) | 2003-08-13 |
AU4906799A (en) | 2000-02-07 |
TW584634B (en) | 2004-04-21 |
ATE251164T1 (de) | 2003-10-15 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B07A | Application suspended after technical examination (opinion) [chapter 7.1 patent gazette] | ||
B09B | Patent application refused [chapter 9.2 patent gazette] |
Free format text: INDEFIRO O PRESENTE PEDIDO DE PATENTE DE ACORDO COM ART. 8O DA LPI. |
|
B09B | Patent application refused [chapter 9.2 patent gazette] |
Free format text: MANTIDO O INDEFERIMENTO UMA VEZ QUE NAO FOI APRESENTADO RECURSO DENTRO DO PRAZO LEGAL. |