BR9810790A - Indole and 2, 3 dihydroindole derivatives, preparation and use thereof - Google Patents
Indole and 2, 3 dihydroindole derivatives, preparation and use thereofInfo
- Publication number
- BR9810790A BR9810790A BR9810790-9A BR9810790A BR9810790A BR 9810790 A BR9810790 A BR 9810790A BR 9810790 A BR9810790 A BR 9810790A BR 9810790 A BR9810790 A BR 9810790A
- Authority
- BR
- Brazil
- Prior art keywords
- indole
- preparation
- derivatives
- dihydroindole derivatives
- dihydroindole
- Prior art date
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Indole Compounds (AREA)
Abstract
<B>"INDOL E DERIVADOS DE 2,3 DIIDROINDOL, PREPARAçAO E UTILIZAçãO DOS MESMOS"<D> A presente invenção refere-se a indol e derivados de 2,3-diidroindol possuindo a fórmula (I), qualquer de seus enantiómeros ou qualquer mistura dos mesmos, ou um sal de adição de ácido dos mesmos, onde A, R^ 1^, R^ 2^, R^ 3^, W, X, Y são como o descrito na descrição. Os compostos são potentes inibidores de recaptação de serotonina e possuem atividade antagonista de receptor 5-HT~ 1A~.<B> "INDOL AND 2,3-DIIDROINDOL DERIVATIVES, PREPARATION AND USE OF THE SAME" <D> The present invention relates to indole and 2,3-dihydroindole derivatives having the formula (I), any of its enantiomers or any mixture thereof, or an acid addition salt thereof, where A, R ^ 1 ^, R ^ 2 ^, R ^ 3 ^, W, X, Y are as described in the description. The compounds are potent serotonin reuptake inhibitors and have 5-HT ~ 1A ~ receptor antagonistic activity.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DK89297 | 1997-07-25 | ||
PCT/DK1998/000336 WO1999005140A1 (en) | 1997-07-25 | 1998-07-20 | Indole and 2,3-dihydroindole derivatives, their preparation and use |
Publications (1)
Publication Number | Publication Date |
---|---|
BR9810790A true BR9810790A (en) | 2000-07-25 |
Family
ID=8098721
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR9810790-9A BR9810790A (en) | 1997-07-25 | 1998-07-20 | Indole and 2, 3 dihydroindole derivatives, preparation and use thereof |
Country Status (13)
Country | Link |
---|---|
CN (3) | CN1286833C (en) |
AR (1) | AR013206A1 (en) |
BR (1) | BR9810790A (en) |
EA (1) | EA001890B1 (en) |
HK (3) | HK1030220A1 (en) |
IL (1) | IL133990A (en) |
IS (1) | IS2024B (en) |
NO (1) | NO318610B1 (en) |
PL (1) | PL190924B1 (en) |
SK (1) | SK284866B6 (en) |
TR (1) | TR200000231T2 (en) |
UA (1) | UA59408C2 (en) |
ZA (1) | ZA986237B (en) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN103420989B (en) * | 2012-05-15 | 2016-03-23 | 华中科技大学 | Benzodioxane derivative and application thereof |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB8830312D0 (en) * | 1988-12-28 | 1989-02-22 | Lundbeck & Co As H | Heterocyclic compounds |
DE4127849A1 (en) * | 1991-08-22 | 1993-02-25 | Merck Patent Gmbh | BENZODIOXAN DERIVATIVES |
FR2692264B1 (en) * | 1992-06-12 | 1994-08-05 | Adir | NOVEL 1,4-DISUBSTITUTED PIPERAZINES, THEIR PREPARATION PROCESS AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM. |
-
1998
- 1998-07-13 AR ARP980103400 patent/AR013206A1/en active IP Right Grant
- 1998-07-14 ZA ZA986237A patent/ZA986237B/en unknown
- 1998-07-20 CN CN 03106002 patent/CN1286833C/en not_active Expired - Fee Related
- 1998-07-20 CN CN 98807554 patent/CN1127501C/en not_active Expired - Fee Related
- 1998-07-20 TR TR2000/00231T patent/TR200000231T2/en unknown
- 1998-07-20 UA UA2000020949A patent/UA59408C2/en unknown
- 1998-07-20 EA EA200000162A patent/EA001890B1/en not_active IP Right Cessation
- 1998-07-20 PL PL338194A patent/PL190924B1/en not_active IP Right Cessation
- 1998-07-20 BR BR9810790-9A patent/BR9810790A/en not_active Application Discontinuation
- 1998-07-20 CN CNB03106003XA patent/CN1293075C/en not_active Expired - Fee Related
- 1998-07-20 IL IL13399098A patent/IL133990A/en not_active IP Right Cessation
- 1998-07-20 SK SK95-2000A patent/SK284866B6/en not_active IP Right Cessation
-
2000
- 2000-01-11 IS IS5334A patent/IS2024B/en unknown
- 2000-01-25 NO NO20000372A patent/NO318610B1/en not_active IP Right Cessation
-
2001
- 2001-02-21 HK HK01101274A patent/HK1030220A1/en not_active IP Right Cessation
-
2004
- 2004-12-13 HK HK04109852A patent/HK1066806A1/en not_active IP Right Cessation
- 2004-12-13 HK HK04109853A patent/HK1066807A1/en not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
UA59408C2 (en) | 2003-09-15 |
NO20000372D0 (en) | 2000-01-25 |
CN1515569A (en) | 2004-07-28 |
CN1293075C (en) | 2007-01-03 |
HK1066807A1 (en) | 2005-04-01 |
AR013206A1 (en) | 2000-12-13 |
IS5334A (en) | 2000-01-11 |
IL133990A0 (en) | 2001-04-30 |
CN1265107A (en) | 2000-08-30 |
TR200000231T2 (en) | 2000-07-21 |
EA200000162A1 (en) | 2000-10-30 |
HK1066806A1 (en) | 2005-04-01 |
CN1286833C (en) | 2006-11-29 |
IS2024B (en) | 2005-08-15 |
PL190924B1 (en) | 2006-02-28 |
HK1030220A1 (en) | 2001-04-27 |
CN1127501C (en) | 2003-11-12 |
SK952000A3 (en) | 2001-03-12 |
SK284866B6 (en) | 2006-01-05 |
IL133990A (en) | 2003-09-17 |
EA001890B1 (en) | 2001-10-22 |
PL338194A1 (en) | 2000-10-09 |
NO318610B1 (en) | 2005-04-18 |
NO20000372L (en) | 2000-03-21 |
ZA986237B (en) | 1999-03-31 |
CN1515568A (en) | 2004-07-28 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B06A | Patent application procedure suspended [chapter 6.1 patent gazette] | ||
B06A | Patent application procedure suspended [chapter 6.1 patent gazette] | ||
B06A | Patent application procedure suspended [chapter 6.1 patent gazette] | ||
B11B | Dismissal acc. art. 36, par 1 of ipl - no reply within 90 days to fullfil the necessary requirements |