TR200000231T2 - Indole and 2,3-dihydroindole derivatives, their preparation and use. - Google Patents

Indole and 2,3-dihydroindole derivatives, their preparation and use.

Info

Publication number
TR200000231T2
TR200000231T2 TR2000/00231T TR200000231T TR200000231T2 TR 200000231 T2 TR200000231 T2 TR 200000231T2 TR 2000/00231 T TR2000/00231 T TR 2000/00231T TR 200000231 T TR200000231 T TR 200000231T TR 200000231 T2 TR200000231 T2 TR 200000231T2
Authority
TR
Turkey
Prior art keywords
indole
preparation
dihydroindole derivatives
formula
dihydroindole
Prior art date
Application number
TR2000/00231T
Other languages
Turkish (tr)
Inventor
Knud Moltzen Ejner
Kristian Perregaard Jens
Mikkelsen Ivan
Garrick Smith Paul
Original Assignee
H. Lundbeck A/S
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by H. Lundbeck A/S filed Critical H. Lundbeck A/S
Publication of TR200000231T2 publication Critical patent/TR200000231T2/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)

Abstract

Mevcut bulus, enantiyomerlerinden herhangi biri veya bunlarin herhangi bir karisimindan olusan formül (I)' e veya A, R1, R2, R3, W, X, Y ve Z' nin tarifte belirtildigi gibi oldugu bunlarin asit ilaveli bir tuzuna sahip indol ve 2,3-dihidroindol türevleri ile ilgilidir. Bilesikler, potansiyel bir sekilde serotoninin yeniden alinmasini önlerler ve 5-HT1A alici antagonist aktivitesi gösterirler. Formül (I)The present invention consists of formula (I) consisting of any of its enantiomers or any combination thereof, or an acid addition salt of A, R1, R2, R3, W, X, Y and Z, as specified in the description, and 2, It relates to 3-dihydroindole derivatives. The compounds potentially prevent re-uptake of serotonin and show 5-HT1A receptor antagonist activity. Formula (I)

TR2000/00231T 1997-07-25 1998-07-20 Indole and 2,3-dihydroindole derivatives, their preparation and use. TR200000231T2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DK89297 1997-07-25

Publications (1)

Publication Number Publication Date
TR200000231T2 true TR200000231T2 (en) 2000-07-21

Family

ID=8098721

Family Applications (1)

Application Number Title Priority Date Filing Date
TR2000/00231T TR200000231T2 (en) 1997-07-25 1998-07-20 Indole and 2,3-dihydroindole derivatives, their preparation and use.

Country Status (13)

Country Link
CN (3) CN1127501C (en)
AR (1) AR013206A1 (en)
BR (1) BR9810790A (en)
EA (1) EA001890B1 (en)
HK (3) HK1030220A1 (en)
IL (1) IL133990A (en)
IS (1) IS2024B (en)
NO (1) NO318610B1 (en)
PL (1) PL190924B1 (en)
SK (1) SK284866B6 (en)
TR (1) TR200000231T2 (en)
UA (1) UA59408C2 (en)
ZA (1) ZA986237B (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN103420989B (en) * 2012-05-15 2016-03-23 华中科技大学 Benzodioxane derivative and application thereof

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8830312D0 (en) * 1988-12-28 1989-02-22 Lundbeck & Co As H Heterocyclic compounds
DE4127849A1 (en) * 1991-08-22 1993-02-25 Merck Patent Gmbh BENZODIOXAN DERIVATIVES
FR2692264B1 (en) * 1992-06-12 1994-08-05 Adir NOVEL 1,4-DISUBSTITUTED PIPERAZINES, THEIR PREPARATION PROCESS AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM.

Also Published As

Publication number Publication date
IS2024B (en) 2005-08-15
HK1066807A1 (en) 2005-04-01
CN1293075C (en) 2007-01-03
CN1127501C (en) 2003-11-12
CN1515569A (en) 2004-07-28
EA001890B1 (en) 2001-10-22
BR9810790A (en) 2000-07-25
IL133990A0 (en) 2001-04-30
IL133990A (en) 2003-09-17
EA200000162A1 (en) 2000-10-30
PL338194A1 (en) 2000-10-09
SK284866B6 (en) 2006-01-05
CN1265107A (en) 2000-08-30
ZA986237B (en) 1999-03-31
PL190924B1 (en) 2006-02-28
NO20000372D0 (en) 2000-01-25
NO318610B1 (en) 2005-04-18
CN1515568A (en) 2004-07-28
HK1066806A1 (en) 2005-04-01
AR013206A1 (en) 2000-12-13
UA59408C2 (en) 2003-09-15
CN1286833C (en) 2006-11-29
HK1030220A1 (en) 2001-04-27
NO20000372L (en) 2000-03-21
IS5334A (en) 2000-01-11
SK952000A3 (en) 2001-03-12

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