BR9611628A - Derivados de pirido [2,3-d] pirimidina e composições medicinais dos mesmos - Google Patents

Derivados de pirido [2,3-d] pirimidina e composições medicinais dos mesmos

Info

Publication number
BR9611628A
BR9611628A BR9611628A BR9611628A BR9611628A BR 9611628 A BR9611628 A BR 9611628A BR 9611628 A BR9611628 A BR 9611628A BR 9611628 A BR9611628 A BR 9611628A BR 9611628 A BR9611628 A BR 9611628A
Authority
BR
Brazil
Prior art keywords
pyrido
pyrimidine derivatives
medicinal compositions
medicinal
compositions
Prior art date
Application number
BR9611628A
Other languages
English (en)
Inventor
Kazuhisa Takayama
Hiroyuki Hisamichi
Masahiro Iwata
Hideki Kubota
Motonori Aoki
Original Assignee
Yamanouchi Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Yamanouchi Pharma Co Ltd filed Critical Yamanouchi Pharma Co Ltd
Publication of BR9611628A publication Critical patent/BR9611628A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
BR9611628A 1995-11-21 1996-11-20 Derivados de pirido [2,3-d] pirimidina e composições medicinais dos mesmos BR9611628A (pt)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
JP30306595 1995-11-21
JP772596 1996-01-19
JP4385396 1996-02-29
JP14186896 1996-06-04
PCT/JP1996/003389 WO1997019078A1 (en) 1995-11-21 1996-11-20 Pyrido[2, 3-d] pyrimidine derivatives and medicinal compositions thereof

Publications (1)

Publication Number Publication Date
BR9611628A true BR9611628A (pt) 1999-06-01

Family

ID=27454776

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9611628A BR9611628A (pt) 1995-11-21 1996-11-20 Derivados de pirido [2,3-d] pirimidina e composições medicinais dos mesmos

Country Status (12)

Country Link
US (1) US6136810A (pt)
EP (1) EP0885894A4 (pt)
JP (1) JP3110765B2 (pt)
KR (1) KR19990071520A (pt)
CN (1) CN1202171A (pt)
AU (1) AU705039B2 (pt)
BR (1) BR9611628A (pt)
CA (1) CA2236683A1 (pt)
HU (1) HUP9900607A3 (pt)
NZ (1) NZ322197A (pt)
TW (1) TW377352B (pt)
WO (1) WO1997019078A1 (pt)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6417190B1 (en) * 1998-12-17 2002-07-09 Boehringer Ingelheim Pharma Kg Tricyclic nitrogen heterocycles as PDE IV inhibitors
CA2715683A1 (en) 1999-08-21 2001-03-01 Nycomed Gmbh Synergistic combination
EP1267903A4 (en) * 2000-02-08 2003-08-06 Pharmacia Corp METHODS OF TREATING GLAUCOMA
US6413968B1 (en) * 2000-06-30 2002-07-02 O'donnell, Jr. Francis E. Treatment of myasthenia gravis by cyclic nucleotide phosphodiesterase inhibition
WO2002032374A2 (en) * 2000-10-18 2002-04-25 Immunex Corporation Methods for treating il-18 mediated disorders
UA80676C2 (en) * 2001-01-29 2007-10-25 Applied Research Systems Use of il-18 inhibitors for the treatment and/or prevention of cardiomyopathy
MXPA03007623A (es) * 2001-02-26 2003-12-04 Tanabe Seiyaku Co Derivado de piridopirimidina o naftiridina.
AU2002324625B2 (en) * 2001-08-07 2008-05-08 Immunex Corporation Interleukin-1 receptors in the treatment of diseases
KR100490970B1 (ko) * 2002-03-22 2005-05-24 씨제이 주식회사 신규 피리도[2,3-ｄ]피리미딘 카르보알데히드 옥심계ＰＤＥ Ⅳ 효소 저해 화합물 및 이의 제조방법
ES2378374T3 (es) * 2003-11-20 2012-04-11 Astellas Pharma Inc. Inhibidores de la PDE 4 para el tratamiento de la cistitis intersticial
TW200738243A (en) * 2005-11-15 2007-10-16 Glaxo Group Ltd Novel process and formulations
US7750019B2 (en) 2006-08-11 2010-07-06 Kowa Company, Ltd. Pyrimidine compound having benzyl(pyridylmethyl)amine structure and medicament comprising the same
NZ578744A (en) 2007-01-31 2012-02-24 Vertex Pharma 2-aminopyridine derivatives useful as kinase inhibitors
US7790737B2 (en) 2007-03-13 2010-09-07 Kowa Company, Ltd. Substituted pyrimidine compounds and their utility as CETP inhibitors
CA2711865A1 (en) 2008-01-11 2009-07-16 Astellas Pharma Inc. A pathological animal model simultaneously developing testicular pain or discomfort behaviors and urinary frequency
US8569337B2 (en) 2008-07-23 2013-10-29 Vertex Pharmaceuticals Incorporated Tri-cyclic pyrazolopyridine kinase inhibitors
WO2010011768A1 (en) 2008-07-23 2010-01-28 Vertex Pharmaceuticals Incorporated Tri-cyclic pyrazolopyridine kinase inhibitors
CA2731451A1 (en) 2008-07-23 2010-01-28 Vertex Pharmaceuticals Incorporated Pyrazolopyridine kinase inhibitors
MX2011001319A (es) 2008-08-06 2011-04-05 Vertex Pharma Inhibidores de aminopiridina cinasa.
CN102459259A (zh) 2009-05-06 2012-05-16 沃泰克斯药物股份有限公司 吡唑并吡啶类
AU2011209649A1 (en) 2010-01-27 2012-08-09 Vertex Pharmaceuticals Incorporated Pyrazolopyrazine kinase inhibitors
WO2011094290A1 (en) 2010-01-27 2011-08-04 Vertex Pharmaceuticals Incorporated Pyrazolopyrimidine kinase inhibitors
US9067932B2 (en) 2010-01-27 2015-06-30 Vertex Pharmaceuticals Incorporated Pyrazolopyridine kinase inhibitors

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA932731A (en) * 1968-12-10 1973-08-28 E. Hardtmann Goetz 1,2-dihydro-pyrido(2,3-d)pyrimidin-2-ones
BE757702A (fr) * 1969-10-20 1971-04-19 Sandoz Sa Derives de la pyrido (2,3-d) pyrimidine, leur preparation et medicaments les contenant.
US3709888A (en) * 1970-06-01 1973-01-09 Sandoz Ag Aryl-substituted-pyrido(2,3-d)pyrimidin-2-ones
US3853898A (en) * 1971-07-20 1974-12-10 Sandoz Ag 3-(2-substituted amino) pyridyl-phenyl ketone imines
US3758475A (en) * 1971-07-20 1973-09-11 Sandoz Ag Pyrido(2,3-d)pyrimidin 2 ones
JPS5394040A (en) * 1976-12-06 1978-08-17 Sandoz Ag Coagolation controlling agent for blood platelet
US4224328A (en) * 1979-04-11 1980-09-23 Sandoz, Inc. Methods with 1-substituted-4-aryl-quinazolin-2(1H)-ones and thiones and pyrido[2,3-d]pyrimidin-2-ones as platelet aggregation inhibitors
WO1988001270A1 (en) * 1986-08-21 1988-02-25 Pfizer Inc. Pyridopyrimidinediones
US5264437A (en) * 1992-03-20 1993-11-23 Syntex (U.S.A.) Inc. Optionally substituted pyrido[2,3-d]pyridine-2,4(1H,3H)-diones and pyrido[2,]pyrimidine-2(1H,3H)-ones
TW299333B (pt) * 1992-12-29 1997-03-01 Takeda Pharm Industry Co Ltd

Also Published As

Publication number Publication date
WO1997019078A1 (en) 1997-05-29
AU705039B2 (en) 1999-05-13
HUP9900607A2 (hu) 1999-06-28
JP3110765B2 (ja) 2000-11-20
EP0885894A1 (en) 1998-12-23
HUP9900607A3 (en) 1999-11-29
TW377352B (en) 1999-12-21
CA2236683A1 (en) 1997-05-29
EP0885894A4 (en) 2000-01-19
CN1202171A (zh) 1998-12-16
AU7588696A (en) 1997-06-11
KR19990071520A (ko) 1999-09-27
US6136810A (en) 2000-10-24
NZ322197A (en) 1999-02-25

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Legal Events

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FA10 Dismissal: dismissal - article 33 of industrial property law