BR7807097A - Processo para preparacao de derivados de imidazolidina,sua aplicacao,derivados de ureia e derivados de imidazolidina - Google Patents
Processo para preparacao de derivados de imidazolidina,sua aplicacao,derivados de ureia e derivados de imidazolidinaInfo
- Publication number
- BR7807097A BR7807097A BR7807097A BR7807097A BR7807097A BR 7807097 A BR7807097 A BR 7807097A BR 7807097 A BR7807097 A BR 7807097A BR 7807097 A BR7807097 A BR 7807097A BR 7807097 A BR7807097 A BR 7807097A
- Authority
- BR
- Brazil
- Prior art keywords
- derivatives
- imidazolidine
- ure
- preparation
- application
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/88—Nitrogen atoms, e.g. allantoin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/72—Two oxygen atoms, e.g. hydantoin
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Endocrinology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Diabetes (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
LU78407 | 1977-10-28 | ||
CH546578A CH642944A5 (en) | 1978-05-19 | 1978-05-19 | Urea derivatives |
CH936778 | 1978-09-06 |
Publications (1)
Publication Number | Publication Date |
---|---|
BR7807097A true BR7807097A (pt) | 1979-05-08 |
Family
ID=27175218
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR7807097A BR7807097A (pt) | 1977-10-28 | 1978-10-27 | Processo para preparacao de derivados de imidazolidina,sua aplicacao,derivados de ureia e derivados de imidazolidina |
Country Status (26)
Country | Link |
---|---|
US (2) | US4407814A (pt) |
EP (1) | EP0001813B1 (pt) |
JP (1) | JPS5470271A (pt) |
AR (2) | AR219560A1 (pt) |
AT (2) | AT366374B (pt) |
AU (1) | AU522536B2 (pt) |
BR (1) | BR7807097A (pt) |
CA (1) | CA1107744A (pt) |
CU (1) | CU34980A (pt) |
DE (2) | DE2861289D1 (pt) |
DK (1) | DK481678A (pt) |
ES (3) | ES474592A1 (pt) |
FI (1) | FI68618C (pt) |
FR (1) | FR2422643A1 (pt) |
GB (1) | GB2008102B (pt) |
GR (1) | GR70681B (pt) |
IE (1) | IE47962B1 (pt) |
IL (1) | IL55773A (pt) |
IT (1) | IT1099450B (pt) |
MC (1) | MC1220A1 (pt) |
NL (1) | NL7810563A (pt) |
NO (1) | NO151461C (pt) |
NZ (1) | NZ188721A (pt) |
PH (1) | PH13569A (pt) |
PT (1) | PT68705A (pt) |
SE (1) | SE7811194L (pt) |
Families Citing this family (30)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FI801184A (fi) * | 1979-04-24 | 1980-10-25 | Hoffmann La Roche | Foerfarande foer framstaellning av imidazolidinderivat |
DE2933917A1 (de) * | 1979-08-22 | 1981-03-26 | Basf Ag, 67063 Ludwigshafen | 5-imino-imidazolidin-2-one und diese enthaltende herbizide. |
DE3134933A1 (de) * | 1981-09-03 | 1983-03-31 | Hoechst Ag, 6230 Frankfurt | "harnstoffderivate, verfahren zu ihrer herstellung und diese enthaltende medikamente sowie deren verwendung" |
EP0091596B1 (de) * | 1982-04-08 | 1991-09-11 | Shell Internationale Researchmaatschappij B.V. | Neue Hydantoine, ihre Herstellung und Verwendung |
US5112983A (en) * | 1987-09-28 | 1992-05-12 | Olin Corporation | Process for producing 1,2,4-triazol-5-one using organic sulfonic acids and polymers thereof as a catalyst |
US5411981A (en) * | 1991-01-09 | 1995-05-02 | Roussel Uclaf | Phenylimidazolidines having antiandrogenic activity |
FR2693461B1 (fr) * | 1992-07-08 | 1994-09-02 | Roussel Uclaf | Nouvelles phénylimidazolidines substituées, leur procédé de préparation, leur application comme médicaments et les compositions pharmaceutiques les renfermant. |
FR2671348B1 (fr) * | 1991-01-09 | 1993-03-26 | Roussel Uclaf | Nouvelles phenylimidazolidines, leur procede de preparation, leur application comme medicaments et les compositions pharmaceutiques les renfermant. |
USRE35956E (en) * | 1991-01-09 | 1998-11-10 | Roussel Uclaf | Phenylimidazolidines having antiandrogenic activity |
FR2694290B1 (fr) * | 1992-07-08 | 1994-09-02 | Roussel Uclaf | Nouvelles phénylimidazolidines éventuellement substituées, leur procédé de préparation, leur application comme médicaments et les compositions pharmaceutiques les renfermant. |
FR2724169B1 (fr) * | 1994-09-06 | 1997-01-03 | Roussel Uclaf | Nouvelles phenylimidazolidines eventuellement substituees, leur procede et des intermediaires de preparation, leur application comme medicaments et les compositions pharmaceutiques les renfermant |
FR2715402B1 (fr) * | 1994-01-05 | 1996-10-04 | Roussel Uclaf | Nouvelles phénylimidazolines éventuellement substituées, leur procédé et des intermédiaires de préparation, leur application comme médicaments et les compositions pharmaceutiques les renfermant. |
TW521073B (en) * | 1994-01-05 | 2003-02-21 | Hoechst Marion Roussel Inc | New optionally substituted phenylimidazolidines, their preparation process, their use as anti-androgenic agent and the pharmaceutical compositions containing them |
FR2741346B1 (fr) * | 1995-11-16 | 1997-12-19 | Roussel Uclaf | Nouveau procede de preparation de derives phenylimidazolidine |
FR2741342B1 (fr) * | 1995-11-22 | 1998-02-06 | Roussel Uclaf | Nouvelles phenylimidazolidines fluorees ou hydroxylees, procede, intermediaires de preparation, application comme medicaments, nouvelle utilisation et compositions pharmaceutiques |
CA2413417A1 (en) * | 2000-06-28 | 2002-01-03 | Bristol-Myers Squibb Company | Selective androgen receptor modulators and methods for their identification, design and use |
EP1854798A3 (en) | 2000-09-19 | 2007-11-28 | Bristol-Myers Squibb Company | Fused heterocyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function |
US6953679B2 (en) | 2000-09-19 | 2005-10-11 | Bristol-Myers Squibb Company | Method for the preparation of fused heterocyclic succinimide compounds and analogs thereof |
US20040087548A1 (en) | 2001-02-27 | 2004-05-06 | Salvati Mark E. | Fused cyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function |
AU2004305075A1 (en) * | 2003-12-19 | 2005-07-07 | The Regents Of The University Of California | Methods and materials for assessing prostate cancer therapies |
NZ550102A (en) * | 2004-02-24 | 2010-10-29 | Univ California | Methods and materials for assessing prostate cancer therapies and compounds (thiohydantoine derivatives) |
US7709517B2 (en) | 2005-05-13 | 2010-05-04 | The Regents Of The University Of California | Diarylhydantoin compounds |
HUE027894T2 (en) | 2006-03-27 | 2016-11-28 | Univ California | An androgen receptor modulator for the treatment of prostate cancer and androgen receptor related diseases |
SG10201408699TA (en) * | 2006-03-29 | 2015-02-27 | Univ California | Diarylthiohydantoin compounds |
EP2620432A3 (en) | 2007-10-26 | 2013-12-18 | The Regents Of the University of California | Diarylhydantoin compounds |
EP3124481B1 (en) | 2010-02-16 | 2018-03-28 | Aragon Pharmaceuticals, Inc. | Androgen receptor modulators and uses thereof |
SG10201912719TA (en) | 2012-09-26 | 2020-02-27 | Aragon Pharmaceuticals Inc | Anti-androgens for the treatment of non-metastatic castrate-resistant prostate cancer |
JOP20200097A1 (ar) | 2013-01-15 | 2017-06-16 | Aragon Pharmaceuticals Inc | معدل مستقبل أندروجين واستخداماته |
TWI726969B (zh) | 2016-01-11 | 2021-05-11 | 比利時商健生藥品公司 | 用作雄性激素受體拮抗劑之經取代之硫尿囊素衍生物 |
AU2018351714A1 (en) | 2017-10-16 | 2020-04-30 | Aragon Pharmaceuticals, Inc. | Anti-androgens for the treatment of non-metastatic castration-resistant prostate cancer |
Family Cites Families (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BE629779A (pt) * | ||||
US3134663A (en) * | 1957-07-23 | 1964-05-26 | Geigy Chem Corp | Herbicidal composition and method employing hydantoins |
FR1405725A (fr) * | 1963-08-23 | 1965-07-09 | Shell Int Research | Procédé de préparation de la 5, 5-diméthyl-4-iminohydantoine |
NO124370B (pt) * | 1968-03-28 | 1972-04-10 | Ciba Geigy Ag | |
US3690863A (en) * | 1968-04-19 | 1972-09-12 | Du Pont | Esters of 3-(carboxyamino)-and 3-(thiocarboxyamino)-2-substituted crotonamides andtheir use as herbicides |
DK123717B (da) * | 1968-11-25 | 1972-07-24 | Sumitomo Chemical Co | 3-(3',5'-Dihalogenphenyl)-imidazolidin-2,4-dionderivater med mirobicid virkning. |
JPS4916937B1 (pt) * | 1970-01-21 | 1974-04-25 | ||
US3676456A (en) * | 1970-02-27 | 1972-07-11 | Ciba Geigy Corp | Derivatives of 3-aryl-5-alkylhydantoins |
JPS5136332B1 (pt) * | 1970-12-09 | 1976-10-07 | ||
US4044021A (en) * | 1971-10-21 | 1977-08-23 | American Cyanamid Company | Tetrasubstituted imidazolidine diuretics useful in the treatment of hyperaldosteronism |
IL45459A (en) * | 1973-09-03 | 1978-01-31 | Ciba Geigy Ag | 1-(dichlorofluoromethylthio)-3-phenyl-imidazolidine-2,4-dione derivatives their preparation and their use as bactericides and fungicides |
FR2329276A1 (fr) * | 1975-10-29 | 1977-05-27 | Roussel Uclaf | Nouvelles imidazolidines substituees, procede de preparation, application comme medicament et compositions les renfermant |
JPS5315373A (en) * | 1976-07-29 | 1978-02-13 | Mitsubishi Chem Ind Ltd | Hydantoin derivatives and fungicides containing same for agriculture and horiticulture |
IL55774A (en) * | 1977-10-28 | 1982-04-30 | Sparamedica Ag | Pharmaceutical compositions containing urea derivatives,certain such novel derivatives and their manufacture |
US4358606A (en) * | 1981-06-19 | 1982-11-09 | Zoecon Corporation | Esters of phenalkyloxycarbonylamino acids |
-
1978
- 1978-10-13 MC MC781334A patent/MC1220A1/xx unknown
- 1978-10-18 FI FI783170A patent/FI68618C/fi not_active IP Right Cessation
- 1978-10-20 IL IL55773A patent/IL55773A/xx unknown
- 1978-10-20 CA CA313,826A patent/CA1107744A/en not_active Expired
- 1978-10-23 AU AU40961/78A patent/AU522536B2/en not_active Expired
- 1978-10-23 NL NL7810563A patent/NL7810563A/xx not_active Application Discontinuation
- 1978-10-24 NZ NZ188721A patent/NZ188721A/xx unknown
- 1978-10-24 IT IT29040/78A patent/IT1099450B/it active
- 1978-10-25 FR FR7830329A patent/FR2422643A1/fr active Granted
- 1978-10-25 GR GR57503A patent/GR70681B/el unknown
- 1978-10-26 PT PT68705A patent/PT68705A/pt unknown
- 1978-10-26 AR AR274243A patent/AR219560A1/es active
- 1978-10-27 SE SE7811194A patent/SE7811194L/xx unknown
- 1978-10-27 AT AT0768978A patent/AT366374B/de active
- 1978-10-27 BR BR7807097A patent/BR7807097A/pt unknown
- 1978-10-27 NO NO783642A patent/NO151461C/no unknown
- 1978-10-27 DK DK481678A patent/DK481678A/da not_active Application Discontinuation
- 1978-10-27 DE DE7878101244T patent/DE2861289D1/de not_active Expired
- 1978-10-27 EP EP78101244A patent/EP0001813B1/de not_active Expired
- 1978-10-27 IE IE2130/78A patent/IE47962B1/en unknown
- 1978-10-27 JP JP13177278A patent/JPS5470271A/ja active Granted
- 1978-10-27 DE DE19782846946 patent/DE2846946A1/de not_active Withdrawn
- 1978-10-27 CU CU7834980A patent/CU34980A/es unknown
- 1978-10-27 ES ES474592A patent/ES474592A1/es not_active Expired
- 1978-10-27 GB GB7842247A patent/GB2008102B/en not_active Expired
- 1978-10-30 PH PH21743A patent/PH13569A/en unknown
-
1979
- 1979-04-30 ES ES480114A patent/ES480114A1/es not_active Expired
- 1979-04-30 ES ES480109A patent/ES480109A1/es not_active Expired
- 1979-10-02 AR AR278316A patent/AR220004A1/es active
-
1981
- 1981-01-19 AT AT0018281A patent/AT366671B/de not_active IP Right Cessation
- 1981-12-14 US US06/330,364 patent/US4407814A/en not_active Expired - Fee Related
-
1983
- 1983-05-12 US US06/493,855 patent/US4482739A/en not_active Expired - Fee Related
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