BR6573584D0 - Processo para a preparacao de derivados de alcanolamina - Google Patents
Processo para a preparacao de derivados de alcanolaminaInfo
- Publication number
- BR6573584D0 BR6573584D0 BR173584/65A BR17358465A BR6573584D0 BR 6573584 D0 BR6573584 D0 BR 6573584D0 BR 173584/65 A BR173584/65 A BR 173584/65A BR 17358465 A BR17358465 A BR 17358465A BR 6573584 D0 BR6573584 D0 BR 6573584D0
- Authority
- BR
- Brazil
- Prior art keywords
- preparation
- alkanolamine derivatives
- alkanolamine
- derivatives
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C233/00—Carboxylic acid amides
- C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C233/16—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
- C07C311/15—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Furan Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB39774/64A GB1078852A (en) | 1964-09-30 | 1964-09-30 | Alkanolamine derivatives |
Publications (1)
Publication Number | Publication Date |
---|---|
BR6573584D0 true BR6573584D0 (pt) | 1973-08-02 |
Family
ID=10411417
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR173584/65A BR6573584D0 (pt) | 1964-09-30 | 1965-09-29 | Processo para a preparacao de derivados de alcanolamina |
Country Status (13)
Country | Link |
---|---|
US (1) | US3408387A (pt) |
JP (2) | JPS5031136B1 (pt) |
AT (2) | AT261586B (pt) |
BE (1) | BE670364A (pt) |
BR (1) | BR6573584D0 (pt) |
CH (1) | CH504407A (pt) |
DE (1) | DE1493887C3 (pt) |
DK (2) | DK113295B (pt) |
ES (2) | ES318019A1 (pt) |
FR (1) | FR5662M (pt) |
GB (1) | GB1078852A (pt) |
NL (1) | NL6512676A (pt) |
SE (1) | SE313061B (pt) |
Families Citing this family (33)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3857952A (en) * | 1967-12-22 | 1974-12-31 | May & Baker Ltd | Certain benzene derivatives useful in treating cardiac disorders |
ZA6808345B (en) * | 1967-12-22 | May & Baker Ltd | Benzene derivatives | |
GB1269775A (en) * | 1968-07-18 | 1972-04-06 | Ici Ltd | Alkanolamine derivatives |
DE1957706C3 (de) * | 1968-11-18 | 1978-06-29 | Pfizer Corp., Colon (Panama) | Kernsubstituierte 3-Phenoxy-l-phenoxyalkylamino-propan-2-ole und Arzneimittel auf deren Basis |
US3934032A (en) * | 1969-02-21 | 1976-01-20 | Imperial Chemical Industries Limited | Alkanolamine derivatives for treating hypertension |
US3873618A (en) * | 1969-07-18 | 1975-03-25 | Ici Ltd | 1-{8 4-(4-Acetamidophenyl)phenoxy{9 -3-isopropyl-2-propanol |
US4120978A (en) * | 1970-01-08 | 1978-10-17 | Ciba-Geigy Corporation | Pharmaceutical composition for inhibiting and blocking cardioselective beta-receptors |
US4038313A (en) * | 1970-01-08 | 1977-07-26 | Ciba-Geigy Corporation | Cycloalkylureido phenoxy propanolamines |
US3864398A (en) * | 1972-05-01 | 1975-02-04 | Teikoku Hormone Mfg Co Ltd | Process for the preparation of acylamino alkanol derivatives |
JPS5323826B2 (pt) * | 1972-05-15 | 1978-07-17 | ||
FR2330383A1 (fr) * | 1975-11-06 | 1977-06-03 | Synthelabo | Nouveaux ethers de phenols substitues, leurs sels, leur preparation et les medicaments qui les renferment |
US4064125A (en) * | 1976-10-29 | 1977-12-20 | E. R. Squibb And Sons, Inc. | Substituted amides having antiinflammatory activity |
US4177280A (en) * | 1978-07-03 | 1979-12-04 | Syntex (U.S.A.) Inc. | Bicyclo[3.1.0]hexyl-substituted carbonylaminophenoxy cardiovascular agents |
DE2948056A1 (de) * | 1979-11-29 | 1981-06-04 | Boehringer Mannheim Gmbh, 6800 Mannheim | Neue aminopropanolderivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel |
US4342783A (en) * | 1980-06-30 | 1982-08-03 | Synthelabo | Anti-glaucoma agent |
DE3640829A1 (de) * | 1986-11-28 | 1988-06-09 | Boehringer Ingelheim Kg | Neue 1-aryloxy-3-amino-2-propanole, ihre herstellung und verwendung |
AU2003250483A1 (en) | 2002-08-19 | 2004-03-11 | Pfizer Products Inc. | Combination therapy for hyperproliferative diseases |
US20060063803A1 (en) * | 2004-09-23 | 2006-03-23 | Pfizer Inc | 4-Amino substituted-2-substituted-1,2,3,4-tetrahydroquinoline compounds |
GT200600381A (es) | 2005-08-25 | 2007-03-28 | Compuestos organicos | |
US7741317B2 (en) | 2005-10-21 | 2010-06-22 | Bristol-Myers Squibb Company | LXR modulators |
US7888376B2 (en) | 2005-11-23 | 2011-02-15 | Bristol-Myers Squibb Company | Heterocyclic CETP inhibitors |
JP5498168B2 (ja) | 2006-12-01 | 2014-05-21 | ブリストル−マイヤーズ スクイブ カンパニー | アテローム性動脈硬化および循環器疾患の治療のためのcetp阻害剤としてのn−((3−ベンジル)−2,2−(ビス−フェニル)−プロパン−1−アミン誘導体 |
US8969514B2 (en) | 2007-06-04 | 2015-03-03 | Synergy Pharmaceuticals, Inc. | Agonists of guanylate cyclase useful for the treatment of hypercholesterolemia, atherosclerosis, coronary heart disease, gallstone, obesity and other cardiovascular diseases |
EA020466B1 (ru) | 2007-06-04 | 2014-11-28 | Синерджи Фармасьютикалз Инк. | Агонисты гуанилатциклазы, пригодные для лечения желудочно-кишечных нарушений, воспаления, рака и других заболеваний |
CA2726917C (en) | 2008-06-04 | 2018-06-26 | Synergy Pharmaceuticals Inc. | Agonists of guanylate cyclase useful for the treatment of gastrointestinal disorders, inflammation, cancer and other disorders |
CA2730603C (en) | 2008-07-16 | 2019-09-24 | Synergy Pharmaceuticals Inc. | Agonists of guanylate cyclase useful for the treatment of gastrointestinal disorders, inflammation, cancer and other disorders |
US9616097B2 (en) | 2010-09-15 | 2017-04-11 | Synergy Pharmaceuticals, Inc. | Formulations of guanylate cyclase C agonists and methods of use |
EP2970384A1 (en) | 2013-03-15 | 2016-01-20 | Synergy Pharmaceuticals Inc. | Agonists of guanylate cyclase and their uses |
CA2905435A1 (en) | 2013-03-15 | 2014-09-25 | Synergy Pharmaceuticals Inc. | Compositions useful for the treatment of gastrointestinal disorders |
JP2016516804A (ja) | 2013-04-17 | 2016-06-09 | ファイザー・インク | 心血管疾患を治療するためのn−ピペリジン−3−イルベンズアミド誘導体 |
CN113388007A (zh) | 2013-06-05 | 2021-09-14 | 博士医疗爱尔兰有限公司 | 鸟苷酸环化酶c的超纯激动剂、制备和使用所述激动剂的方法 |
WO2016055901A1 (en) | 2014-10-08 | 2016-04-14 | Pfizer Inc. | Substituted amide compounds |
JOP20210193A1 (ar) | 2019-01-18 | 2023-01-30 | Astrazeneca Ab | مثبطات pcsk9 وطرق استخدامها |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB922600A (en) * | 1960-05-06 | 1963-04-03 | Crookes Lab Ltd | Ortho-tertiary-butyl phenolethers |
-
1964
- 1964-09-30 GB GB39774/64A patent/GB1078852A/en not_active Expired
-
1965
- 1965-09-17 US US488252A patent/US3408387A/en not_active Expired - Lifetime
- 1965-09-24 AT AT239367A patent/AT261586B/de active
- 1965-09-24 AT AT873365A patent/AT261582B/de active
- 1965-09-27 CH CH967068A patent/CH504407A/de not_active IP Right Cessation
- 1965-09-29 SE SE12618/65A patent/SE313061B/xx unknown
- 1965-09-29 BR BR173584/65A patent/BR6573584D0/pt unknown
- 1965-09-30 NL NL6512676A patent/NL6512676A/xx unknown
- 1965-09-30 ES ES0318019A patent/ES318019A1/es not_active Expired
- 1965-09-30 DE DE1493887A patent/DE1493887C3/de not_active Expired
- 1965-09-30 BE BE670364A patent/BE670364A/xx unknown
- 1965-09-30 JP JP40059684A patent/JPS5031136B1/ja active Pending
- 1965-09-30 DK DK504665AA patent/DK113295B/da unknown
- 1965-12-29 FR FR44136A patent/FR5662M/fr not_active Expired
-
1966
- 1966-12-23 DK DK668366AA patent/DK122879B/da unknown
-
1967
- 1967-09-14 JP JP6759060A patent/JPS514978B1/ja active Pending
-
1968
- 1968-09-16 ES ES358534A patent/ES358534A2/es not_active Expired
Also Published As
Publication number | Publication date |
---|---|
JPS5031136B1 (pt) | 1975-10-07 |
ES318019A1 (es) | 1966-07-01 |
DK113295B (da) | 1969-03-10 |
DE1493887B2 (de) | 1977-08-25 |
CH504407A (de) | 1971-03-15 |
US3408387A (en) | 1968-10-29 |
AT261582B (de) | 1968-05-10 |
BE670364A (pt) | 1966-03-30 |
FR5662M (pt) | 1968-01-02 |
DE1493887A1 (de) | 1972-06-15 |
ES358534A2 (es) | 1970-07-01 |
JPS514978B1 (pt) | 1976-02-16 |
NL6512676A (pt) | 1966-03-31 |
AT261586B (de) | 1968-05-10 |
DK122879B (da) | 1972-04-24 |
DE1493887C3 (de) | 1978-06-15 |
SE313061B (pt) | 1969-08-04 |
GB1078852A (en) | 1967-08-09 |
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