BR112022024988A2 - Compostos e métodos para tratamento de infecções fúngicas - Google Patents

Compostos e métodos para tratamento de infecções fúngicas

Info

Publication number
BR112022024988A2
BR112022024988A2 BR112022024988A BR112022024988A BR112022024988A2 BR 112022024988 A2 BR112022024988 A2 BR 112022024988A2 BR 112022024988 A BR112022024988 A BR 112022024988A BR 112022024988 A BR112022024988 A BR 112022024988A BR 112022024988 A2 BR112022024988 A2 BR 112022024988A2
Authority
BR
Brazil
Prior art keywords
treatment
methods
compounds
fungal infections
fungal
Prior art date
Application number
BR112022024988A
Other languages
English (en)
Inventor
joy Shaw Karen
Schlamm Haran
R Hodges Michael
Original Assignee
Amplyx Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Amplyx Pharmaceuticals Inc filed Critical Amplyx Pharmaceuticals Inc
Publication of BR112022024988A2 publication Critical patent/BR112022024988A2/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/66Phosphorus compounds
    • A61K31/675Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Dermatology (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

COMPOSTOS E MÉTODOS PARA TRATAMENTO DE INFECÇÕES FÚNGICAS. A presente invenção refere-se a composições e métodos de uso das mesmas para o tratamento de infecções e doenças fúngicas.
BR112022024988A 2020-06-17 2021-06-16 Compostos e métodos para tratamento de infecções fúngicas BR112022024988A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US202063040450P 2020-06-17 2020-06-17
PCT/US2021/037578 WO2021257670A1 (en) 2020-06-17 2021-06-16 Compounds and methods for treating fungal infections

Publications (1)

Publication Number Publication Date
BR112022024988A2 true BR112022024988A2 (pt) 2022-12-27

Family

ID=79268375

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112022024988A BR112022024988A2 (pt) 2020-06-17 2021-06-16 Compostos e métodos para tratamento de infecções fúngicas

Country Status (12)

Country Link
US (1) US20230233586A1 (pt)
EP (1) EP4167998A4 (pt)
JP (1) JP2023530936A (pt)
KR (1) KR20230024375A (pt)
CN (1) CN115884775A (pt)
AU (1) AU2021293911B2 (pt)
BR (1) BR112022024988A2 (pt)
CA (1) CA3187268A1 (pt)
IL (1) IL299057A (pt)
MX (1) MX2022016179A (pt)
TW (1) TWI888580B (pt)
WO (1) WO2021257670A1 (pt)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20220148881A (ko) 2020-03-04 2022-11-07 앰플릭스 파마슈티컬스, 인크. 진균 감염 치료에서의 화합물의 용도

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI385169B (zh) * 2005-10-31 2013-02-11 Eisai R&D Man Co Ltd 經雜環取代之吡啶衍生物及含有彼之抗真菌劑
US8513287B2 (en) * 2007-12-27 2013-08-20 Eisai R&D Management Co., Ltd. Heterocyclic ring and phosphonoxymethyl group substituted pyridine derivatives and antifungal agent containing same
US20130288956A1 (en) * 2010-11-05 2013-10-31 Eisai R&D Management Co., Ltd. Combined pharmaceutical composition as antifungal agent
CN112996527B (zh) * 2018-08-31 2025-02-21 巴斯利尔药物阿尔施维尔国际股份公司 用于治疗真菌感染的化合物和方法
US11819503B2 (en) * 2019-04-23 2023-11-21 F2G Ltd Method of treating coccidioides infection
KR20220148881A (ko) * 2020-03-04 2022-11-07 앰플릭스 파마슈티컬스, 인크. 진균 감염 치료에서의 화합물의 용도

Also Published As

Publication number Publication date
MX2022016179A (es) 2023-04-20
CN115884775A (zh) 2023-03-31
US20230233586A1 (en) 2023-07-27
KR20230024375A (ko) 2023-02-20
IL299057A (en) 2023-02-01
JP2023530936A (ja) 2023-07-20
EP4167998A1 (en) 2023-04-26
CA3187268A1 (en) 2021-12-23
TW202214258A (zh) 2022-04-16
WO2021257670A1 (en) 2021-12-23
AU2021293911B2 (en) 2024-11-14
AU2021293911A1 (en) 2023-01-19
TWI888580B (zh) 2025-07-01
EP4167998A4 (en) 2024-07-17

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Legal Events

Date Code Title Description
B25G Requested change of headquarter approved

Owner name: AMPLYX PHARMACEUTICALS, INC. (US)

B25A Requested transfer of rights approved

Owner name: BASILEA PHARMACEUTICA INTERNATIONAL AG, ALLSCHWIL (CH)