BR112021012266A2 - Docetaxel para uso em uma terapia de combinação no tratamento de câncer, inibidor de cy3a para uso em uma terapia de combinação no tratamento de câncer, docetaxel ou um inibidor de cy3a para uso em uma terapia de combinação, método para o tratamento de um câncer de próstata resistente à castração metastático e kit - Google Patents
Docetaxel para uso em uma terapia de combinação no tratamento de câncer, inibidor de cy3a para uso em uma terapia de combinação no tratamento de câncer, docetaxel ou um inibidor de cy3a para uso em uma terapia de combinação, método para o tratamento de um câncer de próstata resistente à castração metastático e kit Download PDFInfo
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- BR112021012266A2 BR112021012266A2 BR112021012266-4A BR112021012266A BR112021012266A2 BR 112021012266 A2 BR112021012266 A2 BR 112021012266A2 BR 112021012266 A BR112021012266 A BR 112021012266A BR 112021012266 A2 BR112021012266 A2 BR 112021012266A2
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- docetaxel
- cy3a
- inhibitor
- cancer
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- DDBREPKUVSBGFI-UHFFFAOYSA-N phenobarbital Chemical compound C=1C=CC=CC=1C1(CC)C(=O)NC(=O)NC1=O DDBREPKUVSBGFI-UHFFFAOYSA-N 0.000 description 1
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/337—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP18215488 | 2018-12-21 | ||
| EP18215488.0 | 2018-12-21 | ||
| PCT/EP2019/086125 WO2020127607A1 (en) | 2018-12-21 | 2019-12-18 | Combination treatment for solid tumors using docetaxel and a cyp3a inhibitor |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR112021012266A2 true BR112021012266A2 (pt) | 2021-08-31 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR112021012266-4A BR112021012266A2 (pt) | 2018-12-21 | 2019-12-18 | Docetaxel para uso em uma terapia de combinação no tratamento de câncer, inibidor de cy3a para uso em uma terapia de combinação no tratamento de câncer, docetaxel ou um inibidor de cy3a para uso em uma terapia de combinação, método para o tratamento de um câncer de próstata resistente à castração metastático e kit |
Country Status (13)
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| US (1) | US20220071944A1 (https=) |
| EP (1) | EP3897611A1 (https=) |
| JP (3) | JP2022514960A (https=) |
| KR (1) | KR20220004011A (https=) |
| CN (1) | CN113473982A (https=) |
| AU (2) | AU2019410062A1 (https=) |
| BR (1) | BR112021012266A2 (https=) |
| CA (1) | CA3124319C (https=) |
| CL (1) | CL2021001635A1 (https=) |
| IL (1) | IL284225A (https=) |
| MX (1) | MX2021007480A (https=) |
| PE (1) | PE20220129A1 (https=) |
| WO (1) | WO2020127607A1 (https=) |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PE20220250A1 (es) * | 2018-12-21 | 2022-02-16 | Modra Pharmaceuticals B V | Uso de docetaxel en el tratamiento de cancer mediante control de niveles maximos en plasma |
| GB202201935D0 (en) | 2022-02-14 | 2022-03-30 | Modra Pharmaceuticals B V | Methods and compositions for treating cancer in taxane-resistant patients |
| CN116270617B (zh) * | 2023-03-29 | 2024-01-26 | 济宁医学院附属医院 | Arp2/3复合物抑制剂CK-666和多西他赛组合用于癌症治疗的制药用途 |
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| GB0716591D0 (en) * | 2007-08-24 | 2007-10-03 | Vereniging Het Nl Kanker I | Composition |
| MX2010002179A (es) | 2007-08-24 | 2010-04-27 | Stichting Het Nl Kanker I | Composicion para el tratamiento de enfermedades neoplasicas. |
| US9089544B2 (en) * | 2007-08-24 | 2015-07-28 | Slotervaart Participaties Bv | Composition |
| WO2010020799A2 (en) | 2008-08-22 | 2010-02-25 | Slotervaart Participaties Bv | Composition |
| PE20220250A1 (es) * | 2018-12-21 | 2022-02-16 | Modra Pharmaceuticals B V | Uso de docetaxel en el tratamiento de cancer mediante control de niveles maximos en plasma |
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2019
- 2019-12-18 KR KR1020217022969A patent/KR20220004011A/ko not_active Ceased
- 2019-12-18 BR BR112021012266-4A patent/BR112021012266A2/pt not_active Application Discontinuation
- 2019-12-18 CN CN201980090621.4A patent/CN113473982A/zh active Pending
- 2019-12-18 CA CA3124319A patent/CA3124319C/en active Active
- 2019-12-18 MX MX2021007480A patent/MX2021007480A/es unknown
- 2019-12-18 PE PE2021001053A patent/PE20220129A1/es unknown
- 2019-12-18 US US17/416,946 patent/US20220071944A1/en active Pending
- 2019-12-18 EP EP19828725.2A patent/EP3897611A1/en active Pending
- 2019-12-18 WO PCT/EP2019/086125 patent/WO2020127607A1/en not_active Ceased
- 2019-12-18 AU AU2019410062A patent/AU2019410062A1/en not_active Abandoned
- 2019-12-18 JP JP2021536396A patent/JP2022514960A/ja active Pending
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2025
- 2025-03-24 JP JP2025049063A patent/JP2025094186A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| KR20220004011A (ko) | 2022-01-11 |
| PE20220129A1 (es) | 2022-01-27 |
| MX2021007480A (es) | 2021-10-13 |
| EP3897611A1 (en) | 2021-10-27 |
| JP2025094186A (ja) | 2025-06-24 |
| CL2021001635A1 (es) | 2022-04-22 |
| US20220071944A1 (en) | 2022-03-10 |
| IL284225A (en) | 2021-08-31 |
| WO2020127607A1 (en) | 2020-06-25 |
| CA3124319C (en) | 2023-07-04 |
| CA3124319A1 (en) | 2020-06-25 |
| AU2019410062A1 (en) | 2021-08-12 |
| CN113473982A (zh) | 2021-10-01 |
| JP2022514960A (ja) | 2022-02-16 |
| JP2023102786A (ja) | 2023-07-25 |
| AU2023204693A1 (en) | 2023-08-10 |
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| B06W | Patent application suspended after preliminary examination (for patents with searches from other patent authorities) chapter 6.23 patent gazette] | ||
| B11B | Dismissal acc. art. 36, par 1 of ipl - no reply within 90 days to fullfil the necessary requirements |