BR112017012005B1 - Compostos orgânicos inibidores de pde2, composições farmacêuticas compreendendo os ditos compostos e uso dos mesmos no tratamento de um distúrbio mediado por pde2 - Google Patents
Compostos orgânicos inibidores de pde2, composições farmacêuticas compreendendo os ditos compostos e uso dos mesmos no tratamento de um distúrbio mediado por pde2 Download PDFInfo
- Publication number
- BR112017012005B1 BR112017012005B1 BR112017012005-4A BR112017012005A BR112017012005B1 BR 112017012005 B1 BR112017012005 B1 BR 112017012005B1 BR 112017012005 A BR112017012005 A BR 112017012005A BR 112017012005 B1 BR112017012005 B1 BR 112017012005B1
- Authority
- BR
- Brazil
- Prior art keywords
- pyrazolo
- methyl
- disorder
- butoxy
- naphthyridin
- Prior art date
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201462088540P | 2014-12-06 | 2014-12-06 | |
| US62/088,540 | 2014-12-06 | ||
| PCT/US2015/064331 WO2016090382A1 (en) | 2014-12-06 | 2015-12-07 | Organic compounds |
Publications (2)
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| US9628116B2 (en) | 2015-07-14 | 2017-04-18 | At&T Intellectual Property I, L.P. | Apparatus and methods for transmitting wireless signals |
| TWI795381B (zh) | 2016-12-21 | 2023-03-11 | 比利時商健生藥品公司 | 作為ｍａｌｔ１抑制劑之吡唑衍生物 |
| TWI782056B (zh) * | 2017-07-14 | 2022-11-01 | 日商鹽野義製藥股份有限公司 | 具有ｍｇａｔ２抑制活性的縮合環衍生物 |
| SG11202009735QA (en) | 2018-04-13 | 2020-10-29 | Cancer Research Tech Ltd | Bcl6 inhibitors |
| CN112585128B (zh) | 2018-06-18 | 2023-02-21 | 詹森药业有限公司 | 作为malt1抑制剂的吡唑衍生物 |
| KR20210114001A (ko) | 2019-01-11 | 2021-09-17 | 시오노기 앤드 컴파니, 리미티드 | Mgat2 저해 활성을 갖는 다이하이드로피라졸로피라지논 유도체 |
| EP3953345B1 (en) | 2019-04-11 | 2023-04-05 | Janssen Pharmaceutica NV | Pyridine rings containing derivatives as malt1 inhibitors |
| GB201914860D0 (en) | 2019-10-14 | 2019-11-27 | Cancer Research Tech Ltd | Inhibitor compounds |
| CN112851667B (zh) * | 2019-11-28 | 2022-09-09 | 暨南大学 | 含氮并杂环类化合物及其药用组合物和应用 |
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| CN107205993B (zh) | 2021-03-09 |
| EP3226862B1 (en) | 2020-07-08 |
| CN107205993A (zh) | 2017-09-26 |
| HK1243935A1 (zh) | 2018-07-27 |
| KR20170089001A (ko) | 2017-08-02 |
| US10105349B2 (en) | 2018-10-23 |
| MX373320B (es) | 2020-05-04 |
| MX2017007377A (es) | 2017-11-06 |
| US20190000807A1 (en) | 2019-01-03 |
| KR102562576B1 (ko) | 2023-08-01 |
| US20170360753A1 (en) | 2017-12-21 |
| WO2016090382A1 (en) | 2016-06-09 |
| JP6608933B2 (ja) | 2019-11-20 |
| AU2015357498B2 (en) | 2019-09-12 |
| IL252578B (en) | 2021-05-31 |
| US10543194B2 (en) | 2020-01-28 |
| CA2969597C (en) | 2023-10-24 |
| JP2017536409A (ja) | 2017-12-07 |
| IL252578A0 (en) | 2017-07-31 |
| RU2702732C1 (ru) | 2019-10-10 |
| EP3226862A1 (en) | 2017-10-11 |
| HK1244427A1 (zh) | 2018-08-10 |
| BR112017012005A2 (pt) | 2017-12-26 |
| EP3226862A4 (en) | 2018-05-09 |
| AU2015357498A1 (en) | 2017-07-27 |
| CA2969597A1 (en) | 2016-06-09 |
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