BR112016022743A2 - Método para tratar e/ou evitar pelo menos uma cicatriz de acne, uso de uma combinação fixa de adapaleno e peróxido de benzoíla e composição - Google Patents
Método para tratar e/ou evitar pelo menos uma cicatriz de acne, uso de uma combinação fixa de adapaleno e peróxido de benzoíla e composiçãoInfo
- Publication number
- BR112016022743A2 BR112016022743A2 BR112016022743A BR112016022743A BR112016022743A2 BR 112016022743 A2 BR112016022743 A2 BR 112016022743A2 BR 112016022743 A BR112016022743 A BR 112016022743A BR 112016022743 A BR112016022743 A BR 112016022743A BR 112016022743 A2 BR112016022743 A2 BR 112016022743A2
- Authority
- BR
- Brazil
- Prior art keywords
- adapalene
- benzoyl peroxide
- fixed combination
- composition
- treat
- Prior art date
Links
- 239000004342 Benzoyl peroxide Substances 0.000 title abstract 4
- OMPJBNCRMGITSC-UHFFFAOYSA-N Benzoylperoxide Chemical compound C=1C=CC=CC=1C(=O)OOC(=O)C1=CC=CC=C1 OMPJBNCRMGITSC-UHFFFAOYSA-N 0.000 title abstract 4
- LZCDAPDGXCYOEH-UHFFFAOYSA-N adapalene Chemical compound C1=C(C(O)=O)C=CC2=CC(C3=CC=C(C(=C3)C34CC5CC(CC(C5)C3)C4)OC)=CC=C21 LZCDAPDGXCYOEH-UHFFFAOYSA-N 0.000 title abstract 4
- 229960002916 adapalene Drugs 0.000 title abstract 4
- 235000019400 benzoyl peroxide Nutrition 0.000 title abstract 4
- 208000002874 Acne Vulgaris Diseases 0.000 title abstract 3
- 206010000496 acne Diseases 0.000 title abstract 3
- 231100000241 scar Toxicity 0.000 title abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- 206010039580 Scar Diseases 0.000 abstract 1
- 230000037390 scarring Effects 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/192—Carboxylic acids, e.g. valproic acid having aromatic groups, e.g. sulindac, 2-aryl-propionic acids, ethacrynic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/327—Peroxy compounds, e.g. hydroperoxides, peroxides, peroxyacids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/14—Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/16—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
- A61K47/18—Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
- A61K47/183—Amino acids, e.g. glycine, EDTA or aspartame
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0014—Skin, i.e. galenical aspects of topical compositions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/06—Ointments; Bases therefor; Other semi-solid forms, e.g. creams, sticks, gels
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Dermatology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
- Cosmetics (AREA)
Abstract
MÉTODO PARA TRATAR E/OU EVITAR PELO MENOS UMA CICATRIZ DE ACNE, USO DE UMA COMBINAÇÃO FIXA DE ADAPALENO E PERÓXIDO DE BENZOÍLA E COMPOSIÇÃO. A presente invenção diz respeito a um método para tratar e/ou prevenir as cicatrizes da acne no qual uma quantidade eficaz de uma composição que contém uma combinação fixa de adapaleno ou um de seus sais e peróxido de benzoíla é administrada em um paciente que necessita dela. A presente invenção diz respeito ainda a composição que contém uma combinação fixa de adapaleno ou um de seus sais e peróxido de benzoíla para seu uso para tratar e/ou evitar as cicatrizes da acne.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201461973350P | 2014-04-01 | 2014-04-01 | |
PCT/EP2015/056906 WO2015150332A1 (en) | 2014-04-01 | 2015-03-30 | Combination of adapalene and benzoyl peroxide for treating acne scars |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112016022743A2 true BR112016022743A2 (pt) | 2017-08-15 |
Family
ID=52780548
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112016022743A BR112016022743A2 (pt) | 2014-04-01 | 2015-03-30 | Método para tratar e/ou evitar pelo menos uma cicatriz de acne, uso de uma combinação fixa de adapaleno e peróxido de benzoíla e composição |
Country Status (11)
Country | Link |
---|---|
US (1) | US20170020833A1 (pt) |
EP (1) | EP3125880B1 (pt) |
KR (2) | KR20160130862A (pt) |
AU (1) | AU2015239688B2 (pt) |
BR (1) | BR112016022743A2 (pt) |
CA (1) | CA2944073A1 (pt) |
CL (1) | CL2016002489A1 (pt) |
MX (1) | MX2016012623A (pt) |
RU (1) | RU2016142678A (pt) |
SG (2) | SG10202100745QA (pt) |
WO (1) | WO2015150332A1 (pt) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BR112022003367A2 (pt) * | 2019-08-23 | 2022-05-17 | Allergan Pharmaceuticals Int Ltd | Tropoelastina para uso em tratamento de cicatrizes de acne |
WO2023068233A1 (ja) * | 2021-10-18 | 2023-04-27 | マルホ株式会社 | 活性阻害及び/又は産生抑制剤 |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2833841B1 (fr) | 2001-12-21 | 2005-07-22 | Galderma Res & Dev | Gel comprenant au moins un retinoide et du peroxyde de benzoyle |
FR2901139B1 (fr) * | 2006-05-17 | 2009-03-20 | Galderma Res & Dev S N C Snc | Compositions comprenant au moins un derive de l'acide naphtoique et du peroxyde de benzoyle, leurs procedes de preparation, et leurs utilisations |
US8080537B2 (en) * | 2006-07-13 | 2011-12-20 | Galderma Research & Development | Combinations of adapalene and benzoyl peroxide for treating acne lesions |
FR2903603B1 (fr) * | 2006-07-13 | 2009-03-20 | Galderma Res & Dev S N C Snc | Combinaison d'adapalene et de peroxyde de benzole dans le traitement de l'acne |
EP2114392B1 (en) * | 2007-01-30 | 2015-06-10 | Galderma Research & Development | Use of adapalene and benzoyl peroxide for the long term treatment of acne vulgaris |
MX2012008871A (es) * | 2010-02-09 | 2012-08-31 | Galderma Res & Dev | Composicion dermatologica que comprende combinacion de adapaleno y peroxido de benzoilo para el tratamiento del acne en poblacion no caucasica con reduccion de hiperpigmentacion post-inflamatoria. |
CA2796412A1 (en) * | 2010-04-29 | 2011-11-03 | Galderma Research & Development | Method for treating scars with adapalene 0.3% |
EP3082785A1 (en) * | 2013-12-19 | 2016-10-26 | Galderma Research & Development | Therapy regimen for treating severe acne related diseases |
-
2015
- 2015-03-30 AU AU2015239688A patent/AU2015239688B2/en active Active
- 2015-03-30 RU RU2016142678A patent/RU2016142678A/ru unknown
- 2015-03-30 SG SG10202100745QA patent/SG10202100745QA/en unknown
- 2015-03-30 WO PCT/EP2015/056906 patent/WO2015150332A1/en active Application Filing
- 2015-03-30 EP EP15713330.7A patent/EP3125880B1/en active Active
- 2015-03-30 KR KR1020167030495A patent/KR20160130862A/ko active Application Filing
- 2015-03-30 US US15/301,197 patent/US20170020833A1/en not_active Abandoned
- 2015-03-30 KR KR1020227037052A patent/KR20220148939A/ko not_active Application Discontinuation
- 2015-03-30 SG SG11201608222WA patent/SG11201608222WA/en unknown
- 2015-03-30 MX MX2016012623A patent/MX2016012623A/es active IP Right Grant
- 2015-03-30 CA CA2944073A patent/CA2944073A1/en not_active Abandoned
- 2015-03-30 BR BR112016022743A patent/BR112016022743A2/pt not_active Application Discontinuation
-
2016
- 2016-09-30 CL CL2016002489A patent/CL2016002489A1/es unknown
Also Published As
Publication number | Publication date |
---|---|
CL2016002489A1 (es) | 2017-02-03 |
EP3125880A1 (en) | 2017-02-08 |
WO2015150332A1 (en) | 2015-10-08 |
MX2016012623A (es) | 2016-12-14 |
KR20160130862A (ko) | 2016-11-14 |
CA2944073A1 (en) | 2015-10-08 |
RU2016142678A (ru) | 2018-05-07 |
AU2015239688A1 (en) | 2016-10-13 |
US20170020833A1 (en) | 2017-01-26 |
SG11201608222WA (en) | 2016-10-28 |
EP3125880B1 (en) | 2019-11-20 |
KR20220148939A (ko) | 2022-11-07 |
AU2015239688B2 (en) | 2020-06-25 |
SG10202100745QA (en) | 2021-02-25 |
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Legal Events
Date | Code | Title | Description |
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B11A | Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing | ||
B11Y | Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette] | ||
B350 | Update of information on the portal [chapter 15.35 patent gazette] |