BR112016018594B8 - Método para produção do derivado de 2-aciliminopiridina - Google Patents

Método para produção do derivado de 2-aciliminopiridina

Info

Publication number
BR112016018594B8
BR112016018594B8 BR112016018594A BR112016018594A BR112016018594B8 BR 112016018594 B8 BR112016018594 B8 BR 112016018594B8 BR 112016018594 A BR112016018594 A BR 112016018594A BR 112016018594 A BR112016018594 A BR 112016018594A BR 112016018594 B8 BR112016018594 B8 BR 112016018594B8
Authority
BR
Brazil
Prior art keywords
formula
compound represented
production
acyliminopyridine
derivative
Prior art date
Application number
BR112016018594A
Other languages
English (en)
Other versions
BR112016018594B1 (pt
Inventor
Nakanishi Nozomu
Kitsuda Shigeki
Fukuda Yoshimasa
Original Assignee
Meiji Seika Pharma Co Ltd
Mmag Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Meiji Seika Pharma Co Ltd, Mmag Co Ltd filed Critical Meiji Seika Pharma Co Ltd
Publication of BR112016018594B1 publication Critical patent/BR112016018594B1/pt
Publication of BR112016018594B8 publication Critical patent/BR112016018594B8/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

MÉTODO PARA PRODUÇÃO DO DERIVADO DE 2-ACILIMINOPIRIDINA. A presente invenção refere-se a um método para produção de um composto representado pela fórmula (I) que compreende: uma etapa de acilação de um grupo amino localizado na posição 2 em um composto representado pela fórmula (A) utilizando o ácido trifluoroacético como um agente de acilação, produzindo assim um composto representado pela fórmula (B); e uma etapa de alquilação adicional de um átomo de nitrogênio localizado na posição 1 do composto representado pela fórmula (B).
BR112016018594A 2014-03-10 2015-03-04 Método para produção do derivado de 2-aciliminopiridina BR112016018594B8 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2014-046202 2014-03-10
JP2014046202 2014-03-10
PCT/JP2015/056409 WO2015137216A1 (ja) 2014-03-10 2015-03-04 ２－アシルイミノピリジン誘導体の製造法

Publications (2)

Publication Number Publication Date
BR112016018594B1 BR112016018594B1 (pt) 2021-02-17
BR112016018594B8 true BR112016018594B8 (pt) 2022-11-22

Family

ID=54071662

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112016018594A BR112016018594B8 (pt) 2014-03-10 2015-03-04 Método para produção do derivado de 2-aciliminopiridina

Country Status (10)

Country Link
US (1) US9975851B2 (pt)
EP (1) EP3118194B1 (pt)
JP (1) JP6398124B2 (pt)
CN (1) CN105980360B (pt)
BR (1) BR112016018594B8 (pt)
CA (1) CA2941215A1 (pt)
MX (1) MX2016010868A (pt)
PH (1) PH12016501704A1 (pt)
TW (1) TWI650314B (pt)
WO (1) WO2015137216A1 (pt)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2749555B1 (en) * 2011-08-26 2018-11-14 Meiji Seika Pharma Co., Ltd. Method for producing pest controlling agent
TW201711566A (zh) * 2015-09-28 2017-04-01 拜耳作物科學公司 製備ｎ－（１，３，４－㗁二唑－２－基）芳基甲醯胺之方法
HUE060155T2 (hu) 2016-09-16 2023-02-28 Mmag Co Ltd Növényvédõszer optimalizált elõállítási módszere
CN111320573B (zh) * 2018-12-13 2022-11-01 江苏中旗科技股份有限公司 一种吡啶胺类化合物的制备方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3639877A1 (de) 1986-11-21 1988-05-26 Bayer Ag Hetarylalkyl substituierte 5- und 6-ringheterocyclen
DE4021439A1 (de) * 1989-12-14 1991-06-20 Bayer Ag 2-iminopyridin-derivate
EP0639569A4 (en) 1991-03-11 1995-09-20 Nippon Soda Co NEW HETEROCYCLIC COMPOUND.
JPH0578323A (ja) 1991-03-11 1993-03-30 Nippon Soda Co Ltd 新規なヘテロ環化合物、その製造方法及び殺虫剤
JP2009292799A (ja) 2008-06-02 2009-12-17 Yasuo Kikukawa トリフルオロ酢酸をアシル化剤とするトリフルオロアセタミド類の製造方法
EP2959775A1 (en) * 2010-08-31 2015-12-30 Meiji Seika Pharma Co., Ltd. Pest control agent
EP2749555B1 (en) 2011-08-26 2018-11-14 Meiji Seika Pharma Co., Ltd. Method for producing pest controlling agent

Also Published As

Publication number Publication date
EP3118194A4 (en) 2017-08-02
TWI650314B (zh) 2019-02-11
CN105980360B (zh) 2019-03-15
BR112016018594B1 (pt) 2021-02-17
CN105980360A (zh) 2016-09-28
JP6398124B2 (ja) 2018-10-03
PH12016501704B1 (en) 2017-02-06
CA2941215A1 (en) 2015-09-17
EP3118194B1 (en) 2020-07-29
US9975851B2 (en) 2018-05-22
US20170073312A1 (en) 2017-03-16
MX2016010868A (es) 2016-11-17
WO2015137216A1 (ja) 2015-09-17
TW201623240A (zh) 2016-07-01
JPWO2015137216A1 (ja) 2017-04-06
PH12016501704A1 (en) 2017-02-06
EP3118194A1 (en) 2017-01-18

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Legal Events

Date Code Title Description
B06U Preliminary requirement: requests with searches performed by other patent offices: procedure suspended [chapter 6.21 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 04/03/2015, OBSERVADAS AS CONDICOES LEGAIS.

B25A Requested transfer of rights approved

Owner name: MMAG CO., LTD. (JP)

B25G Requested change of headquarter approved

Owner name: MMAG CO., LTD. (JP)