BR112015028751A2 - processo para a preparação de derivados de 3,5-bis (fluoralquil)pirazol a partir de alfa,alfa-dihaloaminas - Google Patents

processo para a preparação de derivados de 3,5-bis (fluoralquil)pirazol a partir de alfa,alfa-dihaloaminas

Info

Publication number
BR112015028751A2
BR112015028751A2 BR112015028751A BR112015028751A BR112015028751A2 BR 112015028751 A2 BR112015028751 A2 BR 112015028751A2 BR 112015028751 A BR112015028751 A BR 112015028751A BR 112015028751 A BR112015028751 A BR 112015028751A BR 112015028751 A2 BR112015028751 A2 BR 112015028751A2
Authority
BR
Brazil
Prior art keywords
alpha
dihaloamines
fluoralkyl
bis
preparation
Prior art date
Application number
BR112015028751A
Other languages
English (en)
Other versions
BR112015028751B1 (pt
Inventor
Neeff Arnd
Leroux Frédéric
Landelle Grégory
Vors Jean-Pierre
James Ford Mark
Lui Norbert
Pazenok Sergii
Etzel Winfried
Original Assignee
Bayer Cropscience Ag
Centre Nat Rech Scient
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag, Centre Nat Rech Scient filed Critical Bayer Cropscience Ag
Publication of BR112015028751A2 publication Critical patent/BR112015028751A2/pt
Publication of BR112015028751B1 publication Critical patent/BR112015028751B1/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

Abstract

resumo processo para a preparação de derivados de 3,5-bis (fluoralquil)pirazol a partir de alfa,alfa-dihaloaminas a presente invenção refere-se a um novo processo para a preparação de derivados de 3,5-bis (fluoralquil)pirazol a partir de a,a-dihaloaminas.
BR112015028751-4A 2013-05-22 2014-05-19 Processo para a preparação de derivados de 3,5-bis (fluoralquil)pirazol a partir de alfa, alfa-dihaloaminas e uso destes para preparação de ingredientes fungicidas ativos BR112015028751B1 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP13356007.8 2013-05-22
EP13356007 2013-05-22
PCT/EP2014/060238 WO2014187773A1 (en) 2013-05-22 2014-05-19 PROCESS FOR PREPARING 3,5-BIS(FLUOROALKYL)PYRAZOLE DERIVATIVES FROM α,α-DIHALOAMINES

Publications (2)

Publication Number Publication Date
BR112015028751A2 true BR112015028751A2 (pt) 2017-07-25
BR112015028751B1 BR112015028751B1 (pt) 2021-01-12

Family

ID=48628588

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112015028751-4A BR112015028751B1 (pt) 2013-05-22 2014-05-19 Processo para a preparação de derivados de 3,5-bis (fluoralquil)pirazol a partir de alfa, alfa-dihaloaminas e uso destes para preparação de ingredientes fungicidas ativos

Country Status (12)

Country Link
US (1) US9512081B2 (pt)
EP (1) EP2999694B1 (pt)
JP (1) JP6377727B2 (pt)
KR (1) KR102233655B1 (pt)
CN (1) CN105408314B (pt)
BR (1) BR112015028751B1 (pt)
DK (1) DK2999694T3 (pt)
ES (1) ES2627739T3 (pt)
IL (1) IL242512B (pt)
MX (1) MX361995B (pt)
TW (1) TWI631106B (pt)
WO (1) WO2014187773A1 (pt)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2015016119A (es) * 2013-05-22 2016-03-31 Bayer Cropscience Ag Metodo para preparar derivados de 3,5-bis(fluoroalquil)pirazol.
CN108473433A (zh) * 2016-01-21 2018-08-31 拜耳作物科学股份公司 制备多氟烷基化的喹啉的方法

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6277371A (ja) * 1985-09-30 1987-04-09 Neos Co Ltd 含フツ素ピラゾ−ル誘導体
HUP0104324A3 (en) * 1996-06-20 2002-04-29 Monsanto Co Preparation of substituted 3-aryl-5-halogenalkyl-pyrazoles having herbicidal activity
DE10215292A1 (de) 2002-02-19 2003-08-28 Bayer Cropscience Ag Disubstitutierte Pyrazolylcarbocanilide
DE10349500A1 (de) 2003-10-23 2005-06-02 Bayer Cropscience Ag Verfahren zum Herstellen von 2-Dihalogenacyl-3-amino-acrylsäureestern und 3-Dihalogenmethyl-pyrazol-4-carbonsäureestern
WO2008013622A2 (en) * 2006-07-27 2008-01-31 E. I. Du Pont De Nemours And Company Fungicidal azocyclic amides
DE102006039909A1 (de) * 2006-08-25 2008-03-13 Bayer Cropscience Ag Verfahren zum Herstellen von 3-Dihalomethyl-pyrazol-4-carbonsäurederivaten
EP2133341A1 (de) 2008-02-25 2009-12-16 Bayer CropScience AG Verfahren zur regioselektiven Synthese von 1-Alkyl-3-haloalkyl-pyrazol-4-carbonsäure-Derivaten
EP2100883A1 (de) 2008-03-10 2009-09-16 Bayer CropScience AG Verfahren zur regioselektiven Synthese von 1-Alkyl-3-haloalkyl-pyrazol-4carbonsäure-Derivaten
US8759527B2 (en) 2010-08-25 2014-06-24 Bayer Cropscience Ag Heteroarylpiperidine and -piperazine derivatives as fungicides
MX2015016119A (es) * 2013-05-22 2016-03-31 Bayer Cropscience Ag Metodo para preparar derivados de 3,5-bis(fluoroalquil)pirazol.

Also Published As

Publication number Publication date
IL242512B (en) 2018-06-28
CN105408314A (zh) 2016-03-16
WO2014187773A1 (en) 2014-11-27
MX2015015720A (es) 2016-03-07
BR112015028751B1 (pt) 2021-01-12
JP2016523838A (ja) 2016-08-12
TWI631106B (zh) 2018-08-01
EP2999694B1 (en) 2017-05-17
KR20160009573A (ko) 2016-01-26
EP2999694A1 (en) 2016-03-30
JP6377727B2 (ja) 2018-08-22
ES2627739T3 (es) 2017-07-31
US9512081B2 (en) 2016-12-06
KR102233655B1 (ko) 2021-03-31
TW201536747A (zh) 2015-10-01
CN105408314B (zh) 2018-04-24
DK2999694T3 (en) 2017-06-19
MX361995B (es) 2018-12-19
US20160108000A1 (en) 2016-04-21

Similar Documents

Publication Publication Date Title
BR112018010118A2 (pt) inibidores de cxcr2
BR112016029333A2 (pt) síntese de compostos de carbamoilpiridona policíclico
TR201909606T4 (tr) Pi̇razollari hazirlamak i̇çi̇n i̇şlem
BR112015029933A2 (pt) método de produção de tagatose
BR112016014020A8 (pt) moduladores de tetra-hidropiridopirazinas de gpr6.
EA201590951A1 (ru) Дигидропиразольные модуляторы gpr40
MX2018001793A (es) Compuestos para dispositivos opticamente activos.
EA201590954A1 (ru) Дигидропиразольные модуляторы gpr40
EA201590949A1 (ru) Дигидропиразольные модуляторы gpr40
BR112015029399A2 (pt) produção em etapa única de uma composição de polipropileno
BR112017019850A2 (pt) ?processo melhorado para a preparação de apremilast?
EA201691999A1 (ru) Новые сульфониламинобензамидные соединения
BR112016011899A2 (pt) Processo para preparação de 5-fluoro-1h-pirazóis
BR112017018993A2 (pt) Processo para preparar 3-cloro-2- vinilfenilassulfonatos
NZ720106A (en) A process for the preparation of regadenoson
BR112016027455A2 (pt) moduladores ppar
BR112017011275A2 (pt) composição, e, processo para a produção de xarope de glicose.
BR112012026157A2 (pt) processo para preparar ditiina-tetracarboximidas.
BR112015024859A2 (pt) processo e intermediários para a preparação de pregabalina
BR112016016397A2 (pt) método para preparar 1-alquil-3-difluorometil-5-fluoro-1h-pirazol-4-carbaldeídos e 1-alquil-3-difluorometil-5-fluoro-1h-pirazol-4-carboxilatos.
BR112012026411A2 (pt) processo para preparar ditiina-tetracarboxi-diiminas
BR112016027819A8 (pt) processo de preparação de derivados de tiazole
MX350122B (es) Tinturas dispersas, su preparación y su uso.
BR112012029626A2 (pt) processo para preparar ditianona-tetracarboxi-dimidas
BR112015028751A2 (pt) processo para a preparação de derivados de 3,5-bis (fluoralquil)pirazol a partir de alfa,alfa-dihaloaminas

Legal Events

Date Code Title Description
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B06U Preliminary requirement: requests with searches performed by other patent offices: procedure suspended [chapter 6.21 patent gazette]
B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B06I Publication of requirement cancelled [chapter 6.9 patent gazette]

Free format text: ANULADA A PUBLICACAO CODIGO 6.1 NA RPI NO 2592 DE 08/09/2020 POR TER SIDO INDEVIDA.

B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 19/05/2014, OBSERVADAS AS CONDICOES LEGAIS.