BR112014009220A2 - uso de derivados de aminoacetonitrila contra endoparasitas - Google Patents
uso de derivados de aminoacetonitrila contra endoparasitasInfo
- Publication number
- BR112014009220A2 BR112014009220A2 BR112014009220A BR112014009220A BR112014009220A2 BR 112014009220 A2 BR112014009220 A2 BR 112014009220A2 BR 112014009220 A BR112014009220 A BR 112014009220A BR 112014009220 A BR112014009220 A BR 112014009220A BR 112014009220 A2 BR112014009220 A2 BR 112014009220A2
- Authority
- BR
- Brazil
- Prior art keywords
- compound
- derivatives against
- against endoparasites
- aminoacetonitrile derivatives
- stereoisomer
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/275—Nitriles; Isonitriles
- A61K31/277—Nitriles; Isonitriles having a ring, e.g. verapamil
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C381/00—Compounds containing carbon and sulfur and having functional groups not covered by groups C07C301/00 - C07C337/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Tropical Medicine & Parasitology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
resumo patente de invenção: "uso de derivados de aminoacetonitrila contra endoparasitas". a presente invenção refere-se a um método de tratamento de uma infecção parasítica em um animal, particularmente uma infecção endoparasítica filária, compreendendo administrar uma quantidade eficaz de um composto de fórmula (i) ou um composto de fórmula (ii), (i) estereoisômero do mesmo, ou sal veterinariamente aceitável do referido composto ou estereoisômero do mesmo, ou em combinação com pelo menos um agente veterinário adicional, em que: r1, r2, r3, r4, r5, r1a, r1b, r1c, r1d, r1e são como descrito aqui.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201161549027P | 2011-10-19 | 2011-10-19 | |
PCT/IB2012/055436 WO2013057624A1 (en) | 2011-10-19 | 2012-10-08 | Use of aminoacetonitrile derivatives against endoparasites |
Publications (2)
Publication Number | Publication Date |
---|---|
BR112014009220A2 true BR112014009220A2 (pt) | 2017-06-13 |
BR112014009220A8 BR112014009220A8 (pt) | 2017-06-20 |
Family
ID=47278351
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112014009220A BR112014009220A8 (pt) | 2011-10-19 | 2012-10-08 | uso de derivados de aminoacetonitrila contra endoparasitas |
Country Status (10)
Country | Link |
---|---|
US (1) | US8962681B2 (pt) |
EP (1) | EP2768497A1 (pt) |
JP (2) | JP2014530849A (pt) |
CN (1) | CN104271128A (pt) |
AR (1) | AR088461A1 (pt) |
AU (1) | AU2012324491A1 (pt) |
BR (1) | BR112014009220A8 (pt) |
CA (1) | CA2851412A1 (pt) |
MX (1) | MX2014004743A (pt) |
WO (1) | WO2013057624A1 (pt) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US10238677B2 (en) | 2015-01-09 | 2019-03-26 | Liverpool School Of Tropical Medicine | Treatment of filarial diseases |
CN107183328A (zh) * | 2017-06-28 | 2017-09-22 | 江苏农牧科技职业学院 | 一种防治血液寄生虫的宠物饲料及其制备方法 |
Family Cites Families (22)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
NO176766C (no) | 1989-02-07 | 1995-05-24 | Meiji Seika Kaisha | Fremgangsmåte for fremstilling av en forbindelse med anthelmintaktivitet |
JPH0570366A (ja) | 1991-03-08 | 1993-03-23 | Meiji Seika Kaisha Ltd | 薬用組成物 |
DK0634408T3 (da) | 1992-03-17 | 2002-04-22 | Fujisawa Pharmaceutical Co | Depsipeptidderivater, fremstilling og anvendelse deraf |
DE4317458A1 (de) | 1992-06-11 | 1993-12-16 | Bayer Ag | Verwendung von cyclischen Depsipeptiden mit 18 Ringatomen zur Bekämpfung von Endoparasiten, neue cyclische Depsipeptide mit 18 Ringatomen und Verfahren zu ihrer Herstellung |
WO1994019334A1 (en) | 1993-02-19 | 1994-09-01 | Meiji Seika Kaisha, Ltd. | Pf1022 derivative, cyclic depsipeptide |
DE4317457A1 (de) | 1993-05-26 | 1994-12-01 | Bayer Ag | Octacyclodepsipeptide mit endoparasitizider Wirkung |
DE4437198A1 (de) | 1994-10-18 | 1996-04-25 | Bayer Ag | Verfahren zur Sulfonylierung, Sulfenylierung und Phosphorylierung von cyclischen Depsipeptiden |
DE4440193A1 (de) | 1994-11-10 | 1996-05-15 | Bayer Ag | Verwendung von Dioxomorpholinen zur Bekämpfung von Endoparasiten, neue Dioxomorpholine und Verfahren zur ihrer Herstellung |
GB9518953D0 (en) | 1995-09-15 | 1995-11-15 | Pfizer Ltd | Pharmaceutical formulations |
GB0402677D0 (en) | 2003-11-06 | 2004-03-10 | Novartis Ag | Organic compounds |
AR046757A1 (es) * | 2003-12-10 | 2005-12-21 | Novartis Ag | Amidoacetonitrilos utiles como pesticidas |
ES2526614T3 (es) | 2004-03-05 | 2015-01-13 | Nissan Chemical Industries, Ltd. | Compuesto de benzamida sustituida con isoxazolina y agente de control de organismos nocivos |
TWI412322B (zh) | 2005-12-30 | 2013-10-21 | Du Pont | 控制無脊椎害蟲之異唑啉 |
EP1997813B1 (en) | 2006-03-10 | 2010-05-05 | Nissan Chemical Industries, Ltd. | Substituted isoxazoline compound and pest control agent |
SI2118055T1 (sl) * | 2007-02-09 | 2013-12-31 | Zoetis Uk Limited | Antiparazitska sredstva |
KR20110098012A (ko) * | 2007-02-09 | 2011-08-31 | 화이자 리미티드 | 구충제 |
ES2367332T3 (es) | 2007-02-21 | 2011-11-02 | Pfizer Limited | Agentes antiparasitarios de benzofurano. |
ME03373B (me) | 2007-05-15 | 2020-01-20 | Merial Inc | Ariloazol-2-il cijanoetilamino jedinjenja, postupci dobijanja i postupci njihove primene |
ES2666187T3 (es) | 2007-06-27 | 2018-05-03 | E. I. Du Pont De Nemours And Company | Procedimiento de control de plagas en animales |
NZ590756A (en) | 2008-09-04 | 2013-01-25 | Syngenta Participations Ag | Insecticidal compounds |
SI3050874T1 (sl) | 2008-11-14 | 2019-04-30 | Merial Inc. | Enantiomerno obogatene ariloazol-2-il cianoetilamino paraziticidne spojine |
US8168681B2 (en) | 2008-12-03 | 2012-05-01 | Novartis Ag | Amidoacetonitrile compounds and pesticidal composition thereof |
-
2012
- 2012-10-08 JP JP2014536363A patent/JP2014530849A/ja active Pending
- 2012-10-08 MX MX2014004743A patent/MX2014004743A/es unknown
- 2012-10-08 AU AU2012324491A patent/AU2012324491A1/en not_active Abandoned
- 2012-10-08 US US14/351,945 patent/US8962681B2/en not_active Expired - Fee Related
- 2012-10-08 CN CN201280063028.9A patent/CN104271128A/zh active Pending
- 2012-10-08 EP EP12794772.9A patent/EP2768497A1/en not_active Withdrawn
- 2012-10-08 CA CA2851412A patent/CA2851412A1/en not_active Abandoned
- 2012-10-08 WO PCT/IB2012/055436 patent/WO2013057624A1/en active Application Filing
- 2012-10-08 BR BR112014009220A patent/BR112014009220A8/pt not_active IP Right Cessation
- 2012-10-18 JP JP2012230471A patent/JP2013087120A/ja active Pending
- 2012-10-18 AR ARP120103892A patent/AR088461A1/es unknown
Also Published As
Publication number | Publication date |
---|---|
AR088461A1 (es) | 2014-06-11 |
EP2768497A1 (en) | 2014-08-27 |
AU2012324491A1 (en) | 2014-04-17 |
CA2851412A1 (en) | 2013-04-25 |
JP2014530849A (ja) | 2014-11-20 |
CN104271128A (zh) | 2015-01-07 |
US20140243408A1 (en) | 2014-08-28 |
BR112014009220A8 (pt) | 2017-06-20 |
US8962681B2 (en) | 2015-02-24 |
JP2013087120A (ja) | 2013-05-13 |
WO2013057624A9 (en) | 2014-10-30 |
MX2014004743A (es) | 2014-08-01 |
WO2013057624A1 (en) | 2013-04-25 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application fees: application dismissed [chapter 8.6 patent gazette] | ||
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] | ||
B350 | Update of information on the portal [chapter 15.35 patent gazette] |