BR112014009220A2 - uso de derivados de aminoacetonitrila contra endoparasitas - Google Patents

uso de derivados de aminoacetonitrila contra endoparasitas

Info

Publication number
BR112014009220A2
BR112014009220A2 BR112014009220A BR112014009220A BR112014009220A2 BR 112014009220 A2 BR112014009220 A2 BR 112014009220A2 BR 112014009220 A BR112014009220 A BR 112014009220A BR 112014009220 A BR112014009220 A BR 112014009220A BR 112014009220 A2 BR112014009220 A2 BR 112014009220A2
Authority
BR
Brazil
Prior art keywords
compound
derivatives against
against endoparasites
aminoacetonitrile derivatives
stereoisomer
Prior art date
Application number
BR112014009220A
Other languages
English (en)
Other versions
BR112014009220A8 (pt
Inventor
Jean Woods Debra
Anthony Conder George
Evans Kevin
F M Meeus Patrick
Original Assignee
Zoetis Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zoetis Llc filed Critical Zoetis Llc
Publication of BR112014009220A2 publication Critical patent/BR112014009220A2/pt
Publication of BR112014009220A8 publication Critical patent/BR112014009220A8/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/275Nitriles; Isonitriles
    • A61K31/277Nitriles; Isonitriles having a ring, e.g. verapamil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C381/00Compounds containing carbon and sulfur and having functional groups not covered by groups C07C301/00 - C07C337/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

resumo patente de invenção: "uso de derivados de aminoacetonitrila contra endoparasitas". a presente invenção refere-se a um método de tratamento de uma infecção parasítica em um animal, particularmente uma infecção endoparasítica filária, compreendendo administrar uma quantidade eficaz de um composto de fórmula (i) ou um composto de fórmula (ii), (i) estereoisômero do mesmo, ou sal veterinariamente aceitável do referido composto ou estereoisômero do mesmo, ou em combinação com pelo menos um agente veterinário adicional, em que: r1, r2, r3, r4, r5, r1a, r1b, r1c, r1d, r1e são como descrito aqui.
BR112014009220A 2011-10-19 2012-10-08 uso de derivados de aminoacetonitrila contra endoparasitas BR112014009220A8 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201161549027P 2011-10-19 2011-10-19
PCT/IB2012/055436 WO2013057624A1 (en) 2011-10-19 2012-10-08 Use of aminoacetonitrile derivatives against endoparasites

Publications (2)

Publication Number Publication Date
BR112014009220A2 true BR112014009220A2 (pt) 2017-06-13
BR112014009220A8 BR112014009220A8 (pt) 2017-06-20

Family

ID=47278351

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112014009220A BR112014009220A8 (pt) 2011-10-19 2012-10-08 uso de derivados de aminoacetonitrila contra endoparasitas

Country Status (10)

Country Link
US (1) US8962681B2 (pt)
EP (1) EP2768497A1 (pt)
JP (2) JP2014530849A (pt)
CN (1) CN104271128A (pt)
AR (1) AR088461A1 (pt)
AU (1) AU2012324491A1 (pt)
BR (1) BR112014009220A8 (pt)
CA (1) CA2851412A1 (pt)
MX (1) MX2014004743A (pt)
WO (1) WO2013057624A1 (pt)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US10238677B2 (en) 2015-01-09 2019-03-26 Liverpool School Of Tropical Medicine Treatment of filarial diseases
CN107183328A (zh) * 2017-06-28 2017-09-22 江苏农牧科技职业学院 一种防治血液寄生虫的宠物饲料及其制备方法

Family Cites Families (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NO176766C (no) 1989-02-07 1995-05-24 Meiji Seika Kaisha Fremgangsmåte for fremstilling av en forbindelse med anthelmintaktivitet
JPH0570366A (ja) 1991-03-08 1993-03-23 Meiji Seika Kaisha Ltd 薬用組成物
DK0634408T3 (da) 1992-03-17 2002-04-22 Fujisawa Pharmaceutical Co Depsipeptidderivater, fremstilling og anvendelse deraf
DE4317458A1 (de) 1992-06-11 1993-12-16 Bayer Ag Verwendung von cyclischen Depsipeptiden mit 18 Ringatomen zur Bekämpfung von Endoparasiten, neue cyclische Depsipeptide mit 18 Ringatomen und Verfahren zu ihrer Herstellung
WO1994019334A1 (en) 1993-02-19 1994-09-01 Meiji Seika Kaisha, Ltd. Pf1022 derivative, cyclic depsipeptide
DE4317457A1 (de) 1993-05-26 1994-12-01 Bayer Ag Octacyclodepsipeptide mit endoparasitizider Wirkung
DE4437198A1 (de) 1994-10-18 1996-04-25 Bayer Ag Verfahren zur Sulfonylierung, Sulfenylierung und Phosphorylierung von cyclischen Depsipeptiden
DE4440193A1 (de) 1994-11-10 1996-05-15 Bayer Ag Verwendung von Dioxomorpholinen zur Bekämpfung von Endoparasiten, neue Dioxomorpholine und Verfahren zur ihrer Herstellung
GB9518953D0 (en) 1995-09-15 1995-11-15 Pfizer Ltd Pharmaceutical formulations
GB0402677D0 (en) 2003-11-06 2004-03-10 Novartis Ag Organic compounds
AR046757A1 (es) * 2003-12-10 2005-12-21 Novartis Ag Amidoacetonitrilos utiles como pesticidas
ES2526614T3 (es) 2004-03-05 2015-01-13 Nissan Chemical Industries, Ltd. Compuesto de benzamida sustituida con isoxazolina y agente de control de organismos nocivos
TWI412322B (zh) 2005-12-30 2013-10-21 Du Pont 控制無脊椎害蟲之異唑啉
EP1997813B1 (en) 2006-03-10 2010-05-05 Nissan Chemical Industries, Ltd. Substituted isoxazoline compound and pest control agent
SI2118055T1 (sl) * 2007-02-09 2013-12-31 Zoetis Uk Limited Antiparazitska sredstva
KR20110098012A (ko) * 2007-02-09 2011-08-31 화이자 리미티드 구충제
ES2367332T3 (es) 2007-02-21 2011-11-02 Pfizer Limited Agentes antiparasitarios de benzofurano.
ME03373B (me) 2007-05-15 2020-01-20 Merial Inc Ariloazol-2-il cijanoetilamino jedinjenja, postupci dobijanja i postupci njihove primene
ES2666187T3 (es) 2007-06-27 2018-05-03 E. I. Du Pont De Nemours And Company Procedimiento de control de plagas en animales
NZ590756A (en) 2008-09-04 2013-01-25 Syngenta Participations Ag Insecticidal compounds
SI3050874T1 (sl) 2008-11-14 2019-04-30 Merial Inc. Enantiomerno obogatene ariloazol-2-il cianoetilamino paraziticidne spojine
US8168681B2 (en) 2008-12-03 2012-05-01 Novartis Ag Amidoacetonitrile compounds and pesticidal composition thereof

Also Published As

Publication number Publication date
AR088461A1 (es) 2014-06-11
EP2768497A1 (en) 2014-08-27
AU2012324491A1 (en) 2014-04-17
CA2851412A1 (en) 2013-04-25
JP2014530849A (ja) 2014-11-20
CN104271128A (zh) 2015-01-07
US20140243408A1 (en) 2014-08-28
BR112014009220A8 (pt) 2017-06-20
US8962681B2 (en) 2015-02-24
JP2013087120A (ja) 2013-05-13
WO2013057624A9 (en) 2014-10-30
MX2014004743A (es) 2014-08-01
WO2013057624A1 (en) 2013-04-25

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Legal Events

Date Code Title Description
B08F Application fees: application dismissed [chapter 8.6 patent gazette]
B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]
B350 Update of information on the portal [chapter 15.35 patent gazette]