BR112012027520A2 - formulações e usos de derivados de ácido 2-hidroxi-5-fenilazobenzoico para o tratamento de indivíduos do sexo masculino - Google Patents
formulações e usos de derivados de ácido 2-hidroxi-5-fenilazobenzoico para o tratamento de indivíduos do sexo masculinoInfo
- Publication number
- BR112012027520A2 BR112012027520A2 BR112012027520A BR112012027520A BR112012027520A2 BR 112012027520 A2 BR112012027520 A2 BR 112012027520A2 BR 112012027520 A BR112012027520 A BR 112012027520A BR 112012027520 A BR112012027520 A BR 112012027520A BR 112012027520 A2 BR112012027520 A2 BR 112012027520A2
- Authority
- BR
- Brazil
- Prior art keywords
- males
- formulations
- hydroxy
- treatment
- acid derivatives
- Prior art date
Links
- 239000000203 mixture Substances 0.000 title abstract 3
- JHDYSXXPQIFFJZ-UHFFFAOYSA-N chembl1834961 Chemical class C1=C(O)C(C(=O)O)=CC(N=NC=2C=CC=CC=2)=C1 JHDYSXXPQIFFJZ-UHFFFAOYSA-N 0.000 title abstract 2
- 238000009472 formulation Methods 0.000 title abstract 2
- 206010009900 Colitis ulcerative Diseases 0.000 abstract 1
- 201000006704 Ulcerative Colitis Diseases 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/655—Azo (—N=N—), diazo (=N2), azoxy (>N—O—N< or N(=O)—N<), azido (—N3) or diazoamino (—N=N—N<) compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/06—Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
Landscapes
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| BR122014009845A BR122014009845A2 (pt) | 2010-04-26 | 2011-04-26 | usos de balsalazida para preparação de composição farmacêutica para tratamento de distúrbio gastrointestinal e induzir remissão clínica de colite ulcerativa em indivíduos do sexo masculino, bem como para diminuir o escore de mmdai e cicatrização da mucosa em indivíduos do sexo masculino com colite ulcerativa |
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US32815110P | 2010-04-26 | 2010-04-26 | |
| PCT/US2011/033905 WO2011137103A1 (en) | 2010-04-26 | 2011-04-26 | Formulations and uses of 2-hydroxy-5-phenylazobenzoic acid derivatives for the treatment of males |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR112012027520A2 true BR112012027520A2 (pt) | 2015-09-15 |
Family
ID=44861888
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR112012027520A BR112012027520A2 (pt) | 2010-04-26 | 2011-04-26 | formulações e usos de derivados de ácido 2-hidroxi-5-fenilazobenzoico para o tratamento de indivíduos do sexo masculino |
| BR122014009845A BR122014009845A2 (pt) | 2010-04-26 | 2011-04-26 | usos de balsalazida para preparação de composição farmacêutica para tratamento de distúrbio gastrointestinal e induzir remissão clínica de colite ulcerativa em indivíduos do sexo masculino, bem como para diminuir o escore de mmdai e cicatrização da mucosa em indivíduos do sexo masculino com colite ulcerativa |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR122014009845A BR122014009845A2 (pt) | 2010-04-26 | 2011-04-26 | usos de balsalazida para preparação de composição farmacêutica para tratamento de distúrbio gastrointestinal e induzir remissão clínica de colite ulcerativa em indivíduos do sexo masculino, bem como para diminuir o escore de mmdai e cicatrização da mucosa em indivíduos do sexo masculino com colite ulcerativa |
Country Status (9)
| Country | Link |
|---|---|
| US (3) | US8497256B2 (enExample) |
| EP (1) | EP2563117B1 (enExample) |
| JP (1) | JP2013525440A (enExample) |
| AU (1) | AU2011245455A1 (enExample) |
| BR (2) | BR112012027520A2 (enExample) |
| CA (1) | CA2797560A1 (enExample) |
| IL (1) | IL222642A0 (enExample) |
| MX (1) | MX358142B (enExample) |
| WO (1) | WO2011137103A1 (enExample) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP3801489A4 (en) | 2018-06-05 | 2022-03-30 | Flagship Pioneering Innovations V, Inc. | Acylated active agents and methods of their use for the treatment of autoimmune disorders |
Family Cites Families (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US326364A (en) | 1885-09-15 | Electric-lamp hanger | ||
| US4298595A (en) | 1978-12-20 | 1981-11-03 | Dynapol | Pharmaceutical preparations containing a polymeric agent for releasing 5-aminosalicylic acid or its salts into the gastrointestinal tract |
| DE3887353T2 (de) | 1987-10-12 | 1994-05-05 | Capability Services Pty Ltd | Behandlungsverfahren für magen-darm-krankheiten. |
| US5443826A (en) | 1988-08-02 | 1995-08-22 | Borody; Thomas J. | Treatment of gastro-intestinal disorders with a fecal composition or a composition of bacteroides and E. Coli |
| US5519014A (en) | 1990-10-22 | 1996-05-21 | Borody; Thomas J. | Treatment of non-inflammatory and non-infectious bowel disorders |
| US5498608A (en) | 1994-01-07 | 1996-03-12 | Salix Pharmaceuticals | Use of 2-hydroxy-5-phenylazobenzoic acid derivatives as colon cancer chemopreventative and chemotherapeutic agents |
| US5905073A (en) | 1995-01-06 | 1999-05-18 | Salix Pharmaceuticals, Inc. | Use of 2-hydroxy-5-phenylazobenzoic acid derivatives as colon cancer chemopreventative and chemotherapeutic agents |
| SE9700934D0 (sv) | 1997-03-14 | 1997-03-14 | Astra Ab | New formulation |
| US6551632B2 (en) | 1997-04-01 | 2003-04-22 | Thomas Julius Borody | Methods and compositions for treating inflammatory bowel disease |
| WO1998043667A1 (en) | 1997-04-01 | 1998-10-08 | Borody Thomas J | Methods and compositions for treating inflammatory bowel disease |
| AUPO665397A0 (en) | 1997-05-07 | 1997-05-29 | Borody, Thomas Julius | Novel therapy for constipation |
| AUPP437698A0 (en) | 1998-06-30 | 1998-07-23 | Baumgart, Karl | Methods for treatment of coronary, carotid and other vascular disease |
| US6326364B1 (en) | 1999-02-08 | 2001-12-04 | Cedars-Sinai Medical Center | Use of 5-aminosalicylates as antimicrobial agents |
| US7452872B2 (en) * | 2005-08-24 | 2008-11-18 | Salix Pharmaceuticals, Inc. | Formulations and uses of 2-hydroxy-5-phenylazobenzoic acid derivatives |
| EP2586427A3 (en) | 2005-08-24 | 2013-05-29 | Salix Pharmaceuticals, Inc. | Balsalazide formulations and manufacture thereof |
| US8921344B2 (en) * | 2006-11-03 | 2014-12-30 | Salix Pharmaceuticals, Inc. | Formulations and uses of 2-hydroxy-5-phenylazobenzoic acid derivatives |
| WO2008033125A1 (en) | 2006-09-13 | 2008-03-20 | The Procter & Gamble Company | Methods of treatment for ulcerative colitis using aminosalicylate |
-
2011
- 2011-04-26 EP EP11775497.8A patent/EP2563117B1/en active Active
- 2011-04-26 CA CA2797560A patent/CA2797560A1/en not_active Withdrawn
- 2011-04-26 BR BR112012027520A patent/BR112012027520A2/pt not_active IP Right Cessation
- 2011-04-26 US US13/094,261 patent/US8497256B2/en active Active
- 2011-04-26 BR BR122014009845A patent/BR122014009845A2/pt not_active Application Discontinuation
- 2011-04-26 JP JP2013508147A patent/JP2013525440A/ja active Pending
- 2011-04-26 MX MX2012012324A patent/MX358142B/es active IP Right Grant
- 2011-04-26 AU AU2011245455A patent/AU2011245455A1/en not_active Abandoned
- 2011-04-26 WO PCT/US2011/033905 patent/WO2011137103A1/en not_active Ceased
-
2012
- 2012-10-23 IL IL222642A patent/IL222642A0/en unknown
-
2013
- 2013-07-10 US US13/938,777 patent/US20130295178A1/en not_active Abandoned
-
2014
- 2014-10-08 US US14/509,446 patent/US20150132381A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| US20120058184A1 (en) | 2012-03-08 |
| WO2011137103A1 (en) | 2011-11-03 |
| EP2563117A4 (en) | 2013-09-04 |
| IL222642A0 (en) | 2012-12-31 |
| CA2797560A1 (en) | 2011-11-03 |
| BR122014009845A2 (pt) | 2015-12-29 |
| MX358142B (es) | 2018-08-06 |
| AU2011245455A1 (en) | 2012-11-15 |
| EP2563117A1 (en) | 2013-03-06 |
| EP2563117B1 (en) | 2018-02-21 |
| US20150132381A1 (en) | 2015-05-14 |
| US8497256B2 (en) | 2013-07-30 |
| JP2013525440A (ja) | 2013-06-20 |
| MX2012012324A (es) | 2013-01-29 |
| US20130295178A1 (en) | 2013-11-07 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
| B06T | Formal requirements before examination [chapter 6.20 patent gazette] | ||
| B07D | Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette] |
Free format text: DE ACORDO COM O ARTIGO 229-C DA LEI NO 10196/2001, QUE MODIFICOU A LEI NO 9279/96, A CONCESSAO DA PATENTE ESTA CONDICIONADA A ANUENCIA PREVIA DA ANVISA. CONSIDERANDO A APROVACAO DOS TERMOS DO PARECER NO 337/PGF/EA/2010, BEM COMO A PORTARIA INTERMINISTERIAL NO 1065 DE 24/05/2012, ENCAMINHA-SE O PRESENTE PEDIDO PARA AS PROVIDENCIAS CABIVEIS. |
|
| B07E | Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette] | ||
| B15K | Others concerning applications: alteration of classification |
Free format text: A CLASSIFICACAO ANTERIOR ERA: A01N 33/26 Ipc: A61K 31/655 (2006.01), A61K 9/28 (2006.01), A61K 9 |
|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 10A ANUIDADE. |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2622 DE 06/04/2021. |