BR1100678A - Tetrahidro-benzoatiazol, sua preparação e seu uso como produto intermediário ou como medicamento - Google Patents

Tetrahidro-benzoatiazol, sua preparação e seu uso como produto intermediário ou como medicamento

Info

Publication number
BR1100678A
BR1100678A BR1100678-1A BR1100678A BR1100678A BR 1100678 A BR1100678 A BR 1100678A BR 1100678 A BR1100678 A BR 1100678A BR 1100678 A BR1100678 A BR 1100678A
Authority
BR
Brazil
Prior art keywords
benzoatiazole
tetrahydro
medicine
preparation
intermediate product
Prior art date
Application number
BR1100678-1A
Other languages
English (en)
Portuguese (pt)
Inventor
Gerhart Griss
Claus Schneider
Rudolf Hurnaus
Walter Kobinger
Ludwig Pichler
Rudolf Bauer
Joachim Mierau
Dieter Hinzen
Guenter Schingnitz
Original Assignee
Gerhart Griss
Claus Schneider
Rudolf Hurnaus
Walter Kobinger
Ludwig Pichler
Rudolf Bauer
Joachim Mierau
Dieter Hinzen
Guenter Schingnitz
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gerhart Griss, Claus Schneider, Rudolf Hurnaus, Walter Kobinger, Ludwig Pichler, Rudolf Bauer, Joachim Mierau, Dieter Hinzen, Guenter Schingnitz filed Critical Gerhart Griss
Publication of BR1100678A publication Critical patent/BR1100678A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62Benzothiazoles
    • C07D277/68Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D277/82Nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Health & Medical Sciences (AREA)
  • Cardiology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
BR1100678-1A 1984-12-22 1997-05-08 Tetrahidro-benzoatiazol, sua preparação e seu uso como produto intermediário ou como medicamento BR1100678A (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19843447075 DE3447075A1 (de) 1984-12-22 1984-12-22 Tetrahydro-benzthiazole, deren herstellung und deren verwendung als zwischenprodukte oder als arzneimittel

Publications (1)

Publication Number Publication Date
BR1100678A true BR1100678A (pt) 1999-10-13

Family

ID=6253655

Family Applications (1)

Application Number Title Priority Date Filing Date
BR1100678-1A BR1100678A (pt) 1984-12-22 1997-05-08 Tetrahidro-benzoatiazol, sua preparação e seu uso como produto intermediário ou como medicamento

Country Status (5)

Country Link
JP (1) JPS61155377A (es)
BR (1) BR1100678A (es)
DD (1) DD242230A5 (es)
DE (1) DE3447075A1 (es)
ZA (1) ZA859731B (es)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3620813A1 (de) * 1986-06-21 1987-12-23 Boehringer Ingelheim Kg Neue tetrahydro-benzothiazole, ihre herstellung und verwendung
US5650420A (en) * 1994-12-15 1997-07-22 Pharmacia & Upjohn Company Pramipexole as a neuroprotective agent
SE9802360D0 (sv) * 1998-07-01 1998-07-01 Wikstroem Hakan Vilhelm New 2-aminothiazol-fused 2-aminoindans and 2-aminotetralins ((basic)-N-substituted and (basic)-N,N-disubstituted derivatives of 2,6-diamino-thiazolo(4,5-f)indan and 2,7-di-amino-thiazolo(4,5-g)tetralin
US6277875B1 (en) * 2000-07-17 2001-08-21 Andrew J. Holman Use of dopamine D2/D3 receptor agonists to treat fibromyalgia
CA2468747C (en) * 2001-12-11 2011-05-31 University Of Virginia Patent Foundation Use of pramipexole to treat amyotrophic lateral sclerosis
US20050226926A1 (en) * 2002-07-25 2005-10-13 Pfizer Inc Sustained-release tablet composition of pramipexole
AR040680A1 (es) * 2002-07-25 2005-04-13 Pharmacia Corp Composicion de tabletas de liberacion sostenida
GB2394951A (en) * 2002-11-04 2004-05-12 Cipla Ltd One pot synthesis of 2,6-diamino-4,5,6,7-tetrahydro-benzothiazole
DE102004006808A1 (de) * 2004-02-11 2005-09-01 Grünenthal GmbH Substituierte 4,5,6,7-Tetrahydro-benzothiazol-2-ylamin-Verbindungen
US7741490B2 (en) * 2004-03-19 2010-06-22 Dipharma S.P.A. Intermediates for the preparation of pramipexole
ES2245604B1 (es) * 2004-06-25 2006-12-01 Ragactives, S. L. Procedimiento para la obtencion de 2-amino-6-alquil-amino-4,5,6,7-tetrahidrobenzotiazoles.
ES2264378B1 (es) * 2005-05-09 2007-11-01 Ragactives, S.L. Procedimiento para la resolucion de 2-amino-6propilamino-4,5,6,7-tetrahidrobenzotiazol y compuestos intermedios.
RU2454409C2 (ru) 2007-03-14 2012-06-27 Нопп Ньюросайенсиз, Инк. Синтез хирально очищенных замещенных бензотиазолдиаминов
US20100130569A1 (en) 2007-05-11 2010-05-27 Saten Pharmaceutical Co., Ltd. Prophylactic or therapeutic agent for posterior ocular disease comprising non-ergot selective d2 receptor agonist as active ingredient
CA2734491A1 (en) 2008-08-19 2010-02-25 Knopp Neurosciences, Inc. Compositions and methods of using (r)-pramipexole
WO2013096816A1 (en) 2011-12-22 2013-06-27 Biogen Idec Ma Inc. Improved synthesis of amine substituted 4,5,6,7-tetrahydrobenzothiazole compounds
US9662313B2 (en) 2013-02-28 2017-05-30 Knopp Biosciences Llc Compositions and methods for treating amyotrophic lateral sclerosis in responders
AU2014306683B2 (en) 2013-08-13 2017-10-12 Knopp Biosciences Llc Compositions and methods for treating plasma cell disorders and B-cell prolymphocytic disorders
ES2871556T3 (es) 2013-08-13 2021-10-29 Knopp Biosciences Llc Composiciones y métodos para el tratamiento de la urticaria crónica

Also Published As

Publication number Publication date
JPS61155377A (ja) 1986-07-15
ZA859731B (en) 1987-08-26
DD242230A5 (de) 1987-01-21
DE3447075A1 (de) 1986-07-03
JPH0572907B2 (es) 1993-10-13

Similar Documents

Publication Publication Date Title
BR8701302A (pt) Compostos macrolideos,sua preparacao e seu uso
BR1100678A (pt) Tetrahidro-benzoatiazol, sua preparação e seu uso como produto intermediário ou como medicamento
DE3587577D1 (de) Antimykotische pharmazeutische Präparate.
DE3582124D1 (de) Absorbierbares calcitoninarzneimittel.
NO156835C (no) Sugbar engangsarti omr,det medisin og hygiene.
DE3787836D1 (de) Wegwerfwindel.
DE3783437D1 (de) Heilmittel.
BR8606825A (pt) Corantes reativos,sua preparacao e emprego
DK175685D0 (da) Jernholdige farmaceutiske praeparater
DE3576118D1 (de) Pharmazeutische praeparate.
FI850455A0 (fi) Farmaceutiska produkter.
DE3682960D1 (de) Pharmazeutische praeparate.
DK280085D0 (da) 7alfa-acylthio-9alfa,11alfa-epoxy-20-spirox-4-en-3,21-dioner samt deresfremstilling og anvendelse
NO874193D0 (no) Farmasoeytiske preparater.
DE3763519D1 (de) Heilnahrungsmittel.
BR8701897A (pt) Benzimidazoles e imidazopiridinas sulfonamidas,sua preparacao e sua aplicacao como medicamentos
IT8548385A0 (it) Composti maftalenici,loro preparazi one e loro impiego come medicamenti
BR8707933A (pt) Poliois furanicos,sua preparacao e utilizacao nos polioretanos
DK131586D0 (da) Transdermalt, antiallergisk, farmaceutisk praeparat
DK526985D0 (da) Polycykliske biocide forbindelser, deres fremstilling og mellemprodukter herved samt deres anvendelse i medicinske praeparationer
BR8004505A (pt) Compostos de cumarina, sua preparacao e seu emprego
DE3583536D1 (de) Substituierte und bruecken enthaltende pyridine, als heilmittel verwendbar.
IT8547704A0 (it) Diazepinoindoli,loro preparazione e loro impiego come medicamenti
BR7904952A (pt) Disazocorantes hidro-insoluveis,sua preparacao e seu emprego
MX9203663A (es) Acrecentamiento de actividad farmaceutica.

Legal Events

Date Code Title Description
AN Processing applications according to articles 230 and 231 of law 9279/96: notification of filing an application
HHFK Processing applications according to articles 230 and 231 of law 9.279/96: republication
MT Patent suspended - articles 230 and 231 of law 9279/96
HKAN Grant procedure suspended (correction) - according to articles 230 and 231 of law 9279/96
MT Patent suspended - articles 230 and 231 of law 9279/96
NB Patent issued - articles 230 and 231 of law 9279/96
B22O Other matters related to patents and certificates of addition of invention: legal action concerning patent

Free format text: INPI-52400.000708/06 39A VARA FEDERAL DO RIO DE JANEIRO PROC. NO 2005.51.01.527211-0 MANDATO DE INTIMACAO AUTOR: KARL THOMAE GMBH REU: INSTITUTO NACIONAL DA PROPRIEDADE INDUSTRIAL - INPI REQUER: CORRECAO DOS PRAZOS DE VIGENCIAS DAS PATENTES PI 1100593-3 E PI 1100678-1