BR1100678A - Tetrahidro-benzoatiazol, sua preparação e seu uso como produto intermediário ou como medicamento - Google Patents
Tetrahidro-benzoatiazol, sua preparação e seu uso como produto intermediário ou como medicamentoInfo
- Publication number
- BR1100678A BR1100678A BR1100678-1A BR1100678A BR1100678A BR 1100678 A BR1100678 A BR 1100678A BR 1100678 A BR1100678 A BR 1100678A BR 1100678 A BR1100678 A BR 1100678A
- Authority
- BR
- Brazil
- Prior art keywords
- benzoatiazole
- tetrahydro
- medicine
- preparation
- intermediate product
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D277/82—Nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Medicinal Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Health & Medical Sciences (AREA)
- Cardiology (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Heart & Thoracic Surgery (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19843447075 DE3447075A1 (de) | 1984-12-22 | 1984-12-22 | Tetrahydro-benzthiazole, deren herstellung und deren verwendung als zwischenprodukte oder als arzneimittel |
Publications (1)
Publication Number | Publication Date |
---|---|
BR1100678A true BR1100678A (pt) | 1999-10-13 |
Family
ID=6253655
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR1100678-1A BR1100678A (pt) | 1984-12-22 | 1997-05-08 | Tetrahidro-benzoatiazol, sua preparação e seu uso como produto intermediário ou como medicamento |
Country Status (5)
Country | Link |
---|---|
JP (1) | JPS61155377A (es) |
BR (1) | BR1100678A (es) |
DD (1) | DD242230A5 (es) |
DE (1) | DE3447075A1 (es) |
ZA (1) | ZA859731B (es) |
Families Citing this family (19)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3620813A1 (de) * | 1986-06-21 | 1987-12-23 | Boehringer Ingelheim Kg | Neue tetrahydro-benzothiazole, ihre herstellung und verwendung |
US5650420A (en) * | 1994-12-15 | 1997-07-22 | Pharmacia & Upjohn Company | Pramipexole as a neuroprotective agent |
SE9802360D0 (sv) * | 1998-07-01 | 1998-07-01 | Wikstroem Hakan Vilhelm | New 2-aminothiazol-fused 2-aminoindans and 2-aminotetralins ((basic)-N-substituted and (basic)-N,N-disubstituted derivatives of 2,6-diamino-thiazolo(4,5-f)indan and 2,7-di-amino-thiazolo(4,5-g)tetralin |
US6277875B1 (en) * | 2000-07-17 | 2001-08-21 | Andrew J. Holman | Use of dopamine D2/D3 receptor agonists to treat fibromyalgia |
CA2468747C (en) * | 2001-12-11 | 2011-05-31 | University Of Virginia Patent Foundation | Use of pramipexole to treat amyotrophic lateral sclerosis |
US20050226926A1 (en) * | 2002-07-25 | 2005-10-13 | Pfizer Inc | Sustained-release tablet composition of pramipexole |
AR040680A1 (es) * | 2002-07-25 | 2005-04-13 | Pharmacia Corp | Composicion de tabletas de liberacion sostenida |
GB2394951A (en) * | 2002-11-04 | 2004-05-12 | Cipla Ltd | One pot synthesis of 2,6-diamino-4,5,6,7-tetrahydro-benzothiazole |
DE102004006808A1 (de) * | 2004-02-11 | 2005-09-01 | Grünenthal GmbH | Substituierte 4,5,6,7-Tetrahydro-benzothiazol-2-ylamin-Verbindungen |
US7741490B2 (en) * | 2004-03-19 | 2010-06-22 | Dipharma S.P.A. | Intermediates for the preparation of pramipexole |
ES2245604B1 (es) * | 2004-06-25 | 2006-12-01 | Ragactives, S. L. | Procedimiento para la obtencion de 2-amino-6-alquil-amino-4,5,6,7-tetrahidrobenzotiazoles. |
ES2264378B1 (es) * | 2005-05-09 | 2007-11-01 | Ragactives, S.L. | Procedimiento para la resolucion de 2-amino-6propilamino-4,5,6,7-tetrahidrobenzotiazol y compuestos intermedios. |
RU2454409C2 (ru) | 2007-03-14 | 2012-06-27 | Нопп Ньюросайенсиз, Инк. | Синтез хирально очищенных замещенных бензотиазолдиаминов |
US20100130569A1 (en) | 2007-05-11 | 2010-05-27 | Saten Pharmaceutical Co., Ltd. | Prophylactic or therapeutic agent for posterior ocular disease comprising non-ergot selective d2 receptor agonist as active ingredient |
CA2734491A1 (en) | 2008-08-19 | 2010-02-25 | Knopp Neurosciences, Inc. | Compositions and methods of using (r)-pramipexole |
WO2013096816A1 (en) | 2011-12-22 | 2013-06-27 | Biogen Idec Ma Inc. | Improved synthesis of amine substituted 4,5,6,7-tetrahydrobenzothiazole compounds |
US9662313B2 (en) | 2013-02-28 | 2017-05-30 | Knopp Biosciences Llc | Compositions and methods for treating amyotrophic lateral sclerosis in responders |
AU2014306683B2 (en) | 2013-08-13 | 2017-10-12 | Knopp Biosciences Llc | Compositions and methods for treating plasma cell disorders and B-cell prolymphocytic disorders |
ES2871556T3 (es) | 2013-08-13 | 2021-10-29 | Knopp Biosciences Llc | Composiciones y métodos para el tratamiento de la urticaria crónica |
-
1984
- 1984-12-22 DE DE19843447075 patent/DE3447075A1/de not_active Withdrawn
-
1985
- 1985-12-20 DD DD85284921A patent/DD242230A5/de not_active IP Right Cessation
- 1985-12-20 JP JP60287601A patent/JPS61155377A/ja active Granted
- 1985-12-20 ZA ZA859731A patent/ZA859731B/xx unknown
-
1997
- 1997-05-08 BR BR1100678-1A patent/BR1100678A/pt active IP Right Grant
Also Published As
Publication number | Publication date |
---|---|
JPS61155377A (ja) | 1986-07-15 |
ZA859731B (en) | 1987-08-26 |
DD242230A5 (de) | 1987-01-21 |
DE3447075A1 (de) | 1986-07-03 |
JPH0572907B2 (es) | 1993-10-13 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
AN | Processing applications according to articles 230 and 231 of law 9279/96: notification of filing an application | ||
HHFK | Processing applications according to articles 230 and 231 of law 9.279/96: republication | ||
MT | Patent suspended - articles 230 and 231 of law 9279/96 | ||
HKAN | Grant procedure suspended (correction) - according to articles 230 and 231 of law 9279/96 | ||
MT | Patent suspended - articles 230 and 231 of law 9279/96 | ||
NB | Patent issued - articles 230 and 231 of law 9279/96 | ||
B22O | Other matters related to patents and certificates of addition of invention: legal action concerning patent |
Free format text: INPI-52400.000708/06 39A VARA FEDERAL DO RIO DE JANEIRO PROC. NO 2005.51.01.527211-0 MANDATO DE INTIMACAO AUTOR: KARL THOMAE GMBH REU: INSTITUTO NACIONAL DA PROPRIEDADE INDUSTRIAL - INPI REQUER: CORRECAO DOS PRAZOS DE VIGENCIAS DAS PATENTES PI 1100593-3 E PI 1100678-1 |