BR0307369A - Uso de 4-(2-fluoro-fenil)-6-metil-2-(1-piperazinil)-tieno (2,3-d)-pirimidina para o tratamento de incontinência urinária - Google Patents
Uso de 4-(2-fluoro-fenil)-6-metil-2-(1-piperazinil)-tieno (2,3-d)-pirimidina para o tratamento de incontinência urináriaInfo
- Publication number
- BR0307369A BR0307369A BR0307369-6A BR0307369A BR0307369A BR 0307369 A BR0307369 A BR 0307369A BR 0307369 A BR0307369 A BR 0307369A BR 0307369 A BR0307369 A BR 0307369A
- Authority
- BR
- Brazil
- Prior art keywords
- thieno
- piperazinyl
- pyrimidine
- methyl
- treatment
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/10—Drugs for disorders of the urinary system of the bladder
Landscapes
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Urology & Nephrology (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Abstract
"USO DE 4-(2-FLUORO-FENIL)6-METIL-2-(1-PIPERAZINIL) TIENO (2,3-D)-PIRIMIDINA PARA O TRATAMENTO DE INCONTINêNCIA URINáRIA". A 4-(2-fluoro-fenil)-6-metil-2-(l-piperazinil) tieno (2,3-d) pirimidina, ou um sal da mesma, é útil para o tratamento de incontinência urinária.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB0202265.5A GB0202265D0 (en) | 2002-01-31 | 2002-01-31 | New therapeutic use |
PCT/GB2003/000374 WO2003063873A1 (en) | 2002-01-31 | 2003-01-29 | Use of 4-(2-fluorophenyl)-6-methyl-2-(1-piperazinyl)thieno(2, 3-d)-pyrimidine for treating of urinary incontinence |
Publications (1)
Publication Number | Publication Date |
---|---|
BR0307369A true BR0307369A (pt) | 2004-12-14 |
Family
ID=9930142
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR0307369-6A BR0307369A (pt) | 2002-01-31 | 2003-01-29 | Uso de 4-(2-fluoro-fenil)-6-metil-2-(1-piperazinil)-tieno (2,3-d)-pirimidina para o tratamento de incontinência urinária |
Country Status (14)
Country | Link |
---|---|
US (1) | US7220748B2 (pt) |
EP (1) | EP1469853B1 (pt) |
JP (1) | JP2005516977A (pt) |
KR (1) | KR20040081479A (pt) |
CN (1) | CN1279915C (pt) |
AT (1) | ATE397448T1 (pt) |
AU (1) | AU2003205836B2 (pt) |
BR (1) | BR0307369A (pt) |
CA (1) | CA2474851A1 (pt) |
DE (1) | DE60321445D1 (pt) |
ES (1) | ES2307896T3 (pt) |
GB (1) | GB0202265D0 (pt) |
PT (1) | PT1469853E (pt) |
WO (1) | WO2003063873A1 (pt) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0216027D0 (en) | 2002-07-10 | 2002-08-21 | Arachnova Therapeutics Ltd | New therapeutic use |
US20040048874A1 (en) * | 2001-05-22 | 2004-03-11 | Bardsley Hazel Judith | New therapeutic use of 4-(2-fluorophenyl)-6-methyl-2-(1-piperazinyl)thieno[2,3-D]pyrimidine |
AU2004204825B2 (en) * | 2003-01-13 | 2007-07-19 | Dynogen Pharmaceuticals, Inc. | Method of treating functional bowel disorders |
US20040147510A1 (en) * | 2003-01-13 | 2004-07-29 | Dynogen Pharmaceuticals, Inc. | Method of treating nausea, vomiting, retching or any combination thereof |
EP1795196A3 (en) * | 2003-04-04 | 2008-02-06 | Dynogen Pharmaceuticals, Inc. | Method of treating lower urinary tract disorders |
DE602004007225T2 (de) | 2003-04-04 | 2008-03-06 | Dynogen Pharmaceuticals Inc., Waltham | Methode zur behandlung von erkrankungen der unteren harnwege |
US7643420B2 (en) | 2005-03-11 | 2010-01-05 | Broadcom Corporation | Method and system for transmission control protocol (TCP) traffic smoothing |
US20060293309A1 (en) * | 2005-03-28 | 2006-12-28 | Dynogen Pharmaceuticals, Inc. | Method of treating disorders and conditions using peripherally-restricted antagonists and inhibitors |
FR2895259B1 (fr) * | 2005-12-22 | 2008-02-22 | Urosphere Sas | Methodes de traitement des incontinences urinaires |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2044854A1 (en) * | 1990-07-19 | 1992-01-20 | Hong-I Chen | Method for preventing or treating urinary incontinence |
TW344661B (en) * | 1993-11-24 | 1998-11-11 | Lilly Co Eli | Pharmaceutical composition for treatment of incontinence |
-
2002
- 2002-01-31 GB GBGB0202265.5A patent/GB0202265D0/en not_active Ceased
-
2003
- 2003-01-29 KR KR10-2004-7011877A patent/KR20040081479A/ko not_active Application Discontinuation
- 2003-01-29 CA CA002474851A patent/CA2474851A1/en not_active Abandoned
- 2003-01-29 US US10/502,827 patent/US7220748B2/en not_active Expired - Fee Related
- 2003-01-29 AT AT03702713T patent/ATE397448T1/de not_active IP Right Cessation
- 2003-01-29 AU AU2003205836A patent/AU2003205836B2/en not_active Ceased
- 2003-01-29 EP EP03702713A patent/EP1469853B1/en not_active Expired - Lifetime
- 2003-01-29 DE DE60321445T patent/DE60321445D1/de not_active Expired - Fee Related
- 2003-01-29 PT PT03702713T patent/PT1469853E/pt unknown
- 2003-01-29 JP JP2003563563A patent/JP2005516977A/ja active Pending
- 2003-01-29 WO PCT/GB2003/000374 patent/WO2003063873A1/en active IP Right Grant
- 2003-01-29 CN CNB038030462A patent/CN1279915C/zh not_active Expired - Fee Related
- 2003-01-29 BR BR0307369-6A patent/BR0307369A/pt not_active IP Right Cessation
- 2003-01-29 ES ES03702713T patent/ES2307896T3/es not_active Expired - Lifetime
Also Published As
Publication number | Publication date |
---|---|
ATE397448T1 (de) | 2008-06-15 |
CA2474851A1 (en) | 2003-08-07 |
DE60321445D1 (de) | 2008-07-17 |
ES2307896T3 (es) | 2008-12-01 |
EP1469853A1 (en) | 2004-10-27 |
WO2003063873A1 (en) | 2003-08-07 |
EP1469853B1 (en) | 2008-06-04 |
US20050222162A1 (en) | 2005-10-06 |
CN1625402A (zh) | 2005-06-08 |
US7220748B2 (en) | 2007-05-22 |
PT1469853E (pt) | 2008-06-24 |
KR20040081479A (ko) | 2004-09-21 |
AU2003205836B2 (en) | 2006-06-29 |
GB0202265D0 (en) | 2002-03-20 |
CN1279915C (zh) | 2006-10-18 |
JP2005516977A (ja) | 2005-06-09 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
EA200500721A1 (ru) | Пиримидины, ингибирующие chk, pdk и акт, их получение и применение в качестве лекарственных средств | |
NO20031852D0 (no) | Pyrimidin-2,4,6-trion metalloproteinase inhibitorer | |
BRPI0516242A (pt) | compostos tieno-pirimidina tendo atividade fungicida | |
MA26881A1 (fr) | 5-alkyl-pyrido [2,3-d]pyrimidines inhibitrices de tyrosine-kinases. | |
EA200601659A1 (ru) | Замещенные 4-(4-трифторметилпиразолил)пиримидины, используемые в качестве гербицидов | |
IS2399B (is) | Aðferðir til að framleiða 2-(N-metýl-N-metansúlfónýlamínó)pýrimidín, hýdroxýpýrimidín, halógenpýrimidín eða lífrænar súlfónýloxýpýrimidín afleiður ogefnasambönd sem fást með þeim | |
FR12C0036I2 (fr) | Derives de pyrimidines inhibiteurs de vih | |
AU2003248978A1 (en) | Fused heteroaryl derivatives for use as p38 kinase inhibitors in the treatment of i.a. rheumatoid arthristis | |
ATE362474T1 (de) | Pyrazolo(1,5-a)pyrimidine als hemmstoffe cyclin- abhängiger kinasen | |
ATE388713T1 (de) | 4-amino-6-phenyl-pyrrolo(2,3-d)pyrimidin derivate | |
SG167664A1 (en) | 2,4-pyrimidinediamine compounds and their uses | |
ATE506353T1 (de) | Die hiv-replikation inhibierende indan- substituierte pyrimidine | |
DE60112974D1 (en) | Carbolinderivate | |
ATE244719T1 (de) | N-7 heterocyclyl-pyrrolo( 2,3-d)pyrimidine und ihre verwendung | |
ATE260917T1 (de) | N-(5,7-dimethoxy(1,2,4)triazolo(1,5-a)pyrimidin 2-yl)arylsulfonamid verbindungen und deren verwendung als herbizide | |
DE60336267D1 (de) | Uracilderivate mit herbizider wirkung | |
DE60216233D1 (en) | Carbolinderivate | |
ATE359079T1 (de) | Verfahren zur behandlung von übelkeit, erbrechen, würgereiz oder jede kombination daraus | |
IS6868A (is) | Ný pýrimidínefnasambönd | |
ATE359791T1 (de) | Pyrimidin-2,4-dion-derivate als matrix- metalloproteinase-hemmer | |
BR0307369A (pt) | Uso de 4-(2-fluoro-fenil)-6-metil-2-(1-piperazinil)-tieno (2,3-d)-pirimidina para o tratamento de incontinência urinária | |
DE60112306D1 (de) | Kondensierte pyrazindionderivate als pde5 inhibitore | |
DE60112960D1 (de) | Kondensierte pyridoindolderivate | |
MXPA02012470A (es) | Inhibidores de fosfodiesterasa especificos para gmp ciclico. | |
SE0301654D0 (sv) | Novel compounds |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 8A E 9A ANUIDADE(S). |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: NAO APRESENTADA A GUIA DE CUMPRIMENTO DE EXIGENCIA. REFERENTE AS 8A E 9A ANUIDADES. |