BR0014117A - Uso de sabÈes de acido graxo/aminoácido para aumentar a eficácia antimicrobiana de composições farmacêutica tópicas - Google Patents

Uso de sabÈes de acido graxo/aminoácido para aumentar a eficácia antimicrobiana de composições farmacêutica tópicas

Info

Publication number
BR0014117A
BR0014117A BR0014117-8A BR0014117A BR0014117A BR 0014117 A BR0014117 A BR 0014117A BR 0014117 A BR0014117 A BR 0014117A BR 0014117 A BR0014117 A BR 0014117A
Authority
BR
Brazil
Prior art keywords
pharmaceutical compositions
increase
amino acid
fatty acid
topical pharmaceutical
Prior art date
Application number
BR0014117-8A
Other languages
English (en)
Inventor
Ernesto J Castillo
Steven Howard Gerson
Wesley Wehsin Han
Original Assignee
Alcon Lab Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Alcon Lab Inc filed Critical Alcon Lab Inc
Publication of BR0014117A publication Critical patent/BR0014117A/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0048Eye, e.g. artificial tears
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/16Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
    • A61K47/18Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
    • A61K47/183Amino acids, e.g. glycine, EDTA or aspartame
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0014Skin, i.e. galenical aspects of topical compositions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/02Local antiseptics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Engineering & Computer Science (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Ophthalmology & Optometry (AREA)
  • Dermatology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Patente de Invenção: "USO DE SABõES DE áCIDO GRAXO/AMINOáCIDO PARA AUMENTAR A EFICáCIA ANTIMICROBIANA DE COMPOSIçõES FARMACêUTICA TóPICAS". Sabões de ácido graxo/aminoácido são usados para aumentar a eficácia antimicrobiana em composições farmacêuticas topicamente administráveis contendo pelo menos um ingrediente ativo, um conservante aniónico e um polieletrólito aniónico, tal como polímero de carboxivinila, goma de xantano, polímero de ácido poliestireno sulfónico e resina de troca catiónica.
BR0014117-8A 1999-09-21 2000-09-11 Uso de sabÈes de acido graxo/aminoácido para aumentar a eficácia antimicrobiana de composições farmacêutica tópicas BR0014117A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US39901399A 1999-09-21 1999-09-21
PCT/US2000/024765 WO2001021209A1 (en) 1999-09-21 2000-09-11 Use of fatty acid/amino acid soaps to enhance antimicrobial effectiveness of topical pharmaceutical compositions

Publications (1)

Publication Number Publication Date
BR0014117A true BR0014117A (pt) 2002-05-14

Family

ID=23577764

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0014117-8A BR0014117A (pt) 1999-09-21 2000-09-11 Uso de sabÈes de acido graxo/aminoácido para aumentar a eficácia antimicrobiana de composições farmacêutica tópicas

Country Status (10)

Country Link
EP (1) EP1214094A1 (pt)
JP (1) JP2003509474A (pt)
CN (1) CN1374874A (pt)
AR (1) AR025713A1 (pt)
AU (1) AU7363700A (pt)
BR (1) BR0014117A (pt)
CA (1) CA2391976A1 (pt)
PL (1) PL354365A1 (pt)
TR (1) TR200200724T2 (pt)
WO (1) WO2001021209A1 (pt)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6444710B1 (en) 1998-10-27 2002-09-03 Alcon Manufacturing, Ltd. Use of certain fatty acid/amino acid soaps to enhance antimicrobial effectiveness of topically administrable pharmaceutical compositions
TWI231759B (en) 2001-06-27 2005-05-01 Alcon Inc Olopatadine formulations for topical administration
US7977376B2 (en) 2001-06-27 2011-07-12 Novartis Ag Olopatadine formulations for topical nasal administration
FR2837710B1 (fr) * 2002-03-26 2005-07-08 Innovations Pharma Ag Composition topique a base de resines echangeuses d'ions, notamment pour le traitement des erythemes
US10918618B2 (en) * 2005-03-10 2021-02-16 3M Innovative Properties Company Methods of reducing microbial contamination
US20130149394A1 (en) * 2010-08-27 2013-06-13 Wakamoto Pharmaceutical Co., Ltd. Aqueous ophthalmic composition

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4209722C3 (de) * 1992-03-25 1997-06-19 Medproject Pharma Entwicklungs Tropfbares Gel für die Augenheilkunde
US5520920A (en) * 1992-08-28 1996-05-28 Alcon Laboratories, Inc. Use of certain anionic surfactants to enhance antimicrobial effectiveness of ophthalmic compositions
US5504113A (en) * 1994-03-02 1996-04-02 Allergan, Inc. Enhancement of benzalkonium chloride preservative activity in formulations containing an incompatible drug
JPH0977725A (ja) * 1995-09-13 1997-03-25 Ajinomoto Co Inc 脂肪酸リジン塩の製造方法
WO2000024375A1 (en) * 1998-10-27 2000-05-04 Alcon Laboratories, Inc. Preservative system for topically administrable pharmaceutical compositions containing a fatty acid/amino acid soap

Also Published As

Publication number Publication date
AR025713A1 (es) 2002-12-11
WO2001021209A1 (en) 2001-03-29
CN1374874A (zh) 2002-10-16
JP2003509474A (ja) 2003-03-11
CA2391976A1 (en) 2001-03-29
PL354365A1 (en) 2004-01-12
EP1214094A1 (en) 2002-06-19
AU7363700A (en) 2001-04-24
TR200200724T2 (tr) 2002-06-21

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Legal Events

Date Code Title Description
B11A Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing
B11Y Definitive dismissal acc. article 33 of ipl - extension of time limit for request of examination expired