BR0009014A - Novo intermediário para a sìntese de prostaglandinas - Google Patents

Novo intermediário para a sìntese de prostaglandinas

Info

Publication number
BR0009014A
BR0009014A BR0009014-0A BR0009014A BR0009014A BR 0009014 A BR0009014 A BR 0009014A BR 0009014 A BR0009014 A BR 0009014A BR 0009014 A BR0009014 A BR 0009014A
Authority
BR
Brazil
Prior art keywords
synthesis
new intermediate
prostaglandins
compound
prostaglandines
Prior art date
Application number
BR0009014-0A
Other languages
English (en)
Other versions
BR0009014B1 (pt
Inventor
Philip Mark Jackson
Ian Campbell Lennon
Original Assignee
Chirotech Technology Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chirotech Technology Ltd filed Critical Chirotech Technology Ltd
Publication of BR0009014A publication Critical patent/BR0009014A/pt
Publication of BR0009014B1 publication Critical patent/BR0009014B1/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C405/00—Compounds containing a five-membered ring having two side-chains in ortho position to each other, and having oxygen atoms directly attached to the ring in ortho position to one of the side-chains, one side-chain containing, not directly attached to the ring, a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, and the other side-chain having oxygen atoms attached in gamma-position to the ring, e.g. prostaglandins ; Analogues or derivatives thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1804—Compounds having Si-O-C linkages

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Patente de Invenção: "NOVO INTERMEDIáRIO PARA A SìNTESE DE PROSTAGLANDINAS". Um composto enanciomericamente enriquecido da fórmula 1, na qual Ar é fenila opcionalmente substituída com um ou mais grupos selecionados a partir de haloalquila, alquila e halogeneto. Esse composto pode ser isolado em forma cristalina, e usado na preparação de éster de isopropila de (+) - 16 - [3 - (trifluoro - metil) fenóxi] - 17,18,19,20 tetranor PGF~ 2<244>~.
BRPI0009014-0A 1999-04-12 2000-04-11 composto enanciomericamente enriquecido, processo para preparar um composto enantiomericamente enriquiecido e uso de um composto enantiomericamente enriquecido. BR0009014B1 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB9908326.3 1999-04-12
GBGB9908326.3A GB9908326D0 (en) 1999-04-12 1999-04-12 Novel process intermediate for the synthesis of prostaglandins
PCT/GB2000/001375 WO2000061588A1 (en) 1999-04-12 2000-04-11 Novel intermediate for the synthesis of prostaglandins

Publications (2)

Publication Number Publication Date
BR0009014A true BR0009014A (pt) 2002-03-12
BR0009014B1 BR0009014B1 (pt) 2011-08-09

Family

ID=10851379

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0009014-0A BR0009014B1 (pt) 1999-04-12 2000-04-11 composto enanciomericamente enriquecido, processo para preparar um composto enantiomericamente enriquiecido e uso de um composto enantiomericamente enriquecido.

Country Status (18)

Country Link
EP (1) EP1169325B1 (pt)
JP (1) JP4510300B2 (pt)
CN (1) CN1161362C (pt)
AT (1) ATE240962T1 (pt)
AU (1) AU3980700A (pt)
BR (1) BR0009014B1 (pt)
CA (1) CA2362132C (pt)
CZ (1) CZ20013261A3 (pt)
DE (1) DE60002852T2 (pt)
DK (1) DK1169325T3 (pt)
ES (1) ES2199158T3 (pt)
GB (1) GB9908326D0 (pt)
HU (1) HU230157B1 (pt)
IL (2) IL145076A0 (pt)
MX (1) MXPA01010263A (pt)
PL (1) PL192386B1 (pt)
WO (1) WO2000061588A1 (pt)
ZA (1) ZA200106938B (pt)

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5510383A (en) * 1993-08-03 1996-04-23 Alcon Laboratories, Inc. Use of cloprostenol, fluprostenol and their salts and esters to treat glaucoma and ocular hypertension

Also Published As

Publication number Publication date
ES2199158T3 (es) 2004-02-16
DK1169325T3 (da) 2003-09-08
EP1169325B1 (en) 2003-05-21
CZ20013261A3 (cs) 2002-01-16
PL192386B1 (pl) 2006-10-31
PL351189A1 (en) 2003-03-24
ZA200106938B (en) 2002-08-22
BR0009014B1 (pt) 2011-08-09
CA2362132C (en) 2011-01-04
CA2362132A1 (en) 2000-10-19
GB9908326D0 (en) 1999-06-09
DE60002852D1 (de) 2003-06-26
HUP0200746A3 (en) 2004-07-28
IL145076A0 (en) 2002-06-30
CN1161362C (zh) 2004-08-11
MXPA01010263A (es) 2002-09-18
WO2000061588A1 (en) 2000-10-19
JP4510300B2 (ja) 2010-07-21
WO2000061588A8 (en) 2001-03-08
HUP0200746A2 (hu) 2002-07-29
DE60002852T2 (de) 2004-02-26
CN1345323A (zh) 2002-04-17
AU3980700A (en) 2000-11-14
IL145076A (en) 2006-06-11
JP2002541261A (ja) 2002-12-03
EP1169325A1 (en) 2002-01-09
ATE240962T1 (de) 2003-06-15
HU230157B1 (hu) 2015-09-28

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Legal Events

Date Code Title Description
B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

Free format text: PRAZO DE VALIDADE: 10 (DEZ) ANOS CONTADOS A PARTIR DE 09/08/2011, OBSERVADAS AS CONDICOES LEGAIS.

B21F Lapse acc. art. 78, item iv - on non-payment of the annual fees in time

Free format text: REFERENTE AO NAO RECOLHIMENTO DA 10A ANUIDADE.

B24D Patent annual fee: restoration after fee payment
B21F Lapse acc. art. 78, item iv - on non-payment of the annual fees in time
B24J Lapse because of non-payment of annual fees (definitively: art 78 iv lpi, resolution 113/2013 art. 12)