BR0008872A - Processo para a produção de formas de dosagem sólidas, e, forma de dosagem sólida - Google Patents

Processo para a produção de formas de dosagem sólidas, e, forma de dosagem sólida

Info

Publication number
BR0008872A
BR0008872A BR0008872-2A BR0008872A BR0008872A BR 0008872 A BR0008872 A BR 0008872A BR 0008872 A BR0008872 A BR 0008872A BR 0008872 A BR0008872 A BR 0008872A
Authority
BR
Brazil
Prior art keywords
solid dosage
dosage forms
production
dosage form
components
Prior art date
Application number
BR0008872-2A
Other languages
English (en)
Other versions
BR0008872B1 (pt
Inventor
Gunther Berndl
Ulrich Reinhold
Dirk Simon
Stephan Lehmann
Original Assignee
Basf Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Ag filed Critical Basf Ag
Publication of BR0008872A publication Critical patent/BR0008872A/pt
Publication of BR0008872B1 publication Critical patent/BR0008872B1/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/192—Carboxylic acids, e.g. valproic acid having aromatic groups, e.g. sulindac, 2-aryl-propionic acids, ethacrynic acid 
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N25/00—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
    • A01N25/08—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests containing solids as carriers or diluents
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N25/00—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
    • A01N25/08—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests containing solids as carriers or diluents
    • A01N25/10—Macromolecular compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/02—Cosmetics or similar toiletry preparations characterised by special physical form
    • A61K8/0216—Solid or semisolid forms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/72—Cosmetics or similar toiletry preparations characterised by the composition containing organic macromolecular compounds
    • A61K8/73—Polysaccharides
    • A61K8/738—Cyclodextrins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/72—Cosmetics or similar toiletry preparations characterised by the composition containing organic macromolecular compounds
    • A61K8/84—Cosmetics or similar toiletry preparations characterised by the composition containing organic macromolecular compounds obtained by reactions otherwise than those involving only carbon-carbon unsaturated bonds
    • A61K8/86—Polyethers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2031—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2095—Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q19/00—Preparations for care of the skin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2800/00—Properties of cosmetic compositions or active ingredients thereof or formulation aids used therein and process related aspects
    • A61K2800/40—Chemical, physico-chemical or functional or structural properties of particular ingredients
    • A61K2800/56—Compounds, absorbed onto or entrapped into a solid carrier, e.g. encapsulated perfumes, inclusion compounds, sustained release forms

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Birds (AREA)
  • Plant Pathology (AREA)
  • Environmental Sciences (AREA)
  • Toxicology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Dermatology (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)

Abstract

"PROCESSO PARA A PRODUçãO DE FORMAS DE DOSAGEM SóLIDAS, E, FORMA DE DOSAGEM SóLIDA". A presente invenção refere-se a um processo para a produção de formas de dosagern sólidas, que compreende, como componentes, pelo menos um aglutinante polimérico fisiologicamente tolerado, pelo menos um ingrediente ativo e pelo menos uma ciclodextrina, em que os componentes são misturados e plastificados em uma temperatura abaixo de 220<198>C, sem adição de um solvente, e a mistura plástica resultante é moldada na forma de dosagem, e as formas de dosagem são obteníveis por este processo.
BRPI0008872-2A 1999-03-12 2000-03-10 processo para a produção de formas de dosagem sólidas, e, forma de dosagem sólida. BR0008872B1 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19911097A DE19911097A1 (de) 1999-03-12 1999-03-12 Verfahren zur Herstellung von festen cyclodextrinhaltigen Dosierungsformen
PCT/EP2000/002142 WO2000054751A1 (de) 1999-03-12 2000-03-10 Verfahren zur herstellung von festen cyclodextrinhaltigen dosierungsformen

Publications (2)

Publication Number Publication Date
BR0008872A true BR0008872A (pt) 2002-01-02
BR0008872B1 BR0008872B1 (pt) 2011-05-17

Family

ID=7900771

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0008872-2A BR0008872B1 (pt) 1999-03-12 2000-03-10 processo para a produção de formas de dosagem sólidas, e, forma de dosagem sólida.

Country Status (10)

Country Link
EP (1) EP1158962B1 (pt)
JP (1) JP4861552B2 (pt)
AT (1) ATE228828T1 (pt)
BR (1) BR0008872B1 (pt)
CA (1) CA2367020C (pt)
DE (2) DE19911097A1 (pt)
DK (1) DK1158962T3 (pt)
ES (1) ES2187457T3 (pt)
PT (1) PT1158962E (pt)
WO (1) WO2000054751A1 (pt)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1175205B1 (en) 1999-11-12 2006-06-14 Abbott Laboratories Solid dispersion comprising ritonavir, fenofibrate or griseofulvin
SI1278549T1 (sl) 2000-05-02 2009-04-30 Theravance Inc Sestavek, ki vsebuje ciklodekstrin in glikopeptidni antibiotik
AU2001259298A1 (en) 2000-05-02 2001-11-12 Advanced Medicine, Inc. Polyacid glycopeptide derivatives
DE10026698A1 (de) 2000-05-30 2001-12-06 Basf Ag Selbstemulgierende Wirkstoffformulierung und Verwendung dieser Formulierung
US6828299B2 (en) 2000-06-22 2004-12-07 Theravance, Inc. Polyhydroxy glycopeptide derivatives
US6872804B2 (en) 2000-06-22 2005-03-29 Theravance, Inc. Glycopeptide disulfide and thioester derivatives
ES2302733T3 (es) 2000-06-22 2008-08-01 Theravance, Inc. Derivados carboxi-sacaridos de glucopeptido.
UA75083C2 (uk) 2000-06-22 2006-03-15 Тераванс, Інк. Похідні глікопептидфосфонатів
FR2828380B1 (fr) * 2001-08-10 2005-07-29 Fontarome Composition a structure composite contenant des substances aromatiques et/ou des substances non aromatiques volatiles et/ou sensibles aux agents exterieurs, et son procede de fabrication
DE10141682A1 (de) * 2001-08-25 2003-03-06 Beiersdorf Ag Verwendung von Cyclodextrinen zur Herstellung kosmetischer und dermatologischer Zubereitungen mit verbesserter Verteilbarkeit von Füllstoffen auf der Haut sowie kosmetische und dermatologische Zubereitungen mit einem Gehalt an Cyclodextrinen und Füllstoffen
DE10157350A1 (de) * 2001-11-22 2003-05-28 Stockhausen Chem Fab Gmbh Herstellung von Wirkstoffzusammensetzung durch Extrudieren von wasserabsorbierenden Polymeren
US7001893B2 (en) * 2002-10-28 2006-02-21 Council Of Scientific And Industrial Research Inclusion complex of Rifampicin, an anti-tubercular drug, with β-cyclodextrin or 2-hydroxypropyl β-cyclodextrin and a process thereof
US8025899B2 (en) 2003-08-28 2011-09-27 Abbott Laboratories Solid pharmaceutical dosage form
US8377952B2 (en) 2003-08-28 2013-02-19 Abbott Laboratories Solid pharmaceutical dosage formulation
US7955630B2 (en) * 2004-09-30 2011-06-07 Kraft Foods Global Brands Llc Thermally stable, high tensile strength encapsulated actives
ES2310948B2 (es) 2005-02-25 2009-09-16 Universidade De Santiago De Compostela Procedimiento de obtencion de hidrogeles de ciclodextrinas con glicidileteres, las composiciones obtenidas y sus aplicaciones.
CN108883125B (zh) * 2016-02-04 2022-08-09 西泽普研究与发展有限责任公司 受控释放和层状的环糊精包合物媒介物
DE102016014603A1 (de) 2016-06-30 2018-01-04 Thomas Herkenroth Synthetisches Ayahuasca
WO2020213010A1 (en) * 2019-04-16 2020-10-22 Celagenex Research (India) Pvt. Ltd. Synergistic lipid controlling compositions
CN113081989B (zh) * 2021-03-29 2022-10-21 海南普利制药股份有限公司 别嘌醇缓释片剂
CN113861347A (zh) * 2021-11-02 2021-12-31 南京信息工程大学 改性环糊精高分子缓释薄荷香型材料及制备方法和应用
CN114588123B (zh) * 2022-04-13 2023-12-22 苏州中化药品工业有限公司 一种高稳定性盐酸西替利嗪片剂及其制备方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH0624903A (ja) * 1992-04-09 1994-02-01 Nippon Bayeragrochem Kk 植物処理剤
DE4446470A1 (de) * 1994-12-23 1996-06-27 Basf Ag Verfahren zur Herstellung von teilbaren Tabletten
EP0862463A1 (en) * 1995-11-23 1998-09-09 Janssen Pharmaceutica N.V. Solid mixtures of cyclodextrins prepared via melt-extrusion

Also Published As

Publication number Publication date
BR0008872B1 (pt) 2011-05-17
EP1158962A1 (de) 2001-12-05
ATE228828T1 (de) 2002-12-15
DK1158962T3 (da) 2003-01-06
DE19911097A1 (de) 2000-09-14
JP2002539151A (ja) 2002-11-19
PT1158962E (pt) 2003-04-30
CA2367020A1 (en) 2000-09-21
DE50000866D1 (de) 2003-01-16
WO2000054751A1 (de) 2000-09-21
ES2187457T3 (es) 2003-06-16
CA2367020C (en) 2008-12-16
EP1158962B1 (de) 2002-12-04
JP4861552B2 (ja) 2012-01-25

Similar Documents

Publication Publication Date Title
BR0008872A (pt) Processo para a produção de formas de dosagem sólidas, e, forma de dosagem sólida
WO2004078797A8 (en) Macromolecular ketoaldehydes
WO1998010752A3 (de) Verfahren zur herstellung fester pharmazeutischer formen durch extrudierung
EP1726299A3 (en) Cores and microcapsules suitable for parenteral administration as well as process for their manufacture
BRPI0414600A (pt) composição de elastÈmero termoplástico contendo microgel
ATE410400T1 (de) Verfahren zur herstellung von c13- alkoholgemischen
WO2005090460A8 (en) Composite materials comprising ppta and nanotubes
ATE487740T1 (de) Polyrotaxan und herstellungsverfahren dafür
ID27377A (id) Bentuk baru dari irbesartan, proses pembuatannya dan komposisi farmasi yang mengandung irbesartan tersebut
ATE407664T1 (de) Hydrogel zusammensetzungen, geeignet zur verzögerten freisetzung von makromolekülen sowie verfahren zur herstellung derselben.
ATE315596T1 (de) Verfahren zur herstellung kautschukhaltiger thermoplastischer formmassen
DE60117651D1 (de) Bioabbaubare Zusammensetzung und Verfahren zur deren Herstellung
ATE369959T1 (de) Verfahren zur herstellung von verbindungssystemen und nach diesem verfahren hergestellte verbindungssysteme
BRPI0416672A (pt) método de produção de uma composição granular contendo lecitina e composição granular contendo lecitina
ATE387089T1 (de) Granulatförmige zusammensetzungen und verfahren zu ihrer herstellung
BRPI0513881A (pt) processo para a preparação de compostos opticamente ativos
DE60130575D1 (de) Verfahren zur herstellung von acylphenylalaninen
DE59903189D1 (de) Verfahren zur herstellung von cellulosecarbamat
DE69925992D1 (de) VERFAHREN ZUR HERSTELLUNG VON 5-HYDROXYBENZO[b]THIOPHEN-3-CARBONSÄURE
ATE274896T1 (de) Verfahren zur herstellung von festen dosierungsformen
WO2002072675A3 (en) Predispersions, compositions therefore, and processes for preparing same
DE502004009237D1 (de) Kaumasse zur remineralisation von zahnschmelz
AU2001246900A1 (en) Plastic lens material, production process of the material, composition for plastic lens, plastic lens obtained by curing the composition, and production processof the plastic lens
WO2002048074A1 (fr) Procede de preparation d&#39;un compose moleculaire
WO2004078846A8 (fr) Composition comprenant une matrice et un additif fonctionnalise et articles realises a partir de cette composition

Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 3A ANUIDADE

B08G Application fees: restoration [chapter 8.7 patent gazette]
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

Free format text: PRAZO DE VALIDADE: 10 (DEZ) ANOS CONTADOS A PARTIR DE 17/05/2011, OBSERVADAS AS CONDICOES LEGAIS.

B15K Others concerning applications: alteration of classification

Free format text: PROCEDIMENTO AUTOMATICO DE RECLASSIFICACAO. AS CLASSIFICACOES IPC ANTERIORES ERAM: A61K 9/20; A61K 47/48.

Ipc: A61K 31/192 (2006.01), A01N 25/08 (2006.01), A01N

Ipc: A61K 31/192 (2006.01), A01N 25/08 (2006.01), A01N

B21F Lapse acc. art. 78, item iv - on non-payment of the annual fees in time

Free format text: REFERENTE A 21A ANUIDADE.

B24J Lapse because of non-payment of annual fees (definitively: art 78 iv lpi, resolution 113/2013 art. 12)

Free format text: EM VIRTUDE DA EXTINCAO PUBLICADA NA RPI 2621 DE 30-03-2021 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDA A EXTINCAO DA PATENTE E SEUS CERTIFICADOS, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.