BG102238A - Нови имидазолин-2,4-диони с антиконвулсивно действие, съдържащи в 1-ва позиция един ортозаместен ар(алк)илов радикал, и метод за тяхното получаване - Google Patents
Нови имидазолин-2,4-диони с антиконвулсивно действие, съдържащи в 1-ва позиция един ортозаместен ар(алк)илов радикал, и метод за тяхното получаванеInfo
- Publication number
- BG102238A BG102238A BG102238A BG10223898A BG102238A BG 102238 A BG102238 A BG 102238A BG 102238 A BG102238 A BG 102238A BG 10223898 A BG10223898 A BG 10223898A BG 102238 A BG102238 A BG 102238A
- Authority
- BG
- Bulgaria
- Prior art keywords
- orthosubstituted
- dions
- alk
- radical
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/72—Two oxygen atoms, e.g. hydantoin
- C07D233/74—Two oxygen atoms, e.g. hydantoin with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to other ring members
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
Съединенията проявяват антиконвулсивно действие. Те имат обща формула в която Х означава С1-С4алкил, трифлуорметил и халоген, Y - водород и халоген, n има стойност 0 и 1, а m - 0, 1, 2, 3 и 4.
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19529425A DE19529425A1 (de) | 1995-08-10 | 1995-08-10 | Neue, antikonvulsiv wirkende Imidazolin-2,4-dione, die in 1-Stellung einen orthosubstituierten Ar(alk)yl-Rest enthalten, und Verfahren zu deren Herstellung |
PCT/EP1996/003296 WO1997006149A1 (de) | 1995-08-10 | 1996-07-26 | Neue, antikonvulsiv wirkende imidazolin-2,4-dione, die in 1-stellung einen orthosubstituierten ar(alk)yl-rest enthalten, und verfahren zu deren herstellung |
US08/700,876 US5817685A (en) | 1995-08-10 | 1996-08-21 | Anticonvulsive imidazoline-2,4-diones and process for making |
CA002183928A CA2183928A1 (en) | 1995-08-10 | 1996-08-22 | Anticonvulsive imidazoline-2,4-diones and process for making |
Publications (1)
Publication Number | Publication Date |
---|---|
BG102238A true BG102238A (bg) | 1998-09-30 |
Family
ID=27170189
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BG102238A BG102238A (bg) | 1995-08-10 | 1998-02-09 | Нови имидазолин-2,4-диони с антиконвулсивно действие, съдържащи в 1-ва позиция един ортозаместен ар(алк)илов радикал, и метод за тяхното получаване |
Country Status (14)
Country | Link |
---|---|
US (1) | US5817685A (bg) |
EP (1) | EP0850226A1 (bg) |
CN (1) | CN1192736A (bg) |
AU (1) | AU699802B2 (bg) |
BG (1) | BG102238A (bg) |
CA (1) | CA2183928A1 (bg) |
CZ (1) | CZ38298A3 (bg) |
DE (1) | DE19529425A1 (bg) |
IL (1) | IL123296A0 (bg) |
LT (1) | LT4457B (bg) |
NO (1) | NO980309D0 (bg) |
NZ (1) | NZ315625A (bg) |
PL (1) | PL327452A1 (bg) |
WO (1) | WO1997006149A1 (bg) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2443906A1 (en) * | 2001-04-16 | 2002-10-24 | University Of Virginia Patent Foundation | Novel oral general anesthetics and metabolitically resistant anticonvulsants |
CN101255136B (zh) * | 2008-03-11 | 2011-08-17 | 武汉大学 | 5-环丙烷螺环乙内酰脲衍生物及其制备方法和应用 |
ATE525941T1 (de) * | 2009-10-23 | 2011-10-15 | Gruppo Cimbali Spa | Kaffeemaschine mit abgabedruckregulierung und damit zusammenhängendes verfahren |
CN101863839B (zh) * | 2010-06-04 | 2012-02-15 | 武汉大学 | N-3-芳酰胺-5-环丙烷螺环乙内酰脲衍生物及其制备方法和应用 |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB997037A (en) * | 1962-03-19 | 1965-06-30 | Ici Ltd | New hydrantoin derivatives |
JPH05178802A (ja) * | 1991-12-27 | 1993-07-20 | Sumitomo Seika Chem Co Ltd | N−ベンジルグリシンおよびその誘導体の製造方法 |
TW297813B (bg) * | 1993-09-24 | 1997-02-11 | Takeda Pharm Industry Co Ltd |
-
1995
- 1995-08-10 DE DE19529425A patent/DE19529425A1/de not_active Withdrawn
-
1996
- 1996-07-26 WO PCT/EP1996/003296 patent/WO1997006149A1/de not_active Application Discontinuation
- 1996-07-26 CN CN96196190A patent/CN1192736A/zh active Pending
- 1996-07-26 CZ CZ98382A patent/CZ38298A3/cs unknown
- 1996-07-26 EP EP96927608A patent/EP0850226A1/de not_active Withdrawn
- 1996-07-26 AU AU67376/96A patent/AU699802B2/en not_active Ceased
- 1996-07-26 IL IL12329696A patent/IL123296A0/xx unknown
- 1996-07-26 PL PL96327452A patent/PL327452A1/xx unknown
- 1996-07-26 NZ NZ315625A patent/NZ315625A/xx unknown
- 1996-08-21 US US08/700,876 patent/US5817685A/en not_active Expired - Fee Related
- 1996-08-22 CA CA002183928A patent/CA2183928A1/en not_active Abandoned
-
1998
- 1998-01-23 NO NO980309A patent/NO980309D0/no unknown
- 1998-02-09 BG BG102238A patent/BG102238A/bg unknown
- 1998-03-09 LT LT98-030A patent/LT4457B/lt not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
NO980309L (no) | 1998-01-23 |
LT98030A (en) | 1998-09-25 |
WO1997006149A1 (de) | 1997-02-20 |
AU6737696A (en) | 1997-03-05 |
CN1192736A (zh) | 1998-09-09 |
AU699802B2 (en) | 1998-12-17 |
PL327452A1 (en) | 1998-12-07 |
DE19529425A1 (de) | 1997-02-13 |
IL123296A0 (en) | 1998-10-30 |
NO980309D0 (no) | 1998-01-23 |
CZ38298A3 (cs) | 1998-09-16 |
CA2183928A1 (en) | 1998-02-23 |
US5817685A (en) | 1998-10-06 |
EP0850226A1 (de) | 1998-07-01 |
LT4457B (lt) | 1999-02-25 |
NZ315625A (en) | 1999-01-28 |
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