BE905502A - 2-oxo-1- (((sulfonyle substitue) amino) carbonyl) azetidines, leur preparation et leur utilisation. - Google Patents

2-oxo-1- (((sulfonyle substitue) amino) carbonyl) azetidines, leur preparation et leur utilisation.

Info

Publication number
BE905502A
BE905502A BE0/217217A BE217217A BE905502A BE 905502 A BE905502 A BE 905502A BE 0/217217 A BE0/217217 A BE 0/217217A BE 217217 A BE217217 A BE 217217A BE 905502 A BE905502 A BE 905502A
Authority
BE
Belgium
Prior art keywords
preparation
azetidines
oxo
carbonyl
amino
Prior art date
Application number
BE0/217217A
Other languages
English (en)
French (fr)
Original Assignee
Squibb & Sons Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Squibb & Sons Inc filed Critical Squibb & Sons Inc
Publication of BE905502A publication Critical patent/BE905502A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
BE0/217217A 1985-09-26 1986-09-26 2-oxo-1- (((sulfonyle substitue) amino) carbonyl) azetidines, leur preparation et leur utilisation. BE905502A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US78047985A 1985-09-26 1985-09-26

Publications (1)

Publication Number Publication Date
BE905502A true BE905502A (fr) 1987-01-16

Family

ID=25119699

Family Applications (1)

Application Number Title Priority Date Filing Date
BE0/217217A BE905502A (fr) 1985-09-26 1986-09-26 2-oxo-1- (((sulfonyle substitue) amino) carbonyl) azetidines, leur preparation et leur utilisation.

Country Status (31)

Country Link
JP (1) JPS6284082A (https=)
KR (1) KR900001013B1 (https=)
CN (1) CN86106980A (https=)
AT (1) ATA257986A (https=)
AU (1) AU600912B2 (https=)
BE (1) BE905502A (https=)
CA (1) CA1308719C (https=)
CH (1) CH670828A5 (https=)
DD (1) DD250121A5 (https=)
DE (1) DE3632876A1 (https=)
DK (1) DK460386A (https=)
EG (1) EG18314A (https=)
ES (1) ES2001995A6 (https=)
FI (1) FI863890A7 (https=)
FR (1) FR2587700B1 (https=)
GB (1) GB2181130B (https=)
GR (1) GR862449B (https=)
HU (1) HU198044B (https=)
IE (1) IE59686B1 (https=)
IL (1) IL80160A (https=)
IT (1) IT1214533B (https=)
LU (1) LU86611A1 (https=)
NL (1) NL8602446A (https=)
NO (1) NO863837L (https=)
NZ (1) NZ217704A (https=)
PH (1) PH23315A (https=)
PL (1) PL151546B1 (https=)
PT (1) PT83440B (https=)
SE (1) SE8604089L (https=)
YU (1) YU46177B (https=)
ZA (1) ZA867373B (https=)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4975538A (en) * 1987-03-03 1990-12-04 The Upjohn Company Antibiotic sulfonylaminocarbonyl activated beta-lactams
US5001235A (en) * 1987-02-27 1991-03-19 The Upjohn Company Antibiotic beta-lactams containing a pyridone carboxylic acid or acid derivative
US5006650A (en) * 1987-02-11 1991-04-09 The Upjohn Company Novel N-1 substituted beta-lactams as antibiotics
US5015737A (en) * 1987-07-22 1991-05-14 The Upjohn Company Therapeutically useful beta-lactams

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU7541487A (en) * 1986-05-23 1987-12-22 Upjohn Company, The N-1 substituted sulfonylaminocarbonyl, c-4 substituted monobactams
JPH02502378A (ja) * 1987-02-11 1990-08-02 ジ・アップジョン・カンパニー 抗生物質としての新規なN‐1置換β‐ラクタム
US4762922A (en) * 1987-07-01 1988-08-09 Squibb Corporation 2-oxo-1-[[(substituted sulfonyl)amino]-carbonyl]azetidines
US4772693A (en) * 1987-07-01 1988-09-20 E. R. Squibb & Sons, Inc. 2-oxo-1-((Substituted sulfonyl)amino)-carbonyl)azetidines
JPH02504272A (ja) * 1987-07-22 1990-12-06 ジ・アップジョン・カンパニー 治療上有用なβ‐ラクタム類
US4777252A (en) * 1987-08-13 1988-10-11 E. R. Squibb & Sons, Inc. 2-oxo-1-[[(substituted sulfonyl)amino]-carbonyl]azetidines
US4889930A (en) * 1987-12-21 1989-12-26 E. R. Squibb & Sons, Inc. Process for making 2-oxo-1-((substituted sulfonyl)amino)carbonzyl)azetidines and intermediates used therein
US4871841A (en) * 1987-12-23 1989-10-03 E. R. Squibb & Sons, Inc. 2-Oxo-1-[[(substituted sulfonyl)amino]-carbonyl]azetidines
EP0336667A3 (en) * 1988-04-04 1991-04-10 E.R. Squibb & Sons, Inc. [3S(Z)]-3-[[(2-amino-4-thiazolyl)[[2-(hydroxyamino)-2-oxoethoxy]imino]acetyl]-amino]-2,2-dimethyl-4-oxo-1-azetidinyl sulfate
US4959470A (en) * 1988-08-17 1990-09-25 E. R. Squibb & Sons, Inc. 2-oxo-[[(substituted sulfonyl)-amino]carbonyl]-azetidines
EP0604365B1 (en) * 1992-12-23 1999-05-26 Novartis AG Imidazole derivatives and their use as agrochemical agents
EP0671654B1 (en) * 1994-03-11 1997-09-10 Agfa-Gevaert N.V. Photographic material containing a new type of hydrazide
KR100596360B1 (ko) * 2003-07-15 2006-07-03 한국생명공학연구원 항암 활성을 갖는 신규 2-옥소-피페리딘 유도체(ⅰ)화합물을 포함하는 암 질환 치료를 위한 약학 조성물
WO2005063704A1 (ja) * 2003-12-25 2005-07-14 Ono Pharmaceutical Co., Ltd. アゼチジン環化合物およびその医薬
GB201111704D0 (en) 2011-07-07 2011-08-24 Takeda Pharmaceutical Novel compounds
GB201111705D0 (en) 2011-07-07 2011-08-24 Takeda Pharmaceutical Compounds and their use
JO3115B1 (ar) 2011-08-22 2017-09-20 Takeda Pharmaceuticals Co مركبات بيريدازينون واستخدامها كمثبطات daao
UA111861C2 (uk) 2011-11-15 2016-06-24 Такеда Фармасьютікал Компані Лімітед Ароматична гетероциклічна сполука дигідрокси
GB201222711D0 (en) 2012-12-17 2013-01-30 Takeda Pharmaceutical Novel compounds
CN106986820B (zh) * 2017-02-24 2019-05-21 浙江工商大学 多功能的羟基吡啶酮衍生物及其水合物的制备法和用途

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ199981A (en) * 1981-04-09 1985-08-16 Squibb & Sons Inc 2-oxo-1-(((substituted sulphonyl)amino)carbonyl)azetidines
CA1272726C (en) * 1982-01-04 1990-08-14 2-oxo-1-(aminocarbonylaminosulfonyl- aminocarbonyl)azetidines
US4939253A (en) * 1982-08-04 1990-07-03 E. R. Squibb & Sons, Inc. 2-oxoazetidin-1-yloxy acetic acids and analogs
US4801705A (en) * 1986-06-23 1989-01-31 E. R. Squibb & Sons, Inc. 2-oxo-1-(((substituted sulfonyl)amino)-carbonyl)azetidines

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5006650A (en) * 1987-02-11 1991-04-09 The Upjohn Company Novel N-1 substituted beta-lactams as antibiotics
US5001235A (en) * 1987-02-27 1991-03-19 The Upjohn Company Antibiotic beta-lactams containing a pyridone carboxylic acid or acid derivative
US4975538A (en) * 1987-03-03 1990-12-04 The Upjohn Company Antibiotic sulfonylaminocarbonyl activated beta-lactams
US5015737A (en) * 1987-07-22 1991-05-14 The Upjohn Company Therapeutically useful beta-lactams

Also Published As

Publication number Publication date
SE8604089D0 (sv) 1986-09-26
IL80160A0 (en) 1986-12-31
ZA867373B (en) 1987-05-27
IE59686B1 (en) 1994-03-23
CA1308719C (en) 1992-10-13
GR862449B (en) 1987-01-27
GB2181130B (en) 1989-09-20
GB2181130A (en) 1987-04-15
IL80160A (en) 1991-04-15
EG18314A (en) 1993-02-28
AU600912B2 (en) 1990-08-30
KR900001013B1 (ko) 1990-02-24
CH670828A5 (https=) 1989-07-14
ATA257986A (de) 1994-07-15
ES2001995A6 (es) 1988-07-01
DK460386A (da) 1987-03-27
DK460386D0 (da) 1986-09-26
PH23315A (en) 1989-07-14
PT83440B (pt) 1989-05-12
AU6315686A (en) 1987-04-02
GB8623151D0 (en) 1986-10-29
PL151546B1 (en) 1990-09-28
YU46177B (sh) 1993-05-28
YU165986A (en) 1988-06-30
FR2587700B1 (fr) 1988-09-16
HUT44535A (en) 1988-03-28
IT8621834A0 (it) 1986-09-26
NL8602446A (nl) 1987-04-16
NO863837L (no) 1987-03-27
SE8604089L (sv) 1987-03-27
CN86106980A (zh) 1987-04-08
FI863890A0 (fi) 1986-09-26
LU86611A1 (fr) 1987-04-02
DD250121A5 (de) 1987-09-30
JPS6284082A (ja) 1987-04-17
IE862547L (en) 1987-03-26
KR870003101A (ko) 1987-04-15
PT83440A (pt) 1986-10-01
NO863837D0 (no) 1986-09-26
DE3632876A1 (de) 1987-04-02
PL261575A1 (en) 1988-07-21
FR2587700A1 (fr) 1987-03-27
NZ217704A (en) 1989-02-24
IT1214533B (it) 1990-01-18
FI863890A7 (fi) 1987-03-27
HU198044B (en) 1989-07-28

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: E.R. SQUIBB & SONS, INC.

Effective date: 20000930