BE905113A - NOVEL DERIVATIVES OF CEPH-3-EM-4-CARBOXYLIC ACIDS, THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM. - Google Patents

NOVEL DERIVATIVES OF CEPH-3-EM-4-CARBOXYLIC ACIDS, THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM.

Info

Publication number
BE905113A
BE905113A BE0/216927A BE216927A BE905113A BE 905113 A BE905113 A BE 905113A BE 0/216927 A BE0/216927 A BE 0/216927A BE 216927 A BE216927 A BE 216927A BE 905113 A BE905113 A BE 905113A
Authority
BE
Belgium
Prior art keywords
ceph
preparation
carboxylic acids
medicaments containing
novel derivatives
Prior art date
Application number
BE0/216927A
Other languages
French (fr)
Original Assignee
Biogal Gyogyszergyar
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Biogal Gyogyszergyar filed Critical Biogal Gyogyszergyar
Publication of BE905113A publication Critical patent/BE905113A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/36—Methylene radicals, substituted by sulfur atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/545—Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D257/00—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms
    • C07D257/02—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D257/04—Five-membered rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Ces dérivés sont l'acide 7- (3-chloro-isoxazol-5-yl) -acétamido-3- (1-méthyl-ceph-3-em-4-carboxylique) de formule et ses sels convenant en pharmacologie ; des médicaments présentant notamment une grande activité contre un spectre étendu de micro-organismes et des procédés pour préparer ces dérivés et médicaments sont également décrits.These derivatives are 7- (3-chloro-isoxazol-5-yl) -acetamido-3- (1-methyl-ceph-3-em-4-carboxylic acid) of formula and its salts suitable in pharmacology; drugs particularly exhibiting great activity against a broad spectrum of microorganisms and methods for preparing these derivatives and drugs are also described.

BE0/216927A 1985-07-16 1986-07-15 NOVEL DERIVATIVES OF CEPH-3-EM-4-CARBOXYLIC ACIDS, THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM. BE905113A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU852725A HU203243B (en) 1985-07-16 1985-07-16 Process for producing cefalosporin derivative

Publications (1)

Publication Number Publication Date
BE905113A true BE905113A (en) 1986-11-03

Family

ID=10960853

Family Applications (1)

Application Number Title Priority Date Filing Date
BE0/216927A BE905113A (en) 1985-07-16 1986-07-15 NOVEL DERIVATIVES OF CEPH-3-EM-4-CARBOXYLIC ACIDS, THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM.

Country Status (14)

Country Link
JP (1) JPS6222787A (en)
KR (1) KR930007263B1 (en)
CN (1) CN1012614B (en)
AT (1) AT389877B (en)
BE (1) BE905113A (en)
DE (1) DE3623900A1 (en)
FI (1) FI83877C (en)
FR (1) FR2591598B1 (en)
GB (1) GB2177696B (en)
GR (1) GR861855B (en)
HU (1) HU203243B (en)
IL (1) IL79410A0 (en)
IT (1) IT1196494B (en)
NL (1) NL8601842A (en)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2012729C (en) 1989-04-07 1997-05-20 Takashi Kuroda Dulled stretched molding and process for producing the same
JP2893286B2 (en) * 1990-05-17 1999-05-17 グンゼ株式会社 Heat-shrinkable foamed composite film and method for producing the same
JP2515295Y2 (en) * 1993-06-30 1996-10-30 株式会社川崎製作所 Pipe fitting
KR100408343B1 (en) * 2001-11-01 2003-12-06 주식회사 이앤티 Feed and manufacturing method for maintaining homeostasis of piglets

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2409949A1 (en) * 1973-03-02 1974-09-05 Gist Brocades Nv PENICILLANIC ACID AND CEPHALOSPORIC ACID DERIVATIVES, PROCESS FOR THEIR PRODUCTION AND ANTIBACTERICIDAL PREPARATIONS CONTAINING THESE COMPOUNDS
JPS539787A (en) * 1976-07-16 1978-01-28 Yamanouchi Pharmaceut Co Ltd Novel cephalosporin derivatives and their preparation

Also Published As

Publication number Publication date
FI862965A0 (en) 1986-07-16
FI862965A (en) 1987-01-17
HUT48890A (en) 1989-07-28
IT1196494B (en) 1988-11-16
DE3623900A1 (en) 1987-01-29
FR2591598A1 (en) 1987-06-19
JPS6222787A (en) 1987-01-30
GB2177696B (en) 1989-01-05
IT8621135A0 (en) 1986-07-15
HU203243B (en) 1991-06-28
FI83877B (en) 1991-05-31
KR930007263B1 (en) 1993-08-04
GB2177696A (en) 1987-01-28
CN86104805A (en) 1987-02-18
IL79410A0 (en) 1986-10-31
FI83877C (en) 1991-09-10
GR861855B (en) 1986-11-18
NL8601842A (en) 1987-02-16
ATA192686A (en) 1989-07-15
AT389877B (en) 1990-02-12
FR2591598B1 (en) 1990-01-26
GB8617181D0 (en) 1986-08-20
KR870001219A (en) 1987-03-12
CN1012614B (en) 1991-05-15

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: BIOGAL GYOGYSZERGYAR

Effective date: 19960731